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A Study of Orforglipron (LY3502970) in Participants With Type 2 Diabetes and Inadequate Glycemic Control With Insulin Glargine, With or Without Metformin and/or SGLT-2 Inhibitor

Phase 3
Active, not recruiting
Conditions
Type 2 Diabetes
Interventions
Drug: Placebo
Registration Number
NCT06109311
Lead Sponsor
Eli Lilly and Company
Brief Summary

The main purpose of this study is to determine the safety and efficacy of orforglipron. Participants will have Type 2 Diabetes (T2D) and have inadequate glycemic control with insulin glargine with or without metformin and/or SGLT-2 (sodium-glucose cotransporter-2) inhibitor. The study will last about 46 weeks and may include up to 20 visits.

Detailed Description

Not available

Recruitment & Eligibility

Status
ACTIVE_NOT_RECRUITING
Sex
All
Target Recruitment
520
Inclusion Criteria
  • Have Type 2 Diabetes (T2D)

  • Have HbA1c ≥7.0% [53 mmol/mol] to ≤10.5% [91 mmol/mol]

  • Have been treated with stable doses of the same formulation of the following for ≥90 days prior to screening visit 1 and have maintained the same doses through randomization:

    • insulin glargine U-100 (100 U/mL) ≥0.25 U/kg/QD (units per kilogram per day) or ≥20 U/QD alone, or
    • insulin glargine U-100 (100 U/mL) ≥0.25 U/kg/QD or ≥20 U/QD in combination with
    • metformin, or
    • SGLT-2 inhibitor, or
    • both metformin and SGLT-2 inhibitor.
  • Are of stable body weight (±5%) for at least 90 days prior to screening visit 1 and agree to not initiate an intensive diet or exercise program during the study with the intent of reducing body weight, other than the lifestyle and/or dietary measures for diabetes treatment.

  • Have a Body Mass Index (BMI) ≥23.0 kg/m^2 at baseline.

Exclusion Criteria
  • Have New York Heart Association functional classification III-IV congestive heart failure.

  • Have had any of the following cardiovascular conditions within 60 days prior to baseline.

    • acute myocardial infarction
    • cerebrovascular accident (stroke), or
    • hospitalization for congestive heart failure.
  • Have acute or chronic hepatitis, including a history of autoimmune hepatitis, signs or symptoms of any other liver disease other than nonalcoholic fatty liver disease

  • Have had chronic or acute pancreatitis any time.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Orforglipron Dose 2OrforglipronParticipants will receive orforglipron orally.
Orforglipron Dose 1OrforglipronParticipants will receive orforglipron orally.
Orforglipron Dose 3OrforglipronParticipants will receive orforglipron orally.
PlaceboPlaceboParticipants will receive placebo orally.
Primary Outcome Measures
NameTimeMethod
Orforglipron Dose 1, 2: Change from Baseline in Hemoglobin A1c (HbA1c)Baseline, Week 40
Secondary Outcome Measures
NameTimeMethod
Percentage Change from Baseline in non-HDL (non-high-density lipoprotein) CholesterolBaseline, Week 40
Change from Baseline in Body WeightBaseline, Week 40
Percentage of Participants Who Achieved HbA1c <7.0% (53 millimoles per mole (mmol/mol))Baseline to Week 40
Percentage of Participants Who Achieved HbA1c ≤6.5% (48 mmol/mol)Baseline to Week 40
Percentage Change from Baseline in Body WeightBaseline, Week 40
Percentage of Participants Who Achieved Weight Loss of ≥10%Baseline to Week 40
Orforglipron Dose 3: Change from Baseline in HbA1cBaseline, Week 40
Change from Baseline in Fasting Serum GlucoseBaseline, Week 40
Percentage of Participants Who Achieved Weight Loss of ≥15% from BaselineBaseline to Week 40
Percentage Change from Baseline in TriglyceridesBaseline, Week 40
Change from Baseline in Systolic Blood PressureBaseline, Week 40
Change from Baseline in Daily Insulin Glargine DoseBaseline, Week 40
Percentage of Participants Who Achieved Weight Loss of ≥5%Baseline to Week 40
Change from Baseline in Short Form 36-Version 2 (SF-36v2) Acute Form Domain and Summary ScoresBaseline, Week 40

Trial Locations

Locations (70)

Consano Clinical Research, LLC

🇺🇸

Shavano Park, Texas, United States

Texas Valley Clinical Research

🇺🇸

Weslaco, Texas, United States

L2IP - Instituto de Pesquisas Clínicas

🇧🇷

Brasília, Distrito Federal, Brazil

CEDOES

🇧🇷

Vitória, Espírito Santo, Brazil

Quanta Diagnóstico e Terapia

🇧🇷

Curitiba, Paraná, Brazil

Insight Centro de Pesquisas

🇧🇷

Porto Alegre, Rio Grande Do Sul, Brazil

Centro de Pesquisa Sao Lucas

🇧🇷

Campinas, São Paulo, Brazil

Centro Multidisciplinar de Estudos Clinicos

🇧🇷

Sao Bernardo do Campo, São Paulo, Brazil

ISPEM - Instituto São José dos Campos em Pesquisas Médicas

🇧🇷

São José dos Campos, São Paulo, Brazil

IBPClin - Instituto Brasil de Pesquisa Clínica

🇧🇷

Rio de Janeiro, Brazil

CPQuali Pesquisa Clínica

🇧🇷

São Paulo, Brazil

The Second People's Hospital of Hefei

🇨🇳

Hefei, Anhui, China

Wannan Medical College Yijishan Hospital

🇨🇳

Wuhu, Anhui, China

Beijing Hospital

🇨🇳

Beijing, Beijing, China

Chongqing General Hospital

🇨🇳

Chongqing, Chongqing, China

The First Affiliated Hospital of Henan University of Science &Technology

🇨🇳

Luoyang Shi, Henan, China

The Second Affiliated Hospital of Zhengzhou University

🇨🇳

Zhengzhou, Henan, China

The Second Affiliated Hospital of Nanjing Medical University

🇨🇳

Nanjing, Jiangsu, China

Nanjing First Hospital

🇨🇳

Nanjing, Jiangsu, China

Affiliated Hospital of Jiangsu University

🇨🇳

Zhenjiang, Jiangsu, China

Jinan Central Hospital

🇨🇳

Jinan, Shandong, China

Tokuyama Clinic

🇯🇵

Mihama-ku,Chiba City, Chiba, Japan

Hasegawa Medical Clinic

🇯🇵

Chitose, Hokkaido, Japan

MinamiAkatsukaClinic

🇯🇵

Mito, Ibaraki, Japan

Matoba Internal Medicine Clinic

🇯🇵

Ebina, Kanagawa, Japan

Takai Internal Medicine Clinic

🇯🇵

Kamakura-shi, Kanagawa, Japan

Shiraiwa Medical Clinic

🇯🇵

Kashiwara, Osaka, Japan

Fukuwa Clinic

🇯🇵

Chuo-ku, Tokyo, Japan

The Institute of Medical Science, Asahi Life Foundation

🇯🇵

Chuo-ku, Tokyo, Japan

Jinnouchi Hospital

🇯🇵

Kumamoto, Japan

Tokyo-Eki Center-building Clinic

🇯🇵

Chuo-ku, Tokyo, Japan

Medical Corporation Sato Medical clinic

🇯🇵

Ootaku, Tokyo, Japan

Tama Center Clinic Mirai

🇯🇵

Tama, Tokyo, Japan

Abe Clinic

🇯🇵

Oita, Japan

Kansai Electric Power Hospital

🇯🇵

Osaka, Japan

Centro de Endocrinologia y Nutricion

🇵🇷

Caguas, Puerto Rico

FDI Clinical Research

🇵🇷

San Juan, Puerto Rico

Diabdana

🇷🇴

Oradea, Bihor, Romania

C.M.D.T.A. Neomed

🇷🇴

Brasov, Brașov, Romania

Geea Medical Easy Diet

🇷🇴

Bucharest, București, Romania

Centrul Medical NutriLife

🇷🇴

Bucharest, București, Romania

Centrul Medical Endocrinologie si Diabet Dr. Paveliu

🇷🇴

Bucharest, București, Romania

CMI DNBM Dr. Pop Lavinia

🇷🇴

Baia Mare, Maramureș, Romania

SC Dentosim Queen SRL - Centrul Medical Diamed

🇷🇴

Târgu Mureș, Mureș, Romania

Milena Sante

🇷🇴

Galați, Romania

Diamed Obesity

🇷🇴

Galați, Romania

Clinica Korall

🇷🇴

Satu Mare, Romania

MD First Research - Chandler

🇺🇸

Chandler, Arizona, United States

Phoenix Clinical LLC

🇺🇸

Phoenix, Arizona, United States

SanRo Clinical Research Group

🇺🇸

Bryant, Arkansas, United States

Velocity Clinical Research, Gardena

🇺🇸

Gardena, California, United States

Loma Linda University Health System

🇺🇸

Loma Linda, California, United States

Western University of Health Sciences

🇺🇸

Pomona, California, United States

Med Partners, Inc. dba Premiere Medical Center of Burbank, Inc.

🇺🇸

Toluca Lake, California, United States

CMR of Greater New Haven, LLC

🇺🇸

Hamden, Connecticut, United States

Care Access - Brandon

🇺🇸

Brandon, Florida, United States

Encore Medical Research

🇺🇸

Hollywood, Florida, United States

Encore Medical Research - Weston

🇺🇸

Weston, Florida, United States

Orita Clinical Research

🇺🇸

Decatur, Georgia, United States

Bingham Memorial Hospital

🇺🇸

Blackfoot, Idaho, United States

St. Luke's Humphreys Diabetes Center: Boise

🇺🇸

Boise, Idaho, United States

Cotton O'Neil Diabetes & Endocrinology

🇺🇸

Topeka, Kansas, United States

Clinvest Headlands Llc

🇺🇸

Springfield, Missouri, United States

The Research Group of Lexington

🇺🇸

Lexington, Kentucky, United States

Richmond University Medical Center

🇺🇸

Staten Island, New York, United States

Velocity Clinical Research, Mt. Auburn

🇺🇸

Cincinnati, Ohio, United States

Velocity Clinical Research, Medford

🇺🇸

Medford, Oregon, United States

Tristar Clinical Investigations

🇺🇸

Philadelphia, Pennsylvania, United States

Frontier Clinical Research, LLC

🇺🇸

Scottdale, Pennsylvania, United States

Lifedoc Research - Lenox Park Drive

🇺🇸

Memphis, Tennessee, United States

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