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Evaluating the Safety and effectivenesS in Adult KorEaN Patients Treated With Tolvaptan for Management of Autosomal domInAnt poLycystic Kidney Disease

Phase 4
Completed
Conditions
Autosomal Dominant Polycystic Kidney Disease (ADPKD)
Interventions
Registration Number
NCT03949894
Lead Sponsor
Korea Otsuka Pharmaceutical Co., Ltd.
Brief Summary

To evaluate the safety and therapeutic effectiveness of tolvaptan when administered to slow the progression of cyst development and renal function insufficiency in adult Korean patients diagnosed with rapidly progressive ADPKD who have chronic kidney disease (CKD) stages 1-3 at initiation of treatment.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
118
Inclusion Criteria
  1. Subjects who voluntarily participate by giving written informed consent on this trial

  2. Male and female patients aged ≥ 19 to ≤ 50 years

  3. Subjects diagnosed with ADPKD based on the Unified Criteria for Ultrasonographic diagnosis of ADPKD (Pei-Ravine Criteria)

  4. Subjects with confirmed CKD stages 1-3 at the screening visit

  5. Subjects with confirmed rapidly progressive typical ADPKD 'Typical ADPKD'

    • refers to bilateral and diffuse distribution, with mild, moderate or severe replacement of kidney tissue by cysts, where all cysts contribute similarly to TKV.

'rapidly progressive ADPKD'

  • Patients will be defined as 'rapidly progressive ADPKD' if they meet any of the following criteria:

    • Mayo class 1C, 1D or 1E

      • Truncating PKD1 mutation confirmed by genetic testing before participating this trial ③ PRO-PKD score > 6 ④ Patients with ADPKD with a decline in Estimated glomerular filtration rate(eGFR) ≥ 5 mL/min/1.73 m2 within 1 year from the screening visit or with an average annual decline in eGFR ≥ 2.5 mL/min/1.73 m2 over a period of 5 years (excluding patients with an eGFR decline due to factors other than ADPKD, such as uncontrolled type 2 diabetes, early diabetic glomerular disease or immune-mediated glomerulonephritis)
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Exclusion Criteria
  1. Patients with hyponatremia or hypernatremia
  2. Patients with anuria
  3. Patients with volume depletion
  4. Patients who are unable to sense or appropriately respond to thirst
  5. Patients with contraindications to MRI assessment [e.g., ferromagnetic metal prosthesis, aneurysm clips, severe claustrophobia, large tattoo on the abdomen or back, etc.]
  6. Patients with severe renal impairment [e.g., patients with currently active glomerulonephritis, kidney cancer, having a single kidney, history of renal surgery within the last 3 years, etc.]
  7. Patients with severe hepatic impairment [e.g., cirrhosis, viral hepatitis, unspecified liver function test abnormalities (ALT or Aspartate aminotransferase(AST)) > 3 x ULN or Total Bilirubin > 2 x ULN), etc.]
  8. Patients with eGFR decline due to factors other than ADPKD (e.g., uncontrolled type 2 diabetes, early diabetic glomerular disease or immune-mediated glomerulonephritis, etc.)
  9. Patients with a history of hypersensitivity and/or specific reactions to benzazepine or benzazepine derivatives (such as Benazepril), or tolvaptan
  10. Patients with hereditary problems of galactose intolerance, the Lapp lactose deficiency or glucose-galactose malabsorption, etc.
  11. Patients who need chronic diuretic use
  12. Patients who are receiving any experimental (not marketed) or approved therapies that may affect the treatment of ADPKD within 6 months from the screening visit [e.g., anti-sense RNA therapy, rapamycin, sirolimus, everolimus and somatostatin analogs (octreotide, sandostatin), vasopressin antagonist (mozavaptan, conivaptan), vasopressin agonist (desmopressin)]
  13. Patients who have received cyst decompression or sclerotherapy within 3 years from the screening visit
  14. Patients with a history of taking tolvaptan within 6 months from the screening visit
  15. Patients who received any investigational medicinal product in another trial within 30 days from the screening visit
  16. Fertile women who are currently pregnant or breat feeding, or not willing to use or capable of using acceptable contraceptive methods (abstinence, oral, implanted or injected hormonal methods of contraception, intrauterine device or barrier methods of contraception, such as condom, contraceptive diaphragm and spermicidal agents) to avoid pregnancy until completion of the trial
  17. Patients who are, in the opinion of the investigator, unable to comply with the administration of the Investigational Medicinal Product(IMP) or the trial procedures
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Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
tolvaptanTolvaptan-
Primary Outcome Measures
NameTimeMethod
The incidences of TEAEsduring the tolvaptan treatment period and up to 7 days after the date of last dosing

The incidences of TEAEs

The incidences of TEAEs meeting any of the followings will be summarized.during the tolvaptan treatment period and up to 7 days after the date of last dosing

Liver injury \[ALT or AST elevation (\>3 x ULN) or Total Bilirubin elevation (\>2 x ULN), etc.\], AEs leading to death, Serious AEs, AEs leading to treatment discontinuation, AEs whose causal relationship with the IMP cannot be ruled out, Severe AEs, Dehydration, Effects on Sodium, Creatinine

Secondary Outcome Measures
NameTimeMethod
eGFR CKD-EPI annual mean change [mL/min/1.73m^2] (on-treatment)from Completion of Tolvaptan Titration Period (Visit 6, Week 4) to End of Treatment (Visit 25, Month 24)

(on-treatment)

Total kidney volume (TKV) annual mean percent change rate [%/year]from baseline to End of Treatment (Visit 25, Month 24)

Baseline TKV refers to the value measured during the screening period

eGFR CKD-EPI annual mean change [mL/min/1.73m^2] (off-treatment)from baseline to the Follow-up visit (Visit 26, 7 days after End of Treatment(Visit 25, Month 24))

(off-treatment)

Trial Locations

Locations (18)

Inje University Busan Paik Hospital

🇰🇷

Busan, Korea, Republic of

Seoul National University Hospital

🇰🇷

Seoul, Korea, Republic of

Kosin University Gospel Hospital

🇰🇷

Busan, Korea, Republic of

Severance Hospital

🇰🇷

Seoul, Korea, Republic of

The Catholic University of Korea Seoul St. Mary's Hospital

🇰🇷

Seoul, Korea, Republic of

Hallym University Chuncheon Sacred Heart Hospital

🇰🇷

Chuncheon, Korea, Republic of

Keimyung University Dongsan Medical Center

🇰🇷

Daegu, Korea, Republic of

Chungnam National University Hospital

🇰🇷

Daejeon, Korea, Republic of

Gachon University Gil Medical Center

🇰🇷

Incheon, Korea, Republic of

Kyungpook National University Hospital

🇰🇷

Daegu, Korea, Republic of

Chonnam National University Hospital

🇰🇷

Gwangju, Korea, Republic of

Hallym University Medical Center

🇰🇷

Pyeongchon, Korea, Republic of

Seoul National University Bundang Hospital

🇰🇷

Seongnam-si, Korea, Republic of

Gangnam Severance Hospital

🇰🇷

Seoul, Korea, Republic of

Hallym University Kangnam Sacred Heart Hospital

🇰🇷

Seoul, Korea, Republic of

Hanyang University Seoul Hospital

🇰🇷

Seoul, Korea, Republic of

Kangbuk Samsung Hospital

🇰🇷

Seoul, Korea, Republic of

SMG-SNU Boramae Medical Center

🇰🇷

Seoul, Korea, Republic of

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