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Annatto-derived GG for Statin-associated Myopathy

Phase 1
Recruiting
Conditions
Myopathy; Primary
Interventions
Dietary Supplement: Low GG
Dietary Supplement: Placebo
Dietary Supplement: High GG
Registration Number
NCT05312424
Lead Sponsor
Texas Tech University Health Sciences Center
Brief Summary

To evaluate the effects of 3-months annatto-derived geranylgeraniol (GG) supplementation on statin-associated skeletal muscle health.

Detailed Description

Statins are widely prescribed cholesterol-lowering oral drugs. The majority of reported adverse effects due to statin include muscle pain, weakness, cramp, and tiredness. CoQ10 supplementation has been widely used to reduce statin-related muscle complaints. Several human studies have been reported with inconsistent effects of CoQ10 on statin-related symptoms. This study is to investigate the role of 3-month annatto-derived geranylgeraniol (GG) in statin-related muscle outcomes in humans. Qualified subjects will be matched by age, gender, and body weight, and then randomly assigned to a no GG group, a low GG dose group, or a high GG dose group. The outcome measures will be assessed at baseline and after 3 months. Muscle-associated measurements will be recorded using subject questionnaires (also follow-up after 3 and 6 months), muscle performance results, and blood samples. We will monitor the safety of subjects after 3 months. Food intake, physical activity, and medication changes will be recorded at baseline and after 3 months. All data will be analyzed statistically.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
95
Inclusion Criteria
  • Age ≥40 of either sex
  • Statin-treated patients with muscle pain alone or accompanied by other symptoms.
  • Patients currently receiving a statin who developed new-onset myalgias in within 90 day of initiation or a dosage increase
Exclusion Criteria
  • Malignancy or significant neurological or psychiatric disturbances, including alcohol or drug abuse.
  • Woman who is pregnant, breastfeeding, or of childbearing potential and not taking adequate contraceptive precautions.
  • Had CoQ10 supplement one month before starting the study.
  • Genetic musculoskeletal and neurologic disorder known to affect skeletal muscle metabolism
  • Had steroid medication one month before starting the study.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Low GGLow GGLOW GG group: subject will take one pill (150 mg olive oil) after breakfast and another pill (150 mg GG) after dinner
PlaceboPlaceboPlacebo group: subject will take one pill (150 mg olive oil) after breakfast and another pill (150 mg olive oil) after dinner
High GGHigh GGHIGH GG group: subject will take one pill (150 mg GG) after breakfast and another pill (150 mg GG) after dinner
Primary Outcome Measures
NameTimeMethod
SAMS-CIchange in SAMS-CI at 3 months

Statin-Associated Muscle Symptom Clinical Index (SAMS-CI) is to assess muscle pain, muscle weakness, tiredness, and cramps.

BPIchange in BPI at 3 months

Brief Pain Inventory (BPI) is to assess pain and interference of pain with everyday life.

Secondary Outcome Measures
NameTimeMethod
blood biomarkers: hsCRPchanges in serum hsCRP at 3 months

hsCRP is to assess inflammation

blood biomarkers: serum creatinine kinase activitychange in serum creatinine kinase activity at 3 months

Creatine kinase is to assess muscle damage.

blood biomarkers: myostatinchanges in serum myostatin at 3 months

Myostatin is to assess muscle damage

blood biomarkers: atrogin 1changes in serum atrogin 1 at 3 months

atrogin 1 is to assess muscle damage

Lower body isometric strengthchange in lower body isometric strength at 3 months

Lower body (i.e., predominantly of the quadriceps and hip extensors) isometric strength is measured using a dynamometer

Heel raise testchange in heel raise test at 3 months

Heel raise test is commonly used to test calf muscle endurance, function, and performance. Single-leg or both-leg raise will be tested while staining on a step bench

blood biomarker: IL-6changes in serum IL-6 at 3 months

IL-6 is to assess inflammation

Functional lower body strengthchange in functional lower body strength at 3 months

Functional lower body strength is measured using a loaded 50m walk.

blood lipid profileschanges in blood lipid profiles at 3 months

lipid profiles include total triglycerides, total cholesterol, HDL, and calculated LDL

plasma menaquinone-4 (MK4) + menaquinone-4 (MK7)changes in plasma MK4+MK7 at 3 months

MK4 and MK4 are vitamin K2 homologues and are measured by HPLC

Wall-sit testchange in wall-sit test at 3 months

Wall-sit test (wall-slide test) is to assess static leg strength and endurance, particularly of the quadriceps and hip extensors

Trial Locations

Locations (1)

Texas Tech University Health Sciences Center

🇺🇸

Lubbock, Texas, United States

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