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PK Study of Tacrolimus and Cyclosporine When Co-Administered With Adefovir Dipivoxil in Post-Liver Transplant Patients

Phase 2
Completed
Conditions
Hepatitis B
Interventions
Registration Number
NCT00644761
Lead Sponsor
Gilead Sciences
Brief Summary

Open-label pharmacokinetic drug interaction study.

Detailed Description

Multi-center, phase 2, open-label, sequential-cohort, drug interaction study. Cohort 1 subjects (tacrolimus and adefovir dipivoxil) were enrolled first. Based on the findings in Cohort 1, a decision was made on whether to enroll subjects in Cohort 2 (cyclosporine and adefovir dipivoxil)(i.e., if no interaction was observed in Cohort 1, Cohort 2 subjects would not be enrolled). Since no pharmacokinetic interaction was observed in Cohort 1, Cohort 2 was not enrolled.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
16
Inclusion Criteria
  • 18-65 years of age
  • Greater than or equal to 6 months post-liver transplantation
  • Must be on a documented stable total daily dose of tacrolimus or cyclosporine for three months.
  • Must have calculated creatinine clearance greater than or equal 50 mL/min (Cockcroft-Gault method).
Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Treatment Arm 1Adefovir DipivoxilAdefovir dipivoxil 10 mg once daily with tacrolimus or cyclosporine for 14 days
Primary Outcome Measures
NameTimeMethod
To evaluate pharmacokinetics of tacrolimus or cyclosporine when co-administered with adefovir dipivoxil 10 mg once daily to patients post-liver transplantation21 days
Secondary Outcome Measures
NameTimeMethod
To evaluate PK of ADV 10 mg once daily when co-administered with tacrolimus or cyclosporine in patients post-liver transplantation. To evaluate the safety of ADV 10 mg once daily, when co-administered with tacrolimus or cyclosporine for 14 days.21 days

Trial Locations

Locations (11)

University of Miami

🇺🇸

Miami, Florida, United States

University of California, San Francisco

🇺🇸

San Francisco, California, United States

University of Pittsburgh

🇺🇸

Pittsburgh, Pennsylvania, United States

California Pacific Medical Center

🇺🇸

San Francisco, California, United States

University of Alabama at Birmingham

🇺🇸

Birmingham, Alabama, United States

Mayo Clinic

🇺🇸

Rochester, New York, United States

Columbia Presbyterian Medical Center

🇺🇸

New York, New York, United States

NYU Medical Center

🇺🇸

New York, New York, United States

Beth Israel Deaconess Medical Center

🇺🇸

Boston, Massachusetts, United States

Baylor Research Institute

🇺🇸

Dallas, Texas, United States

Cedars Sinai Medical Center

🇺🇸

Los Angeles, California, United States

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