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A Phase 1/2 Study to Investigate CRB-701 in Solid Tumors

Phase 1
Recruiting
Conditions
Solid Tumor, Adult
Interventions
Registration Number
NCT06265727
Lead Sponsor
Corbus Pharmaceuticals Inc.
Brief Summary

The goal of this clinical trial is to define a safe and effective dose of CRB-701 for participants with solid tumors that are expressing a protein called nectin-4.

The main questions it aims to answer are:

What is the the safe and effective dose of CRB-701 when used alone? What cancers can be treated effectively with CRB-701?

Participants will be asked to attend clinic and be given a intravenous infusion of CRB-701 on its own. They will have blood tests and other assessments to measure whether CRB-701 will have CT or MRI scans to measure the effect on tumors.

Detailed Description

This is a three-part open-label, Phase 1/2 clinical trial designed to evaluate the safety, PK, and efficacy of CRB-701 in participants with advanced solid tumors expressing nectin-4.

Part A will include solid tumor types known to express nectin-4. Dose escalation will be guided by the Bayesian optimal interval (BOIN) design to determine the MTD of CRB-701. Four (4) dose groups are pre-determined. Dose escalation/de-escalation decisions are made based on the occurrence of DLT.

Part B will determine the RP2D of CRB-701 by evaluating two dose levels of CRB-701 by using a time-to-event Bayesian optimal Phase 2 (TOP) study design to optimize the dose of CRB-701 in one or more separate cohorts of participants with nectin-4-positive tumors.

During Part C, the RP2D dose of CRB-701 will be evaluated in five planned expansion cohorts using Simon's optimal two-stage design.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
420
Inclusion Criteria
  • Confirmed diagnosis of select advanced or metastatic nectin-4 expressing solid tumors that have progressed following at least one line of therapy or have no other standard therapy with proven clinical benefit.
Exclusion Criteria
  • Active of uncontrolled CNS metastases
  • History of solid tumors other than the diseases under study
  • History of and/or current cardiovascular events or conditions in the previous 6 months
  • Pre-existing >/= Grade 2 neuropathy
  • Hemoglobin A1C (HbA1C) >/= 8%, uncontrolled diabetes mellitus or know diabetic neuropathy
  • Active ocular disease at baseline
  • Chronic severe liver disease or live cirrhosis
  • Interstitial lung disease or pneumonitis within 6 months on initiating treatment on study
  • Other significant cormorbidities.

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
Part A Dose Escalation - CRB-701 Dose Level 1CRB-701CRB-701 Dose level 1, intravenous infusion over 30 mins, Dose schedule 1
Part A Dose Escalation - CRB-701 Dose Level 2CRB-701CRB-701 Dose Level 2, intravenous infusion over 30 mins, Dose schedule 1
Part A Dose Escalation - CRB-701 Dose Level 3CRB-701CRB-701 Dose Level 3, intravenous infusion over 30 mins, dose schedule 1
Part A Dose Escalation - CRB-701 Dose Level 4CRB-701CRB-701 Dose Level 4, intravenous infusion over 30 mins, dose schedule 1
Part B Dose Optimization: CRB-701 low doseCRB-701Selected Low dose of CRB-701, intravenous infusion over 30 mins, once every three weeks
Part C Dose Expansion - Cohort 1CRB-701Recommended Phase 2 dose and schedule of CRB-701, intravenous infusion over 30 mins
Part C Dose Expansion - Cohort 2CRB-701Recommended Phase 2 dose and schedule of CRB-701, intravenous infusion over 30 mins
Part C Dose Expansion - Cohort 3CRB-701Recommended Phase 2 dose of CRB-701 and schedule, intravenous infusion over 30 mins
Part C Dose Expansion - Cohort 4CRB-701Recommended Phase 2 dose of CRB-701 and schedule, intravenous infusion over 30 mins
Part C Dose Expansion - Cohort 5CRB-701Recommended Phase 2 dose of CRB-701 and schedule, intravenous infusion over 30 mins
Part B Dose Optimization: CRB-701 High doseCRB-701Selected high dose of CRB-701, intravenous infusion over 30 mins, dose schedule 1
Primary Outcome Measures
NameTimeMethod
Part A: To confirm the safety and tolerability and determine MTD and PADR for CRB-70121 days

Occurrence of Dose Limiting Toxicities as defined in the protocol

Part B & C : To evaluate efficacy in terms of Disease Control Rate (DCR)Up to 6 months

DCR is the sum of percentage of participants meeting the definition of Complete Response (CR), Partial Response (PR) or Stable Disease (SD) for at least 4 months using RECIST 1.1

Part B & C: To evaluate efficacy in terms of Objective Response Rate (ORR)Up to 6 months

ORR is the percentage of participants that achieve a response (CR + PR) using RECIST 1.1

Secondary Outcome Measures
NameTimeMethod
Parts A, B, % C: To characterize the safety profile of CRB-701Up to 6 months

Numbers of treatment emergent adverse events with severity determined using NCI CTCAE v5.0 after single or multiple doses of CRB-701 or single and multiple doses of CRB-701 and an anti-PD-(L)1 therapy

Maximum observed plasma concentration of CRB-701 [total ADC] (Cmax)Approximately 9 weeks

Maximum observed plasma concentration of total ADC after single and multiple doses

Maximum observed plasma concentration of free MMAE (Cmax)Approximately 9 weeks

Maximum observed plasma concentration of free MMAE after single and multiple doses

Maximum observed plasma concentration of Total CRB-701 antibody [Tab] (Cmax)Approximately 9 weeks

Maximum observed plasma concentration of free MMAE after single and multiple doses

Time to reach Cmax of Total CRB-701 antibody [Tab] (Tmax)Approximately 9 weeks

The amount of time to reach Cmax after single and multiple dose administration of Tab

Time to reach Cmax of free MMAE (Tmax)Approximately 9 weeks

The amount of time to reach Cmax after single and multiple dose administration of free MMAE

Time to reach Cmax of Total CRB-701 [Total ADC] (Tmax)Approximately 9 weeks

The amount of time to reach Cmax after single and multiple dose administration of CRB-701 (Total ADC)

Time to reach Cmax of Total CRB-701 antibody [Tab] (Cmax)Approximately 9 weeks

Maximum observed plasma concentration of free MMAE after single and multiple doses

Total Area Under the plasma concentration-time curve of Total CRB-701 [total ADC] (AUC)Approximately 9 weeks

Maximum observed plasma concentration of free MMAE after single and multiple doses

Total Area Under the plasma concentration-time curve of free MMAE (AUC)Approximately 9 weeks

Area under the plasma concentration versus time curve after single and multiple dose administration of free MMAE

Total Area Under the plasma concentration-time curve of Total CRB-701 antibody [Tab] (AUC)Approximately 9 weeks

Area under the plasma concentration versus time curve after single and multiple dose administration of Tab

Trial Locations

Locations (44)

O'Neal Comprehensive Cancer Center at University of Alabama-Birmingham

🇺🇸

Birmingham, Alabama, United States

City of Hope Cancer Center

🇺🇸

Duarte, California, United States

Moores Cancer Centre at UC San Diego Health

🇺🇸

San Diego, California, United States

Helen Diller Family Comprehensive Cancer Center - UCSF

🇺🇸

San Francisco, California, United States

Rocky Mountain Cancer Centres

🇺🇸

Denver, Colorado, United States

Yale Cancer Center

🇺🇸

New Haven, Connecticut, United States

Florida Cancer Specialists

🇺🇸

Orlando, Florida, United States

University of Chicago

🇺🇸

Chicago, Illinois, United States

Hope and Healing Cancer Center

🇺🇸

Hinsdale, Illinois, United States

Dana-Faber Cancer Institute

🇺🇸

Boston, Massachusetts, United States

Nebraska Hematology Oncology

🇺🇸

Lincoln, Nebraska, United States

Carolina BioOncology Institute

🇺🇸

Huntersville, North Carolina, United States

Texas Oncology

🇺🇸

Tyler, Texas, United States

Virginia Cancer Specialists

🇺🇸

Fairfax, Virginia, United States

Fred Hutchinson Cancer Center at University of Washington

🇺🇸

Seattle, Washington, United States

ICM-Val d'Aurelle

🇫🇷

Montpellier, France

CHU de Poitiers

🇫🇷

Poitiers, France

Institut de Cancerologie de l'Ouest

🇫🇷

St. Herblain, France

Gustave Roussy

🇫🇷

Villejuif, France

Careggi University Hospital

🇮🇹

Florence, Italy

European Institute of Oncology IRCCS

🇮🇹

Milan, Italy

Fondazione Policlinico Gemelli, IRCCS

🇮🇹

Rome, Italy

Centro Richerche Cliniche di Verona

🇮🇹

Verona, Italy

Aresnsia Research Clinic Bucharest

🇷🇴

Bucharest, Romania

Aresnsia Research Clinic Cluj-Napoca

🇷🇴

Cluj-Napoca, Romania

Centrul de Oncologie Sf. Nectarie

🇷🇴

Lasi, Romania

Centrul de Oncologie Euroclinic

🇷🇴

Lasi, Romania

Barcelona IOB Hospital Quironsalud (NEXT)

🇪🇸

Barcelona, Spain

Vall d-Hebron Institut d'Oncologia

🇪🇸

Barcelona, Spain

Fundacion Jimenez Diaz (START)

🇪🇸

Madrid, Spain

Hospital Clinico Universitario de Valencia

🇪🇸

Valencia, Spain

Adana Numune Egitim ve Arastirma Hastanesi (Adana City Education and Research Hospital)

🇹🇷

Adana, Turkey

Ankara University

🇹🇷

Ankara, Turkey

Ankara Etlik City Hospital

🇹🇷

Ankara, Turkey

Istanbul Medeniyet University

🇹🇷

Istanbul, Turkey

University of Birmingham NHS Foundation Trust

🇬🇧

Birmingham, United Kingdom

University of Cambridge NHS Foundation Trust

🇬🇧

Cambridge, United Kingdom

Velindre Cancer Centre

🇬🇧

Cardiff, United Kingdom

Leeds University Hospitals NHS Trust

🇬🇧

Leeds, United Kingdom

Guy's and St Thomas' Clinical Research Facility

🇬🇧

London, United Kingdom

Imperial Experimental Cancer Medicine Centre

🇬🇧

London, United Kingdom

The Christie Hospital

🇬🇧

Manchester, United Kingdom

University of Southampton

🇬🇧

Southampton, United Kingdom

University of Liverpool - Clatterbridge Medical Centre

🇬🇧

Wirral, United Kingdom

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