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Effect of Antifibrotic Therapy on Regression of Myocardial Fibrosis After Transcatheter Aortic Valve Implantation (TAVI) in Aortic Stenosis Patients With High Fibrotic Burden

Phase 3
Recruiting
Conditions
Aortic Stenosis, Severe
Interventions
Registration Number
NCT05230901
Lead Sponsor
University Medical Center Goettingen
Brief Summary

The aim of the study is to evaluate the effect of antifibrotic therapy on regression of myocardial fibrosis after TAVI in patients with baseline high fibrotic burden. Therefore, patients will be treated with Spironolactone in addition to standard of care, Spioronolactone + Dihydralazine in addition to standard of care or according to standard of care alone without any study medication. First, differences between patients in the control arm and patients randomized to anti-fibrotic therapy will be analyzed. The second analysis will determine, whether dihydralazine medication in addition to spironolactone is able to increase a potential antifibrotic effect. Myocardial fibrosis will be assessed by cardiac magnetic resonance imaging (CMR) before TAVI and 1 year after. Quantification of potentially irreversible replacement fibrosis will be carried out by late gadolinium enhancement (LGE), and quantification of the potentially reversible diffuse interstitial fibrosis will be performed by measurement of the extracellular volume fraction (ECV), thereby deriving matrix volume and cell volume.

Detailed Description

Not available

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
300
Inclusion Criteria
  • Male, female age ≥ 60
  • Diagnosis of severe symptomatic aortic stenosis
  • Transcatheter aortic valve implantation (TAVI) scheduled
  • Written informed consent
Exclusion Criteria
    1. Pre-existing dilative or ischemic heart disease with EF<35% and guideline indication for spironolactone
  • Patient on current medication with spironolactone, eplerenone, or dihydralazine
  • Presence of coexistent myocardial pathology such as cardiac amyloidosis, hypertrophic cardiomyopathy, or myocarditis
  • Presence of coexistent severe aortic regurgitation or severe mitral stenosis
  • Previous surgical valve replacement or repair
  • Pacemaker or ICD implanted
  • Renal impairment (serum creatinine > 1,8 mg/dl and/ or GFR < 30 ml/min/1,73 m² BSA)
  • Significant hypotension (blood pressure < 90 mm Hg systolic and/or < 50 mm Hg diastolic
  • Serum potassium > 5,1 mmol/l
  • Contraindications for Spironolactone (anuria, acute renal failure, serum creatinine > 1.8 mg/dl, hyperkalemia, pregnancy)
  • Contraindications for Dihydralazine (known allergy or hypersensitivity, systemic lupus erythematodes, adrenocortical disorders)
  • Known active malignant disease with life expectancy < 1 year
  • Women with child-bearing potential
  • Simultaneous participation (including a waiting period of 4 weeks) in other interventional clinical trials
  • Patient without legal capacity who is unable to understand the nature, significance and consequences of the trial
  • Person who is in a relationship of dependence/employment with the sponsor or the investigator

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Control groupStandard of CarePatients with CMR-derived ECV% levels ≥25.9% will receive Standard of care
SpironolactoneStandard of CarePatients with CMR-derived ECV% levels ≥25.9% will receive Standard of care + Spironolactone (25 mg/d, p.o.)
Spironolactone + DihydralazineStandard of CarePatients with CMR-derived ECV% levels ≥25.9% will receive Standard of care + Spironolactone (25 mg/d, p.o.) + Dihydralazine (2x12.5 mg/d p.o. in slow acethylators, and 2x25mg / d p.o. in fast acethylators, confirmed by genetic testing)
Spironolactone + DihydralazineSpironolactone 25mgPatients with CMR-derived ECV% levels ≥25.9% will receive Standard of care + Spironolactone (25 mg/d, p.o.) + Dihydralazine (2x12.5 mg/d p.o. in slow acethylators, and 2x25mg / d p.o. in fast acethylators, confirmed by genetic testing)
SpironolactoneSpironolactone 25mgPatients with CMR-derived ECV% levels ≥25.9% will receive Standard of care + Spironolactone (25 mg/d, p.o.)
Spironolactone + DihydralazineDihydralazinePatients with CMR-derived ECV% levels ≥25.9% will receive Standard of care + Spironolactone (25 mg/d, p.o.) + Dihydralazine (2x12.5 mg/d p.o. in slow acethylators, and 2x25mg / d p.o. in fast acethylators, confirmed by genetic testing)
Primary Outcome Measures
NameTimeMethod
Extracellular volume (ECV)-derived matrix volume (measured by CMR)12 months

Differences between treatment groups in reduction of extracellular volume (ECV)- derived matrix volume (measured by CMR) after 12 months

Secondary Outcome Measures
NameTimeMethod
Methylation of rfGAP With Coiled-Coil, Ankyrin Repeat And PH Domains 3 (ACAP3)12 months

Measurement of Methylation of ACAP3 in %

Left ventricular blood volumes12 months

Differences in reduction of left ventricular blood volumes (measured by CMR) after 12 months

Kansas City Cardiomyopathy Questionnaire12 months

Differences in quality of life changes according to 23-items Kansas City Cardiomyopathy Questionnaire (KCCQ) after 12 months

NT-proBNP-levels12 months

Differences in NT-proBNP-levels (in pg/ml) after 12 months

Left ventricular ejection fraction12 months

Differences in recovery of left ventricular ejection fraction (EF) in % (measured by CMR) after 12 months

Global longitudinal strain12 months

Differences in recovery of global longitudinal strain (GLS) in % (measured by CMR) after 12 months

diastolic function12 months

Differences in recovery of diastolic function (measured by CMR) after 12 months

Left ventricular myocardial tissue volumes12 months

Differences in reduction of left ventricular myocardial tissue volumes (measured by CMR) after 12 months

6min-walking test distance (6MWT)12 months

Differences in 6min-walking test distance (6MWT; in m) after 12 months

Biomarker Procollagen III N-terminal propeptid (PIIINP)12 months

Measurement of PIIINP in ng/ml

NYHA status12 months

Differences in NYHA status after 12 months

Total mortality12 months

Rate of total mortality within 12 months

Cardiovascular mortality12 months

Rate of Cardiovascular mortality within 12 months

Methylation of Iroquois Homeobox 3 (IRX3)12 months

Measurement of Methylation of IRX3 in %

Methylation of Klotho12 months

Measurement of Methylation of Klotho in %

Methylation of RAS Protein Activator Like 1 (RASAL1)12 months

Measurement of Methylation of RASAL1 in %

Methylation of B9 Domain Containing 1 (B9D1)12 months

Measurement of Methylation of B9D1 in %

Methylation of Latency associated peptide (LAP)12 months

Measurement of Methylation of LAP in %

Heart failure hospitalizations12 months

Rate of Heart failure hospitalizations within 12 months

Biomarker Procollagen type I carboxy-terminal propeptide (PICP)12 months

Measurement of PICP in ng/ml

Ratio of Increased collagen degradation (CITP) vs. matrix metalloproteinase-1 (MMP-1)12 months

Measurement of CITP (in ng/l) and MMP-1 (in ng/ml)

Methylation of Growth Arrest And DNA Damage Inducible Gamma (GADD45G)12 months

Measurement of Methylation of GADD45G in %

Methylation of Chordin (CHRD)12 months

Measurement of Methylation of CHRD in %

Methylation of ATPase Sarcoplasmic/Endoplasmic Reticulum Ca2+ Transporting 2 (ATP2A2)12 months

Measurement of Methylation of ATP2A2 in %

Methylation of Bone Morphogenetic Protein 7 (BMP7)12 months

Measurement of Methylation of BMP7 in %

Serum creatinine12 months

Change in serum creatinine (in mg/dl) after 12 months

Cystatin c12 months

Change in cystatin c (in mg/l) after 12 months

Phosphate12 months

Change in phosphate (in mmol/l) after 12 months

Trial Locations

Locations (1)

University Medical Center Göttingen

🇩🇪

Göttingen, Lower Saxony, Germany

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