MedPath

Linagliptin Response to OGTT in Prediabetes and Type 2 Diabetes Mellitus

Phase 3
Completed
Conditions
PreDiabetes
Type 2 Diabetes
Interventions
Drug: Dipeptidyl-Peptidase IV Inhibitors
Registration Number
NCT05290506
Lead Sponsor
National University of Malaysia
Brief Summary

There are studies that suggest glycemic response to incretin-based therapies differs between Asians and Caucasians, whereby Asians have better response compared to Caucasians. Hence, the therapeutic response could also be augmented by difference in incretin system among various ethnicities. This study is carried out to study the effect of dipeptidyl-peptidase IV (DPPIV) inhibitors in prediabetes and T2DM patients who have different levels of GLP-1 and to determine the effect on glycemic profiles, insulin resistance/sensitivity, beta-cell functon.

Detailed Description

A 12-week, open-label, single treatment study using linagliptin is conducted in 28 prediabetes and 22 T2DM subjects who are divided into low and high fasting GLP-1 groups. Prediabetes are recruited from OGTT screening. Type 2 diabetes patients are recruited from specialised diabetes clinic and routine follow-up. A 75-g oral glucose tolerance test (OGTT) is performed at week 0 and 12. Venous blood samples were drawn at times 0 (before initiation of OGTT), 30, 60, 90, 120 min from the indwelling catheter for measurement of glucose and insulin.All prediabetes and T2DM subjects receive Linagliptin 5mg once daily for a duration of 12 weeks.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
50
Inclusion Criteria
  • Prediabetes diagnosed from OGTT and T2DM subjects
  • HbA1c > 6.5% and <10%
  • Subjects not receiving any glucose-lowering medication or just receiving metformin and/or sulphonylureas and/or alpha-glucosidase inhibitors on stable dose for at least 3 months.
  • Subjects who are willing to participate and sign the informed consent form
Exclusion Criteria
  • Subjects with ketoacidosis or lactic acidosis, overt diabetes, another disease causing secondary glucose intolerance, congestive heart failure (New York Heart Association Class III or IV), myocardial infarction, stroke or ischemic attacks in past 6 months, uncontrolled severe hypertension, active liver conditions such as cirrhosis or hepatitis [elevation in liver enzymes to higher activities than double the respective normal value], moderate to severe renal insufficiency, pregnancy, breast-feeding
  • Patients receiving insulin, GLP-1 receptor agonists, dipeptidyl peptidase IV inhibitors or glucose-lowering medications other than metformin /sulphonylureas /alpha-glucosidase inhibitors as treatment.
  • Subjects with uncontrolled blood glucose HbA1c>10%
  • Subjects who plan to move out of state / country

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Prediabetes Low GLP-1Dipeptidyl-Peptidase IV Inhibitorsprediabetes patients were divided into high GLP-1 and low GLP-1 groups based on the median of fasting GLP-1 level. linagliptin 5mg once daily was administered.
Prediabetes High GLP-1Dipeptidyl-Peptidase IV Inhibitorsprediabetes patients were divided into high GLP-1 and low GLP-1 groups based on the median of fasting GLP-1 level. linagliptin 5mg once daily was administered.
Diabetes Low GLP-1Dipeptidyl-Peptidase IV Inhibitorstype 2 diabetes mellitus patients were divided into high GLP-1 and low GLP-1 groups based on the median of fasting GLP-1 level. linagliptin 5mg once daily was administered.
Diabetes High GLP-1Dipeptidyl-Peptidase IV Inhibitorstype 2 diabetes mellitus patients were divided into high GLP-1 and low GLP-1 groups based on the median of fasting GLP-1 level. linagliptin 5mg once daily was administered.
Primary Outcome Measures
NameTimeMethod
change from baseline in HbA1c after 12-week treatmentbaseline to 12 weeks

plasma level of fasting HbA1c is taken at week 0 and 12 of study before OGTT

change from baseline in glucose after 12-week treatmentbaseline to 12 weeks

OGTT is performed at week 0 (baseline) and 12 (complete treatment). plasma glucose levels are taken at time 0,30,60,90,120 minutes during OGTT.

change from baseline in insulin sensitivity/resistance index after 12-week treatmentbaseline to 12 weeks

OGTT is performed at week 0 (baseline) and 12. Plasma levels of glucose and insulin are taken at time 0,30,60,90,120 min during the OGTT. HOMA-IR, HOMA-IS are used to measure insulin resistance and insulin sensitivity at week 0 and week 12

Secondary Outcome Measures
NameTimeMethod
change from baseline in beta-cell function after 12-week treatmentbaseline to 12 weeks

OGTT is performed at week 0 (baseline) and 12 (treatment complete). HOMS-beta, insulinogenic index, oral disposition index are used to measure beta-cell funciton at week 0 and 12

Trial Locations

Locations (1)

Hospital Sultan Ismail

🇲🇾

Johor Bahru, Johor, Malaysia

© Copyright 2025. All Rights Reserved by MedPath