MedPath

A Study to Investigate the Efficacy and Safety of Verekitug (UPB-101) in Adult Participants With Severe Asthma (VALIANT)

Phase 2
Recruiting
Conditions
Severe Asthma
Interventions
Drug: Verekitug (UPB-101)
Drug: Placebo
Registration Number
NCT06196879
Lead Sponsor
Upstream Bio Inc.
Brief Summary

The purpose of this study is to evaluate the efficacy and safety of verekitug (UPB-101) in participants with severe asthma. The study will evaluate the incidence of asthma exacerbations, other pharmacodynamic (PD) parameters such as lung function and asthma control, and the safety and tolerability of verekitug (UPB-101) compared to placebo.

Detailed Description

This is a multicenter, randomized, placebo-controlled, parallel group study to assess the efficacy and safety of verekitug (UPB-101) administered subcutaneously (SC). A total of approximately 436 adult participants with severe asthma are planned for enrolment and will be randomized in a 1:1:1:1 ratio to receive verekitug (UPB-101) at doses of 100 mg every 12 weeks (Q12W), 400 mg every 24 weeks (Q24W), and 100 mg every 24 weeks (Q24W), or placebo administered SC. In order to maintain the blinding of different doses, all participants will receive 2 SC injections at each dosing visit. This study consists of a Screening/Run-In Period (approximately 4 weeks), Treatment Period (up to 60 weeks with a minimum of 24 weeks) and Follow-up Period (ending approximately 16 weeks after the last administration of study intervention).

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
436
Inclusion Criteria
  • Signed, dated, and received a copy of the Institutional Review Board (IRB)/Independent Ethics Committee (IEC)-approved written informed consent form (ICF).
  • Age 18 to 80 years of age (inclusive) at the time of consent.
  • Physician-diagnosed asthma for at least 12 months prior to Visit 1.
  • Participant has evidence of bronchodilator (BD) reversibility as documented by either historical reversibility (within 12 months prior to study entry) or reversibility during screening.
  • Documented treatment with a total daily dose of either medium or high dose inhaled corticosteroids (ICS) for at least 3 months. Participants on medium dose ICS must also have been taking at least one additional maintenance asthma controller medication for at least 3 months.
  • Documented history of asthma exacerbation(s) within 12 months of Visit 1.
  • Asthma Control Questionnaire-6 (ACQ-6) score greater than or equal to (>=) 1.5 at screening and randomization.
  • Participant must have a pre-BD FEV1 value of >=30 percent (%) and <=80% predicted at Screening.
  • Minimum compliance with daily diary and background asthma medication(s) as captured in the daily diary during the Run-in Period.
  • Agrees to follow the required contraceptive techniques/methods.
  • Female or male participant agrees not to donate eggs or sperm, respectively, for a period of 120 days after the last dose of the study drug intervention or at the Final Visit, whichever occurs last.
Exclusion Criteria
  • Inpatient hospitalization due to asthma at any time within 4 weeks prior to Visit 1 or during the Screening/Run-in Period.
  • Previous exposure to verekitug (UPB-101) or known allergy/sensitivity to any of its excipients.
  • Previous biologics, including those for asthma treatment, for which the appropriate washout period is not fulfilled prior to Visit 1. If the half-life is not known, a 24-week washout period prior to Visit 1 should be applied.
  • Allergen immunotherapy (unless maintenance dose) within 12 weeks prior to Visit 1 or plans to begin therapy or change dosing during the study.
  • For participants taking oral corticosteroids (OCS), the dose has not been stable for at least 2 weeks prior to Visit 1 and/or is >10 milligram (mg) daily, or >20 mg every other day.
  • Evidence of active or suspected bacterial, viral, fungal, or parasitic infections within 2 weeks prior to Visit 1.
  • History compatible with or diagnosis of a parasitic infection and has not been treated or has not responded to standard of care therapy.
  • Current tobacco smokers, nicotine vapers (including electronic cigarettes), snuff users or participants with a smoking history >=10 pack years. (Former nicotine smokers with a smoking history of <10 pack years, former nicotine vapers and former snuff users must have stopped for at least 6 months prior to Visit 1 to be eligible).
  • Positive coronavirus disease 2019 (COVID-19) test with lower respiratory tract symptoms within 28 days before Visit 1.
  • Pregnant or breastfeeding or planning to become pregnant or breastfeed during the study or unwilling to use adequate birth control, if of reproductive potential and sexually active.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Verekitug (UPB-101): 100 mg Q12W / PlaceboVerekitug (UPB-101)Participants will receive 0.5 milliliter (mL) of verekitug (UPB-101) formulated solution (containing 100 milligrams \[mg\] of verekitug \[UPB-101\]) and 2.0 mL of placebo subcutaneously in two separate injections every 12 weeks up to Week 48.
Verekitug (UPB-101): 100 mg Q12W / PlaceboPlaceboParticipants will receive 0.5 milliliter (mL) of verekitug (UPB-101) formulated solution (containing 100 milligrams \[mg\] of verekitug \[UPB-101\]) and 2.0 mL of placebo subcutaneously in two separate injections every 12 weeks up to Week 48.
Verekitug (UPB-101): 400 mg Q24W / PlaceboVerekitug (UPB-101)Participants will receive 2.0 mL of verekitug (UPB-101) formulated solution (containing 400 mg of verekitug \[UPB-101\]) and 0.5 mL of placebo subcutaneously in two separate injections every 24 weeks up to Week 48. Participants will also receive 2 mL and 0.5 mL of placebo subcutaneously in two separate injections at Weeks 12 and 36 visits.
PlaceboPlaceboParticipants will receive 0.5 mL of matching placebo and 2.0 mL of matching placebo subcutaneously in two separate injections every 12 weeks up to Week 48.
Verekitug (UPB-101): 100 mg Q24W / PlaceboPlaceboParticipants will receive 0.5 mL of verekitug (UPB-101) formulated solution (containing 100 mg of verekitug \[UPB-101\]) and 2.0 mL of placebo subcutaneously in two separate injections every 24 weeks up to Week 48. Participants will also receive 2 mL and 0.5 mL of placebo subcutaneously in two separate injections at Weeks 12 and 36 visits.
Verekitug (UPB-101): 400 mg Q24W / PlaceboPlaceboParticipants will receive 2.0 mL of verekitug (UPB-101) formulated solution (containing 400 mg of verekitug \[UPB-101\]) and 0.5 mL of placebo subcutaneously in two separate injections every 24 weeks up to Week 48. Participants will also receive 2 mL and 0.5 mL of placebo subcutaneously in two separate injections at Weeks 12 and 36 visits.
Verekitug (UPB-101): 100 mg Q24W / PlaceboVerekitug (UPB-101)Participants will receive 0.5 mL of verekitug (UPB-101) formulated solution (containing 100 mg of verekitug \[UPB-101\]) and 2.0 mL of placebo subcutaneously in two separate injections every 24 weeks up to Week 48. Participants will also receive 2 mL and 0.5 mL of placebo subcutaneously in two separate injections at Weeks 12 and 36 visits.
Primary Outcome Measures
NameTimeMethod
Annual Asthma Exacerbation Rate (AAER)Baseline up to Week 60

An asthma exacerbation is defined as a worsening of asthma that required treatment with systemic (oral or intravenous) corticosteroids for at least three consecutive days or a single depo-injectable dose of corticosteroids or an emergency room (ER) or urgent care visit that required systemic corticosteroids or an admission to an inpatient facility and/or evaluation and treatment in a healthcare facility for greater than or equal to 24 hours.

Secondary Outcome Measures
NameTimeMethod
Change from Baseline in Forced Expiratory Volume in 1 Second (FEV1) of Pre-bronchodilator (Pre-BD) to Week 60Baseline to Week 60

Spirometry will be performed pre-bronchodilator (BD) to measure lung function. FEV1 is the maximal volume of air exhaled in the first second of a forced expiration from a position of full inspiration.

Change from Baseline in Asthma Control Questionnaire-6 (ACQ-6) to Week 60Baseline to Week 60

ACQ-6 is a participant-reported questionnaire to assess asthma control with 6 items assessing night-time waking, symptoms on waking, activity limitation, shortness of breath, wheeze, and rescue short-acting beta agonist use. Questions are weighted equally and scored from 0 (totally controlled) to 6 (severely uncontrolled). The ACQ-6 score is the mean of the responses.

Number of Participants with Treatment Emergent Adverse Events (TEAEs) and Serious TEAEsUp to Week 64

An AE is any untoward medical occurrence in a participant who received study drug without regard to possibility of causal relationship. SAE is an AE resulting in any of the following outcomes or deemed significant for any other reason: death; initial or prolonged inpatient hospitalization; life-threatening experience (immediate risk of dying); persistent or significant disability/incapacity; congenital anomaly.

Change from Baseline in Fractional exhaled nitric oxide (FeNO) to Week 60Baseline to Week 60

Standardized single breath FeNO test is performed to evaluate airway inflammation.

Trial Locations

Locations (148)

Fundacion Cidea

🇦🇷

Caba, Argentina

InAER

🇦🇷

Caba, Argentina

Toronto Allergists

🇨🇦

Toronto, Ontario, Canada

Winchester Hospital

🇨🇦

Winchester, Ontario, Canada

CIMER

🇨🇱

Providencia, Chile

Sociedad medica Sy G Limitada

🇨🇱

Santiago, Chile

UOSD Allergologia e Immunodeficienze dell'A.O.U. Federico II

🇮🇹

Napoli, Italy

Fondazione IRCCS Policlinico "San Matteo" - SC Pneumologia'

🇮🇹

Pavia, Italy

KKR Sapporo Medical Center

🇯🇵

Sapporo, Hokkaido, Japan

Oji General Hospital

🇯🇵

Tomakomai, Hokkaido, Japan

RCMS/Lungenpraxis Hohenzollerndamm

🇩🇪

Berlin, Germany

AllerVie Clinical Research

🇺🇸

Birmingham, Alabama, United States

Kern Research, Inc.

🇺🇸

Bakersfield, California, United States

Velocity Clinical Research - Lafayette LA

🇺🇸

Los Angeles, California, United States

Newport Native MD Inc

🇺🇸

Newport Beach, California, United States

California Medical Research Associates Inc.

🇺🇸

Northridge, California, United States

Integrated Research of Inland Inc

🇺🇸

Upland, California, United States

Allergy & Asthma Clinical Research

🇺🇸

Walnut Creek, California, United States

Allianz Research Institute

🇺🇸

Westminster, California, United States

Woodland Clinic Medical Group

🇺🇸

Woodland, California, United States

National Jewish Health

🇺🇸

Denver, Colorado, United States

Advance Pharma Research

🇺🇸

Cutler Bay, Florida, United States

Unique Clinical Trials

🇺🇸

Doral, Florida, United States

Health and Life Research Institute, LLC

🇺🇸

Miami, Florida, United States

Phoenix Medical Research

🇺🇸

Miami, Florida, United States

Research Institute of South Florida

🇺🇸

Miami, Florida, United States

Nouvelle Clinical Research

🇺🇸

Miami, Florida, United States

Anderson Allergy And Asthma, PA

🇺🇸

Orlando, Florida, United States

Edward Jenner Research Group, LLC

🇺🇸

Plantation, Florida, United States

R&B Medical Center

🇺🇸

Tampa, Florida, United States

Clinical Site Partners dba Flourish research

🇺🇸

Winter Park, Florida, United States

Clinical Site Partners, LLC dba Flourish Research

🇺🇸

Winter Park, Florida, United States

Pivotal Research Solutions

🇺🇸

Stonecrest, Georgia, United States

RNA America Health Sciences

🇺🇸

Sugar hill, Georgia, United States

Treasure Valley Medical Research

🇺🇸

Boise, Idaho, United States

Velocity Clinical Research - Meridian

🇺🇸

Meridian, Idaho, United States

Howard County Center for Lung and Sleep Medicine LLC

🇺🇸

Columbia, Maryland, United States

Chesapeake Clinical Research Inc

🇺🇸

White Marsh, Maryland, United States

Exordia Medical Research Inc

🇺🇸

Fall River, Massachusetts, United States

Pulmonary Research Institute of Southeast Michigan

🇺🇸

Farmington Hills, Michigan, United States

AA Medical Research Center

🇺🇸

Flint, Michigan, United States

Mayo Clinic

🇺🇸

Rochester, Minnesota, United States

M3 Wake Research

🇺🇸

Las Vegas, Nevada, United States

Urban Health Plan INC

🇺🇸

Bronx, New York, United States

Advanced Respiratory and Sleep Medicine LLC

🇺🇸

Huntersville, North Carolina, United States

Summit Research Group LLC

🇺🇸

Munroe Falls, Ohio, United States

Toledo Institute of Clinical Research Inc

🇺🇸

Toledo, Ohio, United States

OK Clinical Research, LLC

🇺🇸

Edmond, Oklahoma, United States

Velocity Clinical Research - Medford

🇺🇸

Medford, Oregon, United States

Velocity Clinical Research - Anderson

🇺🇸

Anderson, South Carolina, United States

WR-Notus Clinical Research, LLC

🇺🇸

Charleston, South Carolina, United States

Velocity Clinical Research - Spartanburg

🇺🇸

Spartanburg, South Carolina, United States

WR-ClinSearch, LLC

🇺🇸

Chattanooga, Tennessee, United States

Horizon Clinical Research

🇺🇸

Cypress, Texas, United States

Alina Clinical Trials, LLC

🇺🇸

Dallas, Texas, United States

AARA Research Center

🇺🇸

Dallas, Texas, United States

El Paso Pulmonary Association

🇺🇸

El Paso, Texas, United States

Greater Houston Memorial Pulmonary and Sleep

🇺🇸

Houston, Texas, United States

Metroplex Pulmonary and Sleep Center Drive

🇺🇸

McKinney, Texas, United States

Element Research Group

🇺🇸

San Antonio, Texas, United States

DM Clinical Tomball

🇺🇸

Tomball, Texas, United States

Velocity Clinical Research

🇺🇸

West Jordan, Utah, United States

University of Wisconsin--Madison

🇺🇸

Madison, Wisconsin, United States

Centro de Medicina Respiratoria

🇦🇷

Concepción Del Uruguay, Entre Rios, Argentina

Fundacion Scherbovsky

🇦🇷

Ciudad de Mendoza, Mendoza, Argentina

Fundacion Estudios Clinicos (FECLIN)

🇦🇷

Rosario, Santa Fe, Argentina

Instituto Especialidades de la Salud Rosario

🇦🇷

Rosario, Santa Fe, Argentina

Office of Hector H. Altieri MD

🇦🇷

San Miguel De Tucumán, Tucumán, Argentina

Investigaciones En Patologias Respiratorias

🇦🇷

San Miguel De Tucumán, Tucumán, Argentina

CARE: Centro de Alergia y Enfermedades Respiratorias

🇦🇷

Ciudad Autónoma de Buenos Aires, Argentina

Fundacion Respirar - Centro Medico Dra. De Salvo

🇦🇷

Ciudad Autónoma de Buenos Aires, Argentina

Centro Dr. Lazaro Langer Privado Medicina del Aparato Respiratorio

🇦🇷

Córdoba, Argentina

INSARES

🇦🇷

Mendoza, Argentina

Centro Medico Dharma

🇦🇷

Mendoza, Argentina

MHAT "Rahila Angelova" Pernik

🇧🇬

Pernik, Bulgaria

UMHAT Sveti Georgi

🇧🇬

Plovdiv, Bulgaria

Ambulatory For Specialized Outpatient Medical Care - Individual Practice - Dr. Nikolay Evgeniev Ruse Ltd

🇧🇬

Ruse, Bulgaria

Medical Center Excelsior

🇧🇬

Sofia, Bulgaria

Medical Center HERA EOOD

🇧🇬

Sofia, Bulgaria

DCC Convex

🇧🇬

Sofia, Bulgaria

Medconsult Pleven

🇧🇬

Sofia, Bulgaria

Medical center Pulmovizhyn

🇧🇬

Sofia, Bulgaria

Medical Center New Rehabilitation Center EOOD

🇧🇬

Stara Zagora, Bulgaria

MC Zdrave 1

🇧🇬

Vratsa, Bulgaria

Dynamic Drug Advancement

🇨🇦

Ajax, Ontario, Canada

Ottawa Allergy Research Corp

🇨🇦

Ottawa, Ontario, Canada

Fundacion Medica San Cristobal

🇨🇱

Santiago, Metropolitana, Chile

Icegclinic

🇨🇱

Santiago, Region Metropolitana, Chile

Centro Médico BIOREUMA

🇨🇱

Concepción, Chile

Fakultni Nemocnice u Sv. Anny v Brne

🇨🇿

Brno, Czech Republic, Czechia

Alergologie a imunologie Hofstetr Alois MUDr. s.r.o.

🇨🇿

Jihlava, Czech Republic, Czechia

Plicni Stredisko Teplice S.R.O

🇨🇿

Teplice, Czech Republic, Czechia

PNEUMOLOGIE VARNSDORF s.r.o.

🇨🇿

Varnsdorf, Czech Republic, Czechia

KPPK Studienzentrum

🇩🇪

Koblenz, Rheinland-Pfalz, Germany

POIS Sachsen GmbH

🇩🇪

Leipzig, Sachsen, Germany

Velocity Clinical Research Germany , Berlin

🇩🇪

Berlin, Germany

Pneumologisches Studienzentrum

🇩🇪

Berlin, Germany

ME Clinical Respiratory Research Hamburg GmbH

🇩🇪

Hamburg, Germany

IKF Pneumologie Frankfurt, Clinical Research Center Respiratory Diseases

🇩🇪

Hessen, Germany

IKF Pneumologie GmbH & Co. KG

🇩🇪

Mainz, Germany

SSD Asma Grave e Malattie Rare del Polmone, AOU San Luigi Gonzaga

🇮🇹

Orbassano, Torino, Italy

Ospedale San Martino

🇮🇹

Genova, Italy

Yokohama City University Medical Center

🇯🇵

Yokohama-shi, Kanagawa, Japan

Osaka Habikino Medical Center

🇯🇵

Habikino, Osaka, Japan

Kishiwada City Hospital

🇯🇵

Kishiwada, Osaka, Japan

Tokyo-Eki Center-building Clinic

🇯🇵

Chuo-ku, Tokyo, Japan

Fukuwa Clinics

🇯🇵

Chuo-ku, Tokyo, Japan

National Hospital Organization Ibarakihigashi National Hospital

🇯🇵

Ibaraki, Japan

Osaka Metropolitan University Hospital

🇯🇵

Osaka, Japan

Chungbuk National University Hospital

🇰🇷

Cheongju, Chubgbuk, Korea, Republic of

Eunpyeong St. Marys Hospital

🇰🇷

Seoul, Korea, Korea, Republic of

The Catholic University of Korea, Seoul St. Marys Hospital

🇰🇷

Seoul, Republic of Korea, Korea, Republic of

Soonchunhyang University Bucheon Hospital

🇰🇷

Bucheon, Korea, Republic of

Yeungnam University Hospital

🇰🇷

Daegu, Korea, Republic of

Asan Medical Center

🇰🇷

Seoul, Korea, Republic of

Kyung Hee University Hospital

🇰🇷

Seoul, Korea, Republic of

Seoul National University Hospital

🇰🇷

Seoul, Korea, Republic of

Yonsei University Health System - Severance Hospital

🇰🇷

Seoul, Korea, Republic of

Samsung Medical Center

🇰🇷

Seoul, Korea, Republic of

"ALL-MED" Specjalistyczna Opieka Medyczna. Medyczny Instytut Badawczy

🇵🇱

Wroclaw, Dolnoslaskie Voivodeship, Poland

Lekarze Specjalisci - J. Malolepszy I Partnerzy

🇵🇱

Wroclaw, Dolnoslaskie Voivodeship, Poland

Centrum Badan Klinicznych

🇵🇱

Wrocław, Dolnoslaskie Voivodeship, Poland

Nzoz Atopia

🇵🇱

Krakow, Malopolskie Voivodeship, Poland

Malopolskie Centrum Alergologii

🇵🇱

Krakow, Malopolskie Voivodeship, Poland

Centrum Medyczne All-Med Spolka Komandytowa

🇵🇱

Kraków, Malopolskie Voivodeship, Poland

Alergo-Med Specjalistyczna Przychodnia Lekarska Sp Z O.O.

🇵🇱

Tarnow, Malopolskie Voivodeship, Poland

Prywatny Gabinet Lekarski Malgorzata Pawlukiewicz

🇵🇱

Rzeszow, Podkarpackie Voivodeship, Poland

EMED Centrum Uslug Medycznych

🇵🇱

Rzeszow, Podkarpackie Voivodeship, Poland

Centrum Medycyny Oddechowej, Mroz Spolka Jawna

🇵🇱

Białystok, Podlaskie Voivodeship, Poland

Uniwersyteckie Centrum Kliniczne, Klinika Alergologii i Pneumonologii

🇵🇱

Gdańsk, Pomorskie Voivodeship, Poland

Ostrowieckie Centrum Medyczne spolka cywilna Anna Olech-Cudzik, Krzysztof Cudzik

🇵🇱

Ostrowiec Świętokrzyski, Swietokrzyskie, Poland

Newtown Clinical Research Centre

🇿🇦

Johannesburg, Gauteng, South Africa

Emmed Research

🇿🇦

Pretoria, Gauteng, South Africa

FCRN Clinical Trial Centre

🇿🇦

Vereeniging, Gauteng, South Africa

St Augustine's Hospital/Dr. IA Abdullah

🇿🇦

Durban, KwaZulu Natal, South Africa

University of Cape Town Lung Institute

🇿🇦

Cape Town, Western Cape, South Africa

Synapta Clinical Research Centre

🇿🇦

Durban, South Africa

Giromed Institute

🇪🇸

Girona, Barcelona, Spain

Hospital Gregorio Marañon

🇪🇸

Madrid, Spain

Hull University Teaching Hospitals NHS Trust

🇬🇧

Cottingham, East Yorkshire, United Kingdom

Royal Liverpool University Hospital

🇬🇧

Liverpool, Merseyside, United Kingdom

Ormeau Clinical Trials Ltd

🇬🇧

Belfast, N. Ireland, United Kingdom

Churchill Hospital

🇬🇧

Oxford, Oxfordshire, United Kingdom

Asthma/COPD Clinical Research Centre

🇬🇧

Glasgow, Scotland, United Kingdom

St Peter's Hospital

🇬🇧

Chertsey, Surrey, United Kingdom

Heartlands Hospital, University Hospitals Birmingham NHS Trust

🇬🇧

Birmingham, West Midlands, United Kingdom

Bradford Royal Infirmary

🇬🇧

Bradford, West Yorkshire, United Kingdom

Duckworth Lane Clinical Research Facility

🇬🇧

Bradford, West Yorkshire, United Kingdom

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