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Study to Assess Adverse Events and How Intravenously (IV) Infused Telisotuzumab Adizutecan (ABBV-400) Moves Through the Body of Adult Participants With Unresectable Locally Advanced/Metastatic Colorectal Cancer

Phase 1
Recruiting
Conditions
Colorectal Cancer
Interventions
Registration Number
NCT06464692
Lead Sponsor
AbbVie
Brief Summary

Colorectal cancer (CRC) is the third most common type of cancer diagnosed worldwide and in China. The purpose of this study is to assess adverse events and how telisotuzumab adizutecan moves through the body of adult participants with unresectable locally advanced/metastatic CRC.

Telisotuzumab adizutecan is an investigational drug being developed for the treatment of CRC. Study doctors put the participants in cohorts called treatment arms. Each treatment arm receives a different dose of telisotuzumab adizutecan. This study will include a dose escalation phase followed by a dose expansion phase. Up to approximately 30 adult participants with unresectable locally advanced/metastatic CRC, will be enrolled in the study in approximately 8 sites in China.

In the dose escalation arms, participants will receive escalating doses of intravenously (IV) infused telisotuzumab adizutecan dose A or B. In dose expansion arm part 1, participants will receive dose A of IV infused telisotuzumab adizutecan. In dose expansion arm part 2, participants will receive the dose C of IV infused telisotuzumab adizutecan. The total study duration will be approximately 2.5 years.

There may be higher treatment burden for participants in this trial compared to their standard of care. Participants will attend regular visits during the study at an approved institution (hospital or clinic). The effect of the treatment will be frequently checked by medical assessments, blood tests, questionnaires and side effects.

Detailed Description

Not available

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
30
Inclusion Criteria
  • Eastern Cooperative Oncology Group (ECOG) Performance Status (PS) of 0 or 1.

  • Has histologically or cytologically confirmed unresectable advanced/metastatic colorectal cancer (mCRC).

  • Has measurable disease per response evaluation criteria in solid tumors (RECIST) v1.1.

  • Does not harbor the BRAF V600E mutation and is not deficient mismatch repair (dMMR)+/microsatellite instability (MSI)-High.

  • Stage 2 only:

    • Archival or recently obtained tumor material must be submitted for assessment of c-Met protein levels by an AbbVie designated IHC laboratory during the pre-screening period. Tumor material from the primary tumor site and/or metastatic sites are allowed. If archival tissue is negative for c-Met protein expression with 3+ intensity, >= 10% tumor cells, recently obtained biopsy material may be submitted for reassessment of c-Met protein expression with 3+ intensity, >= 10% tumor cells.
Exclusion Criteria
  • History (within 6 months) of congestive heart failure (defined as New York Heart Association, Class 2 or higher), ischemic cardiovascular event, cardiac arrhythmia requiring pharmacological or surgical intervention, pericardial effusion, or pericarditis.

  • Prior systemic regimen containing c-Met protein targeting antibody (e.g., amivantamab-vmjw, ABT-700) or define: antibody-drug conjugate (ADC). Tyrosine kinase inhibitors (TKIs) of Met protein are allowed.

  • History of Interstitial lung disease (ILD)/pneumonitis that required treatment with systemic steroids, or any evidence of active ILD/pneumonitis on screening chest computed tomography (CT) scan.

  • History of idiopathic pulmonary fibrosis, organizing pneumonia (e.g., bronchiolitis obliterans), drug-induced pneumonitis, or idiopathic pneumonitis.

  • History of clinically significant, intercurrent lung-specific illnesses including, but not limited to:

    • Underlying pulmonary disorder (i.e., pulmonary emboli within 3 months of the study enrollment, severe asthma, severe chronic obstructive pulmonary disease [COPD], restrictive lung disease, pleural effusion, dependence on supplemental oxygen, etc.)
    • Any autoimmune, connective tissue or inflammatory disorders with documented or suspicious pulmonary involvement at screening (i.e., rheumatoid arthritis, Sjogren's, sarcoidosis, etc.) and prior pneumonectomy.
  • No resolution of any acute clinically significant treatment-related toxicity from prior therapy to Grade <= 1 prior to study entry, except for neutropenia (Grade <= 2), peripheral neuropathy (Grade <= 2), and alopecia (any grade).

  • Untreated brain or meningeal metastases (i.e., participants with history of metastases are eligible provided they do not require ongoing steroid treatment for cerebral edema and have shown clinical and radiographic stability for at least 14 days after definitive therapy).

  • History of other malignancies within 5 years prior to screening, except for malignancies with a negligible risk of metastasis or death (e.g., 5-year Overall Survival [OS] rate > 90%).

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
Safety Run-In Cohort 1: Telisotuzumab Adizutecan Dose ATelisotuzumab AdizutecanParticipants with unresectable locally advanced/metastatic colorectal cancer (CRC) will receive telisotuzumab adizutecan dose A during the approximately 2.5 year study duration.
Safety Run-In Cohort 2: Telisotuzumab Adizutecan Dose BTelisotuzumab AdizutecanParticipants with unresectable locally advanced/metastatic CRC will receive telisotuzumab adizutecan dose B during the approximately 2.5 year study duration.
Dose Expansion Part 1: Telisotuzumab Adizutecan Dose ATelisotuzumab AdizutecanParticipants with unresectable locally advanced/metastatic CRC will receive telisotuzumab adizutecan dose A during the approximately 2.5 year study duration.
Dose Expansion Part 2: Telisotuzumab Adizutecan Dose CTelisotuzumab AdizutecanIf further analysis is warranted, participants with unresectable locally advanced/metastatic CRC will receive telisotuzumab adizutecan dose C during the approximately 2.5 year study duration.
Primary Outcome Measures
NameTimeMethod
Dose-Limiting Toxicity (DLT) of Telisotuzumab Adizutecan in Stage 1Up to 24 Months

DLTs are defined as grade \>= 3 thrombocytopenia that cannot clinically improve after adequate medical treatment/support, febrile neutropenia grade \>= 3 or grade 4 neutropenia that cannot clinically improve after adequate medical treatment/support, and any grade 2 or higher interstitial lung disease (ILD)/pneumonitis that cannot clinically improve after adequate medical treatment/support.

Maximum observed plasma or serum concentration (Cmax) of Telisotuzumab Adizutecan ConjugateUp to 24 Months

Cmax of telisotuzumab adizutecan conjugate.

Time to Cmax (Tmax) of Telisotuzumab Adizutecan ConjugateUp to 24 Months

Tmax of telisotuzumab adizutecan conjugate.

Area Under the Concentration-Time Curve (AUC) of Telisotuzumab Adizutecan ConjugateUp to 24 Months

AUC of telisotuzumab adizutecan conjugate.

Total Antibody of Telisotuzumab AdizutecanUp to 24 Months

Total antibody of telisotuzumab adizutecan.

Unconjugated Payload of Telisotuzumab AdizutecanUp to 24 Months

Unconjugated payload of telisotuzumab adizutecan.

Secondary Outcome Measures
NameTimeMethod
Objective Response (OR)Up to 24 Months

OR as assessed by the Investigator: Confirmed complete response (CR) or confirmed partial response (PR) as assessed by the Investigator per Response Evaluation Criteria in Solid Tumors (RECIST), version 1.1.

Best Overall Response (BOR)Up to 24 Months

Disease control as assessed by the Investigator: BOR of confirmed CR or confirmed PR, or stable disease based on RECIST, version 1.1.

Progression-Free Survival (PFS)Up to 24 Months

PFS as assessed by Investigator: PFS is defined as the time from the participant's first dose of study treatment until radiographic progression or death from any cause, whichever occurs first.

Duration of Response (DoR)Up to 24 Months

DoR as assessed by Investigator: DoR is defined as the time from the participantt's initial response (CR or PR) to the first occurrence of radiographic progression or death from any cause.

Overall Survival (OS)Up to 24 Months

OS is defined as the time from the participant's first dose of study treatment until death from any cause.

Trial Locations

Locations (8)

The First Affiliated Hospital of Nanchang University /ID# 263193

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Nanchang, Jiangxi, China

Beijing Cancer Hospital /ID# 263297

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Beijing, Beijing, China

The Sixth Affiliated Hospital of Sun Yat-sen University /ID# 263309

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Guangzhou, Guangdong, China

Harbin Medical University Cancer Hospital /ID# 263049

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Harbin, Heilongjiang, China

Henan Cancer Hospital /ID# 263172

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Zhengzhou, Henan, China

Hubei Cancer Hospital /ID# 263248

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Wuhan, Hubei, China

First Affiliated Hospital of China Medical University /ID# 263338

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Shenyang, Liaoning, China

The Second Affiliated Hospital of Zhejiang University School of Medicine /ID# 263094

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Hangzhou, Zhejiang, China

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