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An active extension of LAQ/5062 study. A multinational, multi-center, randomized, double-blind, parallel-group study, to evaluate the safety, tolerability and efficacy of two doses (0.3mg and 0.6mg) of laquinimod, orally administered in relapsing remitting (R-R) Multiple Sclerosis (MS) subjects (study LAQ/5063 active double-blind phase) followed by an open label phase of laquinimod 0.6 mg daily (LAQ/5063 OL).

Phase 1
Conditions
Relapsing Remitting Multiple Sclerosis
MedDRA version: 14.1Level: PTClassification code 10063399Term: Relapsing-remitting multiple sclerosisSystem Organ Class: 10029205 - Nervous system disorders
Therapeutic area: Diseases [C] - Nervous System Diseases [C10]
Registration Number
EUCTR2005-004334-41-IT
Lead Sponsor
Teva Pharmaceutical Industries Ldt
Brief Summary

Not available

Detailed Description

Not available

Recruitment & Eligibility

Status
ot Recruiting
Sex
All
Target Recruitment
246
Inclusion Criteria

1. Subjects must have completed the 36 weeks of treatment (completion of the full 36 weeks or as requested by the Sponsor), of the active double-blind phase. 2. Women of child- bearing potential must practice a reliable method of birth control. (Acceptable methods of birth control in this study include: double barrier methods such as diaphragms with spermicide, condoms and spermicide. Also intrauterine devices; hormonal contraception must be accompanied by an additional method of birth control.). 3. Subjects must be willing and able to comply with the protocol requirements for the duration of the open-label phase (LAQ/5063 OL). 4. Subjects must give signed, written informed consent prior to entering the openlabel phase (LAQ/5063 OL). Inclusion Criteria for the LAQ/5063 OL open-label phase - further extension (after visit month 24) a. Subjects must have completed the 24 months of treatment of the first period of the open label phase. b. Women of child- bearing potential must practice a reliable method of birth control. (Acceptable methods of birth control in this study include: double barrier methods such as diaphragms with spermicide, condoms and spermicide. Also intrauterine devices; hormonal contraception must be accompanied by an additional method of birth control).
Are the trial subjects under 18? no
Number of subjects for this age range: 0
F.1.2 Adults (18-64 years) yes
F.1.2.1 Number of subjects for this age range
F.1.3 Elderly (>=65 years) no
F.1.3.1 Number of subjects for this age range

Exclusion Criteria

Premature discontinuation from LAQ/5063 active double-blind phase for any reason other than sponsor`s request 2. Pregnancy or breastfeeding 3. Subjects with clinically significant or unstable medical or surgical condition, detected or worsened during the active double-blind phase of LAQ/5063, which would preclude safe and complete study participation 4. Use of experimental drugs, immunosuppressive drugs, and/or participation in clinical studies within the period from termination of LAQ/5063 active doubleblind phase to the open-label phase (LAQ/5063 OL) 5. Previous treatment with immunomodulators with the exception of laquinimod (including IFN 1a and 1b, Glatiramer Acetate and IVIG) within 2 months prior to entering the open-label phase for those subjects who have a time gap between termination of LAQ/5063 active double-blind phase to the open-label phase (LAQ/5063 OL) 6. Use of corticosteroids within 30 days prior to entering the open-label phase, except for IV methylprednisolone 1 g/day for a maximum of 3 days, in the period from termination of LAQ/5063 active double-blind phase to the openlabel phase (LAQ/5063 OL) 7. Use of potent inhibitors of CYP3A4 within 2 weeks prior to open label phase (LAQ/5063 OL) and/or use of fluoxetine one month prior entering the open label phase (LAQ/5063 OL), in the period from termination of LAQ/5063 active double-blind phase to the open-label phase (LAQ/5063 OL) (see list in appendix 5) 8. Use of the following substrates of CYP1A2: theophylline and/or warfarin within 2 weeks prior to entering the open-label phase (LAQ/5063 OL), in the label phase (LAQ/5063 OL) 9. Use of amiodarone in the period from termination of LAQ/5063 active doubleblind phase to the open-label phase (LAQ/5063 OL) 10. Following the switch to new formulation (capsules), hypersensitivity to: mannitol, meglumine or sodium stearyl fumarate. Exclusion Criteria for the LAQ/5063 OL open-label phase- further extension (after visit month 24) a. Premature discontinuation from LAQ/5063 OL phase prior to completion of 24 months of treatment period b. Pregnancy or breastfeeding.

Study & Design

Study Type
Interventional clinical trial of medicinal product
Study Design
Not specified
Primary Outcome Measures
NameTimeMethod
Main Objective: To make treatment with laquinimod available to all subjects who previously participated in both LAQ/5062 study and the LAQ/5063 active double-blind phase (completion of the full 36 weeks or as requested by the Sponsor). To assess the long-term safety, and tolerability in the group that received active treatment in LAQ/5062 protocol and additional short term safety and tolerability in the group who received placebo treatment. LAQ/5063 OL phase will assess long-term safety and tolerability of 0.6 mg laquinimod once daily.;Secondary Objective: Further efficacy data will be obtained by comparing baseline to termination in the group who received placebo treatment in LAQ/5062 core study protocol.;Primary end point(s): Long term safety
Secondary Outcome Measures
NameTimeMethod
Secondary end point(s): Not applicable
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