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Study to Assess Drug Concentrations in Plasma of Different Extended-release Formulations of AZD1305

Phase 1
Completed
Conditions
Healthy
Interventions
Registration Number
NCT00957437
Lead Sponsor
AstraZeneca
Brief Summary

The purpose of this study is to evaluate the pharmacokinetics of different extended-release formulations of AZD1305 when given as single and multiple oral doses to healthy male volunteers.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
24
Inclusion Criteria
  • Provision of signed, written and dated informed consent prior to any study specific procedures.
  • Body mass index (BMI) between 19 and 30 kg/m2 and weigh at least 50 kg and no more than 100 kg.
Exclusion Criteria
  • History or presence of any clinically significant disease or disorder in the opinion of the investigator.
  • Use of nicotine in the last 4 weeks before screening and not more than 7 cigarettes per week (equivalent to 1 nicotine patch or 7 nicotine gums per week) before then. There will be no smoking until follow-up visit.
  • Any clinically relevant abnormal findings in physical examination, clinical chemistry, haematology, urinalysis, vital signs or ECG at baseline in the opinion of the investigator.

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
Part A: 3 way crossoverAZD1305AZD1305: ER test formulation 1 (w/wo food) and reference formulation
Part B1: single armAZD1305AZD1305: ER test formulation 1
Part B2: 3 way crossoverAZD1305AZD1305: ER test formulation 2 (w/wo food) and reference formulation
Primary Outcome Measures
NameTimeMethod
Pharmacokinetic variables of AZD1305 by assessment of drug concentrations in plasmaFrom predose until 48 hours post last dose
Secondary Outcome Measures
NameTimeMethod
Adverse Events, ECG variables, vital signs, physical examination, laboratory variables and weightFrequent safety measurements during the study, from screening period to follow-up

Trial Locations

Locations (1)

Research Site

🇬🇧

Harrow, United Kingdom

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