MedPath

A Study Investigating the Efficacy and Safety of LBL-007 Plus Tislelizumab in Combination With Bevacizumab Plus Fluoropyrimidine Versus Bevacizumab Plus Fluoropyrimidine in Participants With Unresectable or Metastatic Colorectal Cancer

Phase 1
Active, not recruiting
Conditions
Unresectable or Metastatic Microsatellite Stable/Mismatch Repair Proficient Colorectal Cancer
Interventions
Registration Number
NCT05609370
Lead Sponsor
BeiGene
Brief Summary

This is a Phase 1b/2 study to investigate the efficacy and safety of LBL-007 plus tislelizumab when administered in combination with bevacizumab plus fluoropyrimidine, and LBL-007 in combination with bevacizumab plus fluoropyrimidine versus bevacizumab plus fluoropyrimidine to participants with colorectal cancer.

Detailed Description

Not available

Recruitment & Eligibility

Status
ACTIVE_NOT_RECRUITING
Sex
All
Target Recruitment
113
Inclusion Criteria
  • Participant must have measurable disease as defined per RECIST version 1.1
  • Has a histologically confirmed colorectal adenocarcinoma with metastatic or unresectable disease (Stage IV as defined by American Joint Committee on Cancer [AJCC] 8th edition)
  • No prior systemic therapy for colorectal cancer (CRC) in the metastatic setting except for the induction treatment of first-line therapy. Note: Local regional treatment performed during induction systemic treatment is allowed
  • Participants who have completed the first-line induction treatment, with an overall response of stable disease or better. The duration of induction treatment should be completed within approximately 6 months. The first dose of study treatment needs to occur within 2 weeks (for 2-week regimen) or 3 weeks (for 3-week regimen) to 6 weeks after Day 1 of the last cycle of induction therapy
Exclusion Criteria
  • Participants whose disease has become resectable at the investigator's discretion during or after induction treatment are not eligible
  • Progressive disease occurred less than 6 months from completion of any prior neoadjuvant therapy (ie, chemotherapy with or without radiotherapy) or adjuvant therapy (ie, chemotherapy with or without radiotherapy), whichever occurred later
  • Participants who have been treated with anti-epidermal growth factor receptor (EGFR) antibody in the induction treatment
  • Any prior therapy targeting T-cell stimulation or checkpoint pathways
  • Participants with B-raf proto-oncogene, serine/threonine kinase (BRAF)V600E mutations
  • Have locally or centrally confirmed microsatellite instability-high (MSI-H) by polymerase chain reaction (PCR) method or dMMR by immunohistochemistry (IHC) method

Note: Other protocol defined criteria may apply.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Phase 1b: Cohort -1: LBL-007 + Tislelizumab + Bevacizumab + CapecitabineBevacizumab or Bevacizumab biosimilarLBL-007 (low dose) + tislelizumab (low dose once every 3 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks) + capecitabine
Phase 1b: Cohort -1: LBL-007 + Tislelizumab + Bevacizumab + CapecitabineCapecitabineLBL-007 (low dose) + tislelizumab (low dose once every 3 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks) + capecitabine
Phase 1b: Cohort 1a: LBL-007 + Tislelizumab + Bevacizumab + CapecitabineLBL-007LBL-007 (medium dose) + tislelizumab (low dose once every 3 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks) + capecitabine
Phase 1b: Cohort 1a: LBL-007 + Tislelizumab + Bevacizumab + CapecitabineTislelizumabLBL-007 (medium dose) + tislelizumab (low dose once every 3 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks) + capecitabine
Phase 1b: Cohort 1a: LBL-007 + Tislelizumab + Bevacizumab + CapecitabineBevacizumab or Bevacizumab biosimilarLBL-007 (medium dose) + tislelizumab (low dose once every 3 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks) + capecitabine
Phase 1b: Cohort 1a: LBL-007 + Tislelizumab + Bevacizumab + CapecitabineCapecitabineLBL-007 (medium dose) + tislelizumab (low dose once every 3 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks) + capecitabine
Phase 1b: Cohort 1b: LBL-007 + Tislelizumab + Bevacizumab + 5-Fluorouracil (5-FU)LBL-007LBL-007 (medium dose) + tislelizumab (high dose once every 4 weeks) + bevacizumab (5 mg/kg once every 2 weeks) + 5-FU
Phase 1b: Cohort 1b: LBL-007 + Tislelizumab + Bevacizumab + 5-Fluorouracil (5-FU)TislelizumabLBL-007 (medium dose) + tislelizumab (high dose once every 4 weeks) + bevacizumab (5 mg/kg once every 2 weeks) + 5-FU
Phase 1b: Cohort 1b: LBL-007 + Tislelizumab + Bevacizumab + 5-Fluorouracil (5-FU)Bevacizumab or Bevacizumab biosimilarLBL-007 (medium dose) + tislelizumab (high dose once every 4 weeks) + bevacizumab (5 mg/kg once every 2 weeks) + 5-FU
Phase 1b: Cohort 1b: LBL-007 + Tislelizumab + Bevacizumab + 5-Fluorouracil (5-FU)5-FluorouracilLBL-007 (medium dose) + tislelizumab (high dose once every 4 weeks) + bevacizumab (5 mg/kg once every 2 weeks) + 5-FU
Phase 1b: Cohort 2: LBL-007 + Tislelizumab + Bevacizumab + FluoropyrimidineLBL-007LBL-007 (high dose) + tislelizumab (low dose every 3 weeks or high dose every 4 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 1b: Cohort 2: LBL-007 + Tislelizumab + Bevacizumab + FluoropyrimidineTislelizumabLBL-007 (high dose) + tislelizumab (low dose every 3 weeks or high dose every 4 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 1b: Cohort 2: LBL-007 + Tislelizumab + Bevacizumab + FluoropyrimidineBevacizumab or Bevacizumab biosimilarLBL-007 (high dose) + tislelizumab (low dose every 3 weeks or high dose every 4 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 1b: Cohort 2: LBL-007 + Tislelizumab + Bevacizumab + FluoropyrimidineCapecitabineLBL-007 (high dose) + tislelizumab (low dose every 3 weeks or high dose every 4 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 1b: Cohort 2: LBL-007 + Tislelizumab + Bevacizumab + Fluoropyrimidine5-FluorouracilLBL-007 (high dose) + tislelizumab (low dose every 3 weeks or high dose every 4 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 2: Arm A and Arm D: LBL-007 + Tislelizumab + Bevacizumab + FluoropyrimidineLBL-007LBL-007 (high dose) + tislelizumab (low dose every 3 weeks or high dose every 4 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 2: Arm A and Arm D: LBL-007 + Tislelizumab + Bevacizumab + FluoropyrimidineTislelizumabLBL-007 (high dose) + tislelizumab (low dose every 3 weeks or high dose every 4 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 2: Arm A and Arm D: LBL-007 + Tislelizumab + Bevacizumab + FluoropyrimidineBevacizumab or Bevacizumab biosimilarLBL-007 (high dose) + tislelizumab (low dose every 3 weeks or high dose every 4 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 2: Arm A and Arm D: LBL-007 + Tislelizumab + Bevacizumab + FluoropyrimidineCapecitabineLBL-007 (high dose) + tislelizumab (low dose every 3 weeks or high dose every 4 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 2: Arm A and Arm D: LBL-007 + Tislelizumab + Bevacizumab + Fluoropyrimidine5-FluorouracilLBL-007 (high dose) + tislelizumab (low dose every 3 weeks or high dose every 4 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 2: Arm B: LBL-007 + Bevacizumab + FluoropyrimidineLBL-007LBL-007 (high dose) + bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 2: Arm B: LBL-007 + Bevacizumab + FluoropyrimidineBevacizumab or Bevacizumab biosimilarLBL-007 (high dose) + bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 2: Arm B: LBL-007 + Bevacizumab + FluoropyrimidineCapecitabineLBL-007 (high dose) + bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 2: Arm B: LBL-007 + Bevacizumab + Fluoropyrimidine5-FluorouracilLBL-007 (high dose) + bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 2: Arm C and Arm E: Bevacizumab + FluoropyrimidineLBL-007Bevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 2: Arm C and Arm E: Bevacizumab + FluoropyrimidineTislelizumabBevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 2: Arm C and Arm E: Bevacizumab + FluoropyrimidineBevacizumab or Bevacizumab biosimilarBevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 2: Arm C and Arm E: Bevacizumab + FluoropyrimidineCapecitabineBevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 2: Arm C and Arm E: Bevacizumab + Fluoropyrimidine5-FluorouracilBevacizumab (7.5 mg/kg once every 3 weeks or 5 mg/kg once every 2 weeks) + fluoropyrimidine (5-FU or capecitabine)
Phase 1b: Cohort -1: LBL-007 + Tislelizumab + Bevacizumab + CapecitabineLBL-007LBL-007 (low dose) + tislelizumab (low dose once every 3 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks) + capecitabine
Phase 1b: Cohort -1: LBL-007 + Tislelizumab + Bevacizumab + CapecitabineTislelizumabLBL-007 (low dose) + tislelizumab (low dose once every 3 weeks) + bevacizumab (7.5 mg/kg once every 3 weeks) + capecitabine
Primary Outcome Measures
NameTimeMethod
Phase 1b: Number of participants with Adverse Events (AEs) and Serious AEs (SAEs)From the first dose of study drug(s) to 30 days after last dose, initiation of new anticancer therapy, death, withdrawal of consent, or loss to follow-up, whichever occurs first (up to approximately 28 months)

Number of participants with AEs and SAEs characterized by type, frequency, severity (as graded by National Cancer Institute Common Terminology Criteria for Adverse Events version 5.0 \[NCI-CTCAE v5.0\]).

Phase 2: Progression Free Survival (PFS) as Assessed by The Investigator in PD-L1 Positive Arms A and CApproximately 28 months

PFS, as assessed by the investigator per RECIST v1.1 is defined as the time from the date of randomization to the date of first documentation of disease progression or death, whichever occurs first.

Secondary Outcome Measures
NameTimeMethod
Phase 2: Objective Response rate (ORR) as Assessed by The Investigator in PD-L1 Positive Arms A and C and PD-L1 Negative Arms D and EApproximately 28 months

ORR is defined as the proportion of participants with a confirmed complete response (CR) or partial response (PR) from the time of randomization.

Phase 2: Duration of response (DOR) as Assessed by The Investigator in PD-L1 Positive Arms A and C and PD-L1 Negative arms D and EApproximately 28 months

DOR is defined as the time from the first confirmed objective response after randomization until the first documentation of disease progression or death, whichever comes first.

Phase 2: Progression Free Survival (PFS) as Assessed by The Investigator in PD-L1 Negative Arms D and EApproximately 28 months

PFS, as assessed by the investigator per RECIST v1.1 is defined as the time from the date of randomization to the date of first documentation of disease progression or death, whichever occurs first.

Phase 2: Number of participants with AEs and SAEsFrom the first dose of study drug(s) to 30 days after the last dose, initiation of new anticancer therapy, death, withdrawal of consent, or loss to follow-up, whichever occurs first (up to approximately 28 months)

Number of participants with AEs and SAEs characterized by type, frequency, severity as graded by NCI-CTCAE v5.0.

Trial Locations

Locations (76)

Baptist Md Anderson Cancer Center

🇺🇸

Jacksonville, Florida, United States

Alaska Oncology and Hematology, Llc

🇺🇸

Anchorage, Alaska, United States

Banner Md Anderson Cancer Center

🇺🇸

Gilbert, Arizona, United States

Toi Clinical Research

🇺🇸

Cerritos, California, United States

Usc Norris Comprehensive Cancer Center (Nccc)

🇺🇸

Los Angeles, California, United States

Valkyrie Clinical Trials

🇺🇸

Los Angeles, California, United States

UCLA

🇺🇸

Los Angeles, California, United States

Hoag Memorial Presbyterian

🇺🇸

Newport, California, United States

Kaiser Permanente Northern California

🇺🇸

Vallejo, California, United States

Shanxi Provincial Cancer Hospital

🇨🇳

Taiyuan, Shanxi, China

Fort Wayne Medical Oncology and Hematology

🇺🇸

Fort Wayne, Indiana, United States

Baptist Health Lexington

🇺🇸

Lexington, Kentucky, United States

University of Kentucky Markey Cancer Center

🇺🇸

Lexington, Kentucky, United States

Norton Cancer Institute

🇺🇸

Louisville, Kentucky, United States

Pontchartrain Cancer Center

🇺🇸

Covington, Louisiana, United States

Ochsner Clinic Foundation

🇺🇸

New Orleans, Louisiana, United States

Washington University School of Medicine

🇺🇸

Saint Louis, Missouri, United States

St Vincent Frontier Cancer Center

🇺🇸

Billings, Montana, United States

Comprehensive Cancer Centers of Nevada

🇺🇸

Las Vegas, Nevada, United States

Cancer Care Specialists

🇺🇸

Reno, Nevada, United States

University of New Mexico Cancer Center

🇺🇸

Albuquerque, New Mexico, United States

Perlmutter Cancer Center At Winthrop Oncology Hematology Associatesnyu Winthrop Hospital

🇺🇸

Mineola, New York, United States

Laura and Isaac Perlmutter Cancer Center At Nyu Langone Health

🇺🇸

New York, New York, United States

Columbia University Medical Center

🇺🇸

New York, New York, United States

Duke Cancer Center

🇺🇸

Durham, North Carolina, United States

University of Tennessee Medical Center

🇺🇸

Knoxville, Tennessee, United States

Ut Southwestern Medical Center

🇺🇸

Dallas, Texas, United States

Ut Health San Antonio Mays Cancer Center

🇺🇸

San Antonio, Texas, United States

Virginia Cancer Specialists

🇺🇸

Fairfax, Virginia, United States

Cancer Care Northwest

🇺🇸

Spokane Valley, Washington, United States

Multicare Health System Institute For Research and Innovation

🇺🇸

Tacoma, Washington, United States

Blacktown Cancer and Haematology Centre

🇦🇺

Blacktown, New South Wales, Australia

Orange Health Service (Central West Cancer Care Centre)

🇦🇺

Orange, New South Wales, Australia

Riverina Cancer Care Centre

🇦🇺

Wagga Wagga, New South Wales, Australia

Calvary Mater Newcastle

🇦🇺

Waratah, New South Wales, Australia

Pindara Private Hospital

🇦🇺

Benowa, Queensland, Australia

Icon Cancer Centre South Brisbane

🇦🇺

South Brisbane, Queensland, Australia

Flinders Centre For Innovation in Cancer (Fcic)

🇦🇺

Bedford Park, South Australia, Australia

Lyell McEwin Hospital

🇦🇺

Elizabeth Vale, South Australia, Australia

Monash Health

🇦🇺

Clayton, Victoria, Australia

Austin Health

🇦🇺

Heidelberg, Victoria, Australia

The Alfred Hospital

🇦🇺

Melbourne, Victoria, Australia

St John of God, Murdoch

🇦🇺

Murdoch, Western Australia, Australia

One Clinical Research

🇦🇺

Nedlands, Western Australia, Australia

The Second Hospital of Anhui Medical University

🇨🇳

Hefei, Anhui, China

Peking University First Hospital

🇨🇳

Beijing, Beijing, China

Beijing Tsinghua Changgung Hospital

🇨🇳

Beijing, Beijing, China

Fujian Medical University Union Hospital

🇨🇳

Fuzhou, Fujian, China

Quanzhou First Affliated Hospital of Fujian Medical University

🇨🇳

Quanzhou, Fujian, China

The First Affiliated Hospital of Xiamen University

🇨🇳

Xiamen, Fujian, China

Gansu Provincial Hospital

🇨🇳

Lanzhou, Gansu, China

Sun Yat Sen Memorial Hospital, Sun Yat Sen University (North)

🇨🇳

Guangzhou, Guangdong, China

Zhujiang Hospital of Southern Medical University

🇨🇳

Guangzhou, Guangdong, China

The First Affiliated Hospital of Shantou University Medical College

🇨🇳

Shantou, Guangdong, China

Nanyang Central Hospital

🇨🇳

Nanyang, Henan, China

Henan Cancer Hospital

🇨🇳

Zhengzhou, Henan, China

Hubei Cancer Hospital

🇨🇳

Wuhan, Hubei, China

Hunan Cancer Hospital

🇨🇳

Changsha, Hunan, China

The First Peoples Hospital of Changzhou

🇨🇳

Changzhou, Jiangsu, China

Nantong First Peoples Hospital

🇨🇳

Nantong, Jiangsu, China

Affiliated Hospital of Jiangnan University South Campus

🇨🇳

Wuxi, Jiangsu, China

The First Hospital of Jilin University

🇨🇳

Changchun, Jilin, China

General Hospital of Ningxia Medical University

🇨🇳

Yinchuan, Ningxia, China

Shandong Cancer Hospital

🇨🇳

Jinan, Shandong, China

Jining No.1 Peoples Hospital West Branch

🇨🇳

Jining, Shandong, China

Linyi Peoples Hospital

🇨🇳

Linyi, Shandong, China

Qingdao Municipal Hospital

🇨🇳

Qingdao, Shandong, China

Renji Hospital Shanghai Jiao Tong University School of Medicine

🇨🇳

Shanghai, Shanghai, China

Shanghai 10Th Peoples Hospital

🇨🇳

Shanghai, Shanghai, China

Shanghai East Hospital Branch Hospital

🇨🇳

Shanghai, Shanghai, China

Tianjin Medical University Cancer Institute and Hospital

🇨🇳

Tianjin, Tianjin, China

Tianjin Union Medical Center (Nankai University Affiliated Hospital)

🇨🇳

Tianjin, Tianjin, China

Karamay Central Hospital of Xinjiang

🇨🇳

Karamay, Xinjiang, China

The Xinjiang Uygur Autonomous Region Peoples Hospital

🇨🇳

Urumqi, Xinjiang, China

The Second Affiliated Hospital of Zhejiang University School of Medicine

🇨🇳

Hangzhou, Zhejiang, China

Pan American Oncology Trials, Llc

🇵🇷

Rio Piedras, Puerto Rico

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