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A Randomised Trial to Evaluate Toxicity and Efficacy of 1200mg and 1800mg Rifampicin for Pulmonary Tuberculosis

Phase 3
Completed
Conditions
Pulmonary Tuberculosis
Interventions
Registration Number
NCT02581527
Lead Sponsor
St George's, University of London
Brief Summary

In this trial, the investigators are assessing whether giving an increased dose of rifampicin to patients receiving the standard treatment for tuberculosis is safe and, when given for 4 months only, will also result in greater and faster killing of the tubercle bacillus in the lungs and result in relapse rates similar to those found in the World Health Organisation (WHO) recommended standard 6 month regimen.

Detailed Description

Type of design An open-label 3-arm trial to compare a standard 6-month control regimen with two 4-month treatment regimens for the treatment of tuberculosis (TB).

Disease/patients studied The trial will include 654 patients newly diagnosed with pulmonary TB with sputum positive or negative for TB on microscopy but with a positive result on a GeneXpert Test with organisms fully sensitive to rifampicin

The treatment regimens - Control and Experimental

Patients enrolled in the trial will be randomly allocated to receive one of the following three chemotherapy treatment regimens:

1. Control regimen (R10): The standard regimen of isoniazid, pyrazinamide and ethambutol plus 10 mg/kg rifampicin for the initial 8 weeks, followed by isoniazid and rifampicin (at the same dose size) for an additional 4 months (2HRZE/4HR)A.

2. Study regimen 1(SR1): 2 months of daily ethambutol, isoniazid, rifampicin, and pyrazinamide followed by 2 months of daily isoniazid and rifampicin. A supplement of either 450 mg (weight bands 35-39kg and 40-54kg) or 600mg (weight band 55-69kg and 70 and more kg) of rifampicin will be given throughout the four months (2EHR 1200Z/2HR1200)B.

3. Study regimen 2(SR2): 2 months of daily ethambutol, isoniazid, rifampicin, and pyrazinamide followed by 2 months of daily isoniazid and rifampicin. A supplement of either 450 mg (weight bands 35-39kg and 40-54kg) or 600mg (weight band 55-69kg and 70 and more kg) of rifampicin will be given throughout the four months (2EHR1800Z/2HR1800)C.

1.1 Outcome measures Primary outcome measure

1. Since the objective of the trial is to reduce treatment duration by increasing the dose of rifampicin, the primary outcome measure is the combined rate of failure at the end of treatment and relapse during the subsequent 12 months in smear positive patients.

2. The occurrence of grade 3 or 4 adverse events at any time during chemotherapy.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
672
Inclusion Criteria
  1. GeneXpert sputum positive, rifampicin susceptible, newly diagnosed pulmonary tuberculosis will be included even if they are microscopy negative.
  2. No previous anti-tuberculosis chemotherapy.
  3. Patients ≥ 18 years
  4. Consent to participation in the trial and to HIV testing
  5. Provide informed consent.
  6. Patient has a stable home address within easy reach of the treatment facility and likely to remain there for the next 18 months.
  7. Pre-menopausal women must be using a barrier form of contraception or be surgically sterilised or have an Intrauterine Contraceptive Device (IUCD) in place for the duration of the treatment phase
Exclusion Criteria
  1. Patients with rifampicin resistance identified by GeneXpert or by direct susceptibility testing (late exclusions).
  2. Has any condition that may prove fatal during the study period.
  3. Has TB meningitis.
  4. Has pre-existing non-tuberculous disease likely to prejudice the response to, or assessment of, treatment e.g. insulin-dependent diabetes, liver or kidney disease, blood disorders, peripheral neuritis, and severe thrombocytopenia, rash, increase of bilirubin and other diseases that are likely to be contraindicated with rifampicin
  5. Is female and known to be pregnant, or breast feeding.
  6. Is suffering from a condition likely to lead to uncooperative behaviour such as psychiatric illness or alcoholism.
  7. Has contraindications to any medications in the study regimens
  8. Is HIV positive
  9. Haemoglobin <7g/l
  10. Aspartate Aminotransferase (AST) or Alanine Aminotransferase (ALT) > 5 times the upper limit of normal (ULN) for that laboratory
  11. Creatinine clearance (CrCl) of < 30mls/min. Calculated as CrCl (mL/min) = N x [140-age (years)] x weight (kg) Serum creatinine (micromol/L) Where N = 1.23 males, 1.04 females
  12. Has glucose in urine
  13. Weight < 35kg

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Rifampicin 1800mg (Regimen 2)Pyrazinamide2 months daily 4FDC - high dose Rifampicin 1800mg, Isoniazid 75mg, Ethambutol 275mg and Pyrazinamide 400mg (intensive phase); followed by 2 months daily 2FDC - high dose Rifampicin 1800mg and Isoniazid 75mg (continuous phase)
Rifampicin 150mg (Control)Rifampicin2 months daily 4FDC - Rifampicin 150mg, Isoniazid 75mg, Ethambutol 275mg and Pyrazinamide 400mg (intensive phase); followed by 4 months daily 2FDC - Rifampicin 150mg and Isoniazid 75mg (continuous phase)
Rifampicin 150mg (Control)Ethambutol2 months daily 4FDC - Rifampicin 150mg, Isoniazid 75mg, Ethambutol 275mg and Pyrazinamide 400mg (intensive phase); followed by 4 months daily 2FDC - Rifampicin 150mg and Isoniazid 75mg (continuous phase)
Rifampicin 150mg (Control)Isoniazid2 months daily 4FDC - Rifampicin 150mg, Isoniazid 75mg, Ethambutol 275mg and Pyrazinamide 400mg (intensive phase); followed by 4 months daily 2FDC - Rifampicin 150mg and Isoniazid 75mg (continuous phase)
Rifampicin 150mg (Control)Pyrazinamide2 months daily 4FDC - Rifampicin 150mg, Isoniazid 75mg, Ethambutol 275mg and Pyrazinamide 400mg (intensive phase); followed by 4 months daily 2FDC - Rifampicin 150mg and Isoniazid 75mg (continuous phase)
Rifampicin 1200mg (Regimen 1)Rifampicin2 months daily 4FDC - high dose Rifampicin 1200mg, Isoniazid 75mg, Ethambutol 275mg and Pyrazinamide 400mg (intensive phase); followed by 2 months daily 2FDC - high dose Rifampicin 1200mg and Isoniazid 75mg (continuous phase)
Rifampicin 1200mg (Regimen 1)Isoniazid2 months daily 4FDC - high dose Rifampicin 1200mg, Isoniazid 75mg, Ethambutol 275mg and Pyrazinamide 400mg (intensive phase); followed by 2 months daily 2FDC - high dose Rifampicin 1200mg and Isoniazid 75mg (continuous phase)
Rifampicin 1200mg (Regimen 1)Ethambutol2 months daily 4FDC - high dose Rifampicin 1200mg, Isoniazid 75mg, Ethambutol 275mg and Pyrazinamide 400mg (intensive phase); followed by 2 months daily 2FDC - high dose Rifampicin 1200mg and Isoniazid 75mg (continuous phase)
Rifampicin 1200mg (Regimen 1)Pyrazinamide2 months daily 4FDC - high dose Rifampicin 1200mg, Isoniazid 75mg, Ethambutol 275mg and Pyrazinamide 400mg (intensive phase); followed by 2 months daily 2FDC - high dose Rifampicin 1200mg and Isoniazid 75mg (continuous phase)
Rifampicin 1800mg (Regimen 2)Rifampicin2 months daily 4FDC - high dose Rifampicin 1800mg, Isoniazid 75mg, Ethambutol 275mg and Pyrazinamide 400mg (intensive phase); followed by 2 months daily 2FDC - high dose Rifampicin 1800mg and Isoniazid 75mg (continuous phase)
Rifampicin 1800mg (Regimen 2)Isoniazid2 months daily 4FDC - high dose Rifampicin 1800mg, Isoniazid 75mg, Ethambutol 275mg and Pyrazinamide 400mg (intensive phase); followed by 2 months daily 2FDC - high dose Rifampicin 1800mg and Isoniazid 75mg (continuous phase)
Rifampicin 1800mg (Regimen 2)Ethambutol2 months daily 4FDC - high dose Rifampicin 1800mg, Isoniazid 75mg, Ethambutol 275mg and Pyrazinamide 400mg (intensive phase); followed by 2 months daily 2FDC - high dose Rifampicin 1800mg and Isoniazid 75mg (continuous phase)
Primary Outcome Measures
NameTimeMethod
The occurrence of grade 3 or 4 adverse events at any time during chemotherapy.18 months
the primary outcome measure is the combined rate of failure at the end of treatment and relapse during the subsequent 12 months in smear positive patients in the modified intent to treat population.18 months
Secondary Outcome Measures
NameTimeMethod
Time to unfavourable outcome in the modified intent-to-treat and per protocol sputum smear microscopy-positive population.18 Months
Combined unfavourable endpoint (rate of failure at the end of treatment and relapse) measured 18 months from randomisation in the Xpert MTB/RIF positive (i) modified intent-to-treat and (ii) per protocol populations18 months
Sputum cultures positive for M.tuberculosis at 8 and 12 weeks from randomisation.18 months
Per protocol analysis of the primary efficacy outcome (the combined rate of failure at the end of treatment and relapse during the subsequent 12 months in smear positive patients)18 months
Any adverse event, up to one month after completion of treatment, graded according to the DAIDS criteria1 month after end of treatment (7 months (Control), 5 months (Study regimens) )

Trial Locations

Locations (6)

Epicentre

🇺🇬

Mbarara, Uganda

Hospital Nacional Dos de Mayo

🇵🇪

Lima, Peru

GENETUP, National Anti-TB Association

🇳🇵

Kathmandu, Nepal

University of Botswana

🇧🇼

Gaborone, Botswana

Aga Khan University Hospital

🇵🇰

Karachi, Pakistan

Hopital National Ignace Deen

🇬🇳

Conakry, Guinea

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