MedPath

Certolizumab Pegol in Subjects With Active Axial Spondyloarthritis

Phase 3
Completed
Conditions
Spondyloarthropathies
Interventions
Biological: CZP 400 mg Q4W
Biological: CZP 200 mg Q2W
Other: Placebo
Registration Number
NCT01087762
Lead Sponsor
UCB BIOSCIENCES GmbH
Brief Summary

The study is a Phase 3, multicenter, randomized, double-blind, placebo-controlled study to evaluate the efficacy and safety of two dose regimens of Certolizumab Pegol (CZP) in subjects with active axial Spondyloarthritis (axial SpA).

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
325
Inclusion Criteria
  • Documented diagnosis of adult-onset axial Spondyloarthritis (SpA) of at least 3 months' duration as defined by the specified Assessment of Spondyloarthritis International Society (ASAS) criteria

  • Active disease as defined by:

    • Bath Ankylosing Spondylitis Disease Activity Index (BASDAI) score ≥ 4
    • Back pain ≥ 4 on a 0 to 10 Neurobehavioral Rating Scale (NRS) (from BASDAI item 2)
    • C-Reactive Protein (CRP) > ULN (Upper Limit of Normal) and/or current evidence (ie, within the last 3 months from Screening) for Sacroiliitis on Magnetic Resonance Imaging (MRI) as defined by Assessment of Spondyloarthritis International Society (ASAS) criteria
  • Intolerance to or inadequate response to at least 1 Nonsteroidal Anti-Inflammatory Drug (NSAID)

Exclusion Criteria
  • Presence of total Spinal Ankylosis ("bamboo spine")
  • Diagnosis of any other Inflammatory Arthritis
  • Prior treatment with any experimental biological agents for treatment of Axial Spondyloarthritis (SpA)
  • Exposure to more than 1 TNF-antagonist or to more than 2 previous biological agents for Axial Spondyloarthritis (SpA)
  • History of or current chronic or recurrent infections
  • High risk of infection
  • Recent live vaccination
  • Concurrent malignancy or a history of malignancy
  • Class III or IV congestive heart failure - New York Heart Association (NYHA)
  • Demyelinating disease of the central nervous system
  • Female subjects who are breastfeeding, pregnant or plan to become pregnant during the study or within 3 months following the last dose of the investigational product
  • Subjects with any other condition which, in the investigator's judgment, would make the subject unsuitable for inclusion in the study

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
CZP 400 mg Q4WCZP 400 mg Q4WSubjects received Certolizumab Pegol (CZP) 400 mg subcutaneous (sc) on Weeks 0, 2 and 4, followed by 400 mg CZP sc every 4 weeks (Q4W) from Week 8 onwards. Subjects received 2 injections of Placebo every 4 weeks in between the 2 injections of 200 mg CZP to maintain the study blind.
Placebo to CZP 200 mg escape on Week 16PlaceboMatching Placebo to CZP injections from Week 0 to Week 16. Subjects who did not achieve certain predefined response criteria at both Weeks 14 and 16 left the Placebo group on Week 16 and were treated with three loading doses of CZP 400 mg sc on Weeks 16, 18 and 20, followed by 200 mg CZP sc every 2 weeks (Q2W) from Week 22 onwards. Additionally, Placebo injections were administered as appropriate in order to maintain the study blind.
CZP 200 mg Q2WCZP 200 mg Q2WSubjects received Certolizumab Pegol (CZP) 400 mg subcutaneous (sc) on Weeks 0, 2 and 4, followed by 200 mg CZP sc every 2 weeks (Q2W) from Week 6 onwards. At every visit, subjects received one injection of 200 mg CZP and one injection of Placebo to maintain the study blind.
CZP 200 mg Q2WPlaceboSubjects received Certolizumab Pegol (CZP) 400 mg subcutaneous (sc) on Weeks 0, 2 and 4, followed by 200 mg CZP sc every 2 weeks (Q2W) from Week 6 onwards. At every visit, subjects received one injection of 200 mg CZP and one injection of Placebo to maintain the study blind.
PlaceboPlaceboMatching Placebo to CZP injections from Week 0 to Week 24. Placebo subjects who did not achieve certain predefined response criteria at both Weeks 14 and 16 left the Placebo group on Week 16. After 24 weeks, all subjects were randomized to active treatment with CZP 200 mg Q2W or CZP 400 mg Q4W.
Placebo to CZP 200 mg escape on Week 16CZP 200 mg Q2WMatching Placebo to CZP injections from Week 0 to Week 16. Subjects who did not achieve certain predefined response criteria at both Weeks 14 and 16 left the Placebo group on Week 16 and were treated with three loading doses of CZP 400 mg sc on Weeks 16, 18 and 20, followed by 200 mg CZP sc every 2 weeks (Q2W) from Week 22 onwards. Additionally, Placebo injections were administered as appropriate in order to maintain the study blind.
Placebo to CZP 400 mg escape on Week 16PlaceboMatching Placebo to CZP injections from Week 0 to Week 16. Subjects who did not achieve certain predefined response criteria at both Weeks 14 and 16 left the Placebo group on Week 16 and were treated with three loading doses of CZP 400 mg sc on Weeks 16, 18 and 20, followed by 400 mg CZP sc every 4 weeks (Q4W) from Week 24 onwards. Additionally, Placebo injections were administered as appropriate in order to maintain the study blind.
Placebo to CZP 400 mg on Week 24CZP 400 mg Q4WMatching Placebo to CZP injections from Week 0 to Week 24. Three loading doses of CZP 400 mg sc were given on Weeks 24, 26 and 28, followed by 400 mg CZP sc every 4 weeks (Q4W) from Week 32 onwards. Additionally, Placebo injections were administered as appropriate in order to maintain the study blind.
CZP 400 mg Q4WPlaceboSubjects received Certolizumab Pegol (CZP) 400 mg subcutaneous (sc) on Weeks 0, 2 and 4, followed by 400 mg CZP sc every 4 weeks (Q4W) from Week 8 onwards. Subjects received 2 injections of Placebo every 4 weeks in between the 2 injections of 200 mg CZP to maintain the study blind.
Placebo to CZP 400 mg on Week 24PlaceboMatching Placebo to CZP injections from Week 0 to Week 24. Three loading doses of CZP 400 mg sc were given on Weeks 24, 26 and 28, followed by 400 mg CZP sc every 4 weeks (Q4W) from Week 32 onwards. Additionally, Placebo injections were administered as appropriate in order to maintain the study blind.
Placebo to CZP 400 mg escape on Week 16CZP 400 mg Q4WMatching Placebo to CZP injections from Week 0 to Week 16. Subjects who did not achieve certain predefined response criteria at both Weeks 14 and 16 left the Placebo group on Week 16 and were treated with three loading doses of CZP 400 mg sc on Weeks 16, 18 and 20, followed by 400 mg CZP sc every 4 weeks (Q4W) from Week 24 onwards. Additionally, Placebo injections were administered as appropriate in order to maintain the study blind.
Placebo to CZP 200 mg on Week 24CZP 200 mg Q2WMatching Placebo to CZP injections from Week 0 to Week 24. Three loading doses of CZP 400 mg sc were given on Weeks 24, 26 and 28, followed by 200 mg CZP sc every 2 weeks (Q2W) from Week 30 onwards. Additionally, Placebo injections were administered as appropriate in order to maintain the study blind.
Placebo to CZP 200 mg on Week 24PlaceboMatching Placebo to CZP injections from Week 0 to Week 24. Three loading doses of CZP 400 mg sc were given on Weeks 24, 26 and 28, followed by 200 mg CZP sc every 2 weeks (Q2W) from Week 30 onwards. Additionally, Placebo injections were administered as appropriate in order to maintain the study blind.
Primary Outcome Measures
NameTimeMethod
Assessment in Axial Spondyloarthritis International Society 20 % (ASAS20) Response Criteria at Week 12Week 12

The ASAS20 is defined as an improvement of at least 20 % and absolute improvement of at least 1 unit on a 0 to 10 Numeric Rating Scale (NRS) in at least 3 of the 4 following domains:

* Patient's Global Assessment of Disease Activity

* Pain assessment (total spinal pain)

* Function (represented by Bath Ankylosing Spondylitis Functional Index (BASFI))

* Inflammation (the mean of the Bath Ankylosing Spondylitis Disease Activity Index (BASDAI) questions 5 and 6 concerning morning stiffness intensity and duration)

and absence of deterioration in the potential remaining domain (deterioration is defined as a relative worsening of at least 20 % and an absolute worsening of at least 1 unit).

Secondary Outcome Measures
NameTimeMethod
Change From Baseline in the Bath Ankylosing Spondylitis Metrology Index (BASMI) at Week 12From Baseline to Week 12

The BASMI characterizes the spinal mobility of subjects with axial Spondyloarthritis (SpA) and Ankylosing Spondylitis (AS). It is a disease-specific measure consisting of 5 clinical measures to reflect subject axial status: cervical rotation; tragus to wall distance; lateral lumbar flexion; lumbar flexion (modified Schober test); intermalleolar distance. According to the linear definition of the BASMI a score of 0 to 10 is calculated for each item based on the measurement. The mean of the sum of the 5 scores provides the BASMI score. The higher the BASMI score the more severe the patient's limitation of movement due to their axial SpA. A negative value in BASMI change from Baseline indicates an improvement from Baseline. The higher the negative value the better the improvement.

Change From Baseline in Sacroiliac Spondyloarthritis Research Consortium of Canada (SPARCC) Score at Week 12From Baseline to Week 12

The SPARCC scoring method for lesions found on the Magnetic Resonance Imaging (MRI) is based on an abnormal increased signal on the Short-Tau-Inversion Recovery (STIR) sequence, representing bone marrow edema. Total Sacroiliac (SI) joint SPARCC score can range from 0 to 72 with higher scores indicating higher joint inflammation. A negative value in SPARCC change from Baseline indicates an improvement from Baseline. The higher the negative value the higher the reduction of inflammation.

Assessment in Axial Spondyloarthritis International Society 20 % (ASAS20) Response Criteria at Week 24Week 24

The ASAS20 is defined as an improvement of at least 20 % and absolute improvement of at least 1 unit on a 0 to 10 Numeric Rating Scale (NRS) in at least 3 of the 4 following domains:

* Patient's Global Assessment of Disease Activity

* Pain assessment (total spinal pain)

* Function (represented by Bath Ankylosing Spondylitis Functional Index (BASFI))

* Inflammation (the mean of the Bath Ankylosing Spondylitis Disease Activity Index (BASDAI) questions 5 and 6 concerning morning stiffness intensity and duration)

and absence of deterioration in the potential remaining domain (deterioration is defined as a relative worsening of at least 20 % and an absolute worsening of at least 1 unit).

Change From Baseline in the Bath Ankylosing Spondylitis Disease Activity Index (BASDAI) at Week 24From Baseline to Week 24

The BASDAI is a validated self-reported instrument which consists of six 10 unit horizontal Numerical Rating Scales (NRSs) to measure severity of fatigue, spinal and peripheral joint pain and swelling, enthesitis, and morning stiffness (both severity and duration, respectively) over the last week. The final BASDAI score ranges from 0 to 10, with lower scores indicating lower disease activity. A negative value in BASDAI change from Baseline indicates an improvement from Baseline. The higher the negative value the better the improvement.

Change From Baseline in the Bath Ankylosing Spondylitis Functional Index (BASFI) at Week 24From Baseline to Week 24

The BASFI assesses physical function in comprising 10 items relating to activities during the past week. Each item ranges from 0 ("Easy") to 10 ("Impossible"). The BASFI is the mean of the 10 scores such that the total score ranges from 0 to 10, with lower scores indicating better physical function. A negative value in BASFI change from Baseline indicates an improvement from Baseline. The higher the negative value the better the improvement.

Change From Baseline in the Spine Ankylosing Spondylitis Spine Magnetic Resonance Imaging (MRI) Scoring System for Disease Activity (ASspiMRI-a) in the Berlin Modification at Week 12From Baseline to Week 12

The Berlin modification of the ASspiMRI-a is a scoring system with a concentration on Short-Tau-Inversion Recovery (STIR) sequences without other fat saturation techniques. It quantifies changes in 23 Vertebral Units (VU) of the spine. A VU is defined as the region between 2 virtual lines through the middle of each vertebra. Active inflammation is scored by grading the degree of bone marrow edema from 0 to 3 in 1 dimension on 1 or more consecutive slices that represent the highest level of inflammation in a particular VU. Total spine ASspiMRI-a score in the Berlin modification can range from 0 to 69 with higher scores indicating higher disease activity. A negative value in total spine ASspiMRI-a score change from Baseline indicates an improvement from Baseline. The higher the negative value the higher the reduction of inflammation.

Change From Baseline in the Bath Ankylosing Spondylitis Functional Index (BASFI) at Week 12From Baseline to Week 12

The BASFI assesses physical function in comprising 10 items relating to activities during the past week. Each item ranges from 0 ("Easy") to 10 ("Impossible"). The BASFI is the mean of the 10 scores such that the total score ranges from 0 to 10, with lower scores indicating better physical function. A negative value in BASFI change from Baseline indicates an improvement from Baseline. The higher the negative value the better the improvement.

Change From Baseline in the Bath Ankylosing Spondylitis Disease Activity Index (BASDAI) at Week 12From Baseline to Week 12

The BASDAI is a validated self-reported instrument which consists of six 10 unit horizontal Numerical Rating Scales (NRSs) to measure severity of fatigue, spinal and peripheral joint pain and swelling, enthesitis, and morning stiffness (both severity and duration, respectively) over the last week. The final BASDAI score ranges from 0 to 10, with lower scores indicating lower disease activity. A negative value in BASDAI change from Baseline indicates an improvement from Baseline. The higher the negative value the better the improvement.

Change From Baseline in the Bath Ankylosing Spondylitis Metrology Index (BASMI) at Week 24From Baseline to Week 24

The BASMI characterizes the spinal mobility of subjects with axial SpA and AS. It is a disease-specific measure consisting of 5 clinical measures to reflect subject axial status: cervical rotation; tragus to wall distance; lateral lumbar flexion; lumbar flexion (modified Schober test); intermalleolar distance. According to the linear definition of the BASMI a score of 0 to 10 is calculated for each item based on the measurement. The mean of the sum of the 5 scores provides the BASMI score. The higher the BASMI score the more severe the patient's limitation of movement due to their axial SpA. A negative value in BASMI change from Baseline indicates an improvement from Baseline. The higher the negative value the better the improvement.

Trial Locations

Locations (104)

964

🇺🇸

Hagerstown, Maryland, United States

975

🇺🇸

Dallas, Texas, United States

907

🇨🇦

Victoria, British Columbia, Canada

987

🇺🇸

Tucson, Arizona, United States

954

🇺🇸

Peoria, Arizona, United States

971

🇺🇸

Scottsdale, Arizona, United States

973

🇺🇸

Los Angeles, California, United States

974

🇺🇸

La Jolla, California, United States

966

🇺🇸

Palm Desert, California, United States

957

🇺🇸

Aventura, Florida, United States

962

🇺🇸

Fort Lauderdale, Florida, United States

990

🇺🇸

Pinellas Park, Florida, United States

977

🇺🇸

Cleveland, Ohio, United States

959

🇺🇸

Orange Park, Florida, United States

958

🇺🇸

Vero Beach, Florida, United States

969

🇺🇸

Eagan, Minnesota, United States

984

🇺🇸

Flowood, Mississippi, United States

965

🇺🇸

Florissant, Missouri, United States

950

🇺🇸

Saint Louis, Missouri, United States

963

🇺🇸

Asheville, North Carolina, United States

985

🇺🇸

Brooklyn, New York, United States

951

🇺🇸

Middleburg Heights, Ohio, United States

972

🇺🇸

Duncansville, Pennsylvania, United States

968

🇺🇸

Seattle, Washington, United States

701

🇦🇷

Buenos Aires, Argentina

910

🇨🇦

Windsor, Ontario, Canada

704

🇦🇷

Buenos Aires, Argentina

705

🇦🇷

Cordoba, Argentina

702

🇦🇷

San Miguel de Tucuman, Argentina

709

🇦🇷

La Plata, Argentina

710

🇦🇷

San Juan, Argentina

706

🇦🇷

Rosario, Argentina

708

🇦🇷

San Miguel de Tucuman, Argentina

153

🇧🇪

Brussels, Belgium

152

🇧🇪

Gent, Belgium

151

🇧🇪

Liege, Belgium

903

🇨🇦

Winnipeg, Manitoba, Canada

750

🇧🇷

Curitiba, Brazil

756

🇧🇷

Sao Paulo, Brazil

761

🇧🇷

Goiânia, Brazil

760

🇧🇷

Campinas, Brazil

902

🇨🇦

Sainte Foy, Quebec, Canada

501

🇨🇿

Hlucin, Czechia

504

🇨🇿

Brno, Czechia

500

🇨🇿

Pardubice, Czechia

200

🇫🇷

Boulogne-Billan Court, France

502

🇨🇿

Praha 2, Czechia

505

🇨🇿

Terezin, Czechia

503

🇨🇿

Zlin, Czechia

201

🇫🇷

Lille, France

205

🇫🇷

Limoges, France

202

🇫🇷

Tours, France

206

🇫🇷

Montpellier, France

204

🇫🇷

Paris, France

257

🇩🇪

Berlin, Germany

258

🇩🇪

Berlin, Germany

250

🇩🇪

Herne, Germany

254

🇩🇪

Hamburg, Germany

255

🇩🇪

Freiburg, Germany

260

🇩🇪

München, Germany

253

🇩🇪

Leipzig, Germany

303

🇭🇺

Budapest, Hungary

306

🇭🇺

Miskolc, Hungary

263

🇩🇪

München, Germany

256

🇩🇪

Ratingen, Germany

305

🇭🇺

Budapest, Hungary

352

🇮🇹

Ancona, Italy

300

🇭🇺

Veszprém, Hungary

351

🇮🇹

Firenze, Italy

401

🇳🇱

Maastricht, Netherlands

350

🇮🇹

Pisa, Italy

458

🇵🇱

Bialystok, Poland

400

🇳🇱

Rotterdam, Netherlands

452

🇵🇱

Dabrowka, Poland

455

🇵🇱

Elblag, Poland

459

🇵🇱

Gdanks, Poland

550

🇪🇸

Mérida, Spain

457

🇵🇱

Krakow, Poland

450

🇵🇱

Lublin, Poland

454

🇵🇱

Poznan, Poland

453

🇵🇱

Torun, Poland

456

🇵🇱

Warszawa, Poland

552

🇪🇸

Santiago de Compostela, Spain

462

🇵🇱

Warszawa, Poland

605

🇬🇧

Barnsley, United Kingdom

554

🇪🇸

Santander, Spain

553

🇪🇸

Sevilla, Spain

600

🇬🇧

Leeds, United Kingdom

602

🇬🇧

London, United Kingdom

700

🇦🇷

Buenos Aires, Argentina

802

🇲🇽

Cuernavaca, Mexico

601

🇬🇧

Salford, United Kingdom

302

🇭🇺

Debrecen, Hungary

953

🇺🇸

Tuscaloosa, Alabama, United States

900

🇨🇦

St. John's, Newfoundland and Labrador, Canada

801

🇲🇽

Monterrey, Mexico

970

🇺🇸

Oklahoma City, Oklahoma, United States

982

🇺🇸

Portland, Oregon, United States

961

🇺🇸

Birmingham, Alabama, United States

952

🇺🇸

San Diego, California, United States

978

🇺🇸

Houston, Texas, United States

983

🇺🇸

Houston, Texas, United States

967

🇺🇸

San Antonio, Texas, United States

981

🇺🇸

Salt Lake City, Utah, United States

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