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Open-Label Extension Study of Trofinetide for Rett Syndrome

Phase 3
Completed
Conditions
Rett Syndrome
Interventions
Registration Number
NCT04776746
Lead Sponsor
ACADIA Pharmaceuticals Inc.
Brief Summary

To investigate the safety and tolerability of continued long-term treatment with oral trofinetide in girls and women with Rett syndrome

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
Female
Target Recruitment
78
Inclusion Criteria
  1. Has completed the EOT visit of the antecedent trofinetide Study ACP-2566-004 (i.e., has completed 40 weeks)

  2. May benefit from continued treatment with open-label trofinetide in the judgment of the Investigator

  3. Can still swallow the study medication provided as a liquid solution or can take it by gastrostomy tube

  4. The subject's caregiver is English-speaking and has sufficient language skills to complete the caregiver assessments

    Childbearing Potential

  5. Subjects of childbearing potential must abstain from sexual activity for the duration of the study and for at least 30 days thereafter. If a subject is sexually active or becomes sexually active during the study, she must use 2 clinically acceptable methods of contraception (e.g., oral, intrauterine device [IUD], diaphragm plus spermicide, injectable, transdermal or implantable contraception) for the duration of the study and for at least 30 days thereafter. Subject must not be pregnant or breastfeeding.

Exclusion Criteria
  1. Began treatment with growth hormone during the antecedent study
  2. Began treatment with IGF-1 during the antecedent study
  3. Began treatment with insulin during the antecedent study
  4. Has developed a clinically significant cardiovascular, endocrine (such as hypo- or hyperthyroidism, Type 1 diabetes mellitus, or uncontrolled Type 2 diabetes mellitus), renal, hepatic, respiratory, or gastrointestinal disease (such as celiac disease or inflammatory bowel disease)
  5. Subject is judged by the Investigator or the Medical Monitor to be inappropriate for the study due to AEs, medical condition, or noncompliance with investigational product or study procedures in the antecedent study
  6. Has a clinically significant abnormality in vital signs at Baseline
  7. Has an average QTcF interval of >450 ms on the Baseline ECG performed before the first dose of trofinetide is given in the present study (i.e., the ECG performed at the EOT visit of the antecedent study)
  8. Has developed a clinically significant ECG finding during the antecedent study

Additional inclusion/exclusion criteria apply. Patients will be evaluated at screening to ensure that all criteria for study participation are met. Patients may be excluded from the study based on these assessments (and specifically, if it is determined that their baseline health and condition do not meet all pre-specified entry criteria).

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Drug - trofinetidetrofinetidetrofinetide oral solution
Primary Outcome Measures
NameTimeMethod
Percentage of Patients With Treatment-emergent Adverse Events (TEAEs), With Serious Adverse Events (SAEs), and With Withdrawals Due to AEsMean study drug exposure was 426 days, corresponding to 1.2 years

Withdrawals due to AEs included both study drug discontinuation as well as study termination

Number (%) of Patients With Potentially Clinically Important Changes in ECG Post-baselineMean study drug exposure was 426 days, corresponding to 1.2 years

Potentially clinically significant ECG changes were defined as QTcF \>500 ms or QTcF change from baseline (CFB) of \>60 ms

Number (%) of Patients With Potentially Clinically Important Changes in Vital Signs Post-baselineMean study drug exposure was 426 days, corresponding to 1.2 years

Potentially clinically important changes from baseline in vital signs were defined as:

Systolic blood pressure (SBP) ≥180 mmHg and increased ≥20 mmHg from baseline; SBP ≤90 mmHg and decreased ≥20 mmHg from baseline; Diastolic blood pressure (DBP) ≥105 mmHg and increased ≥15 mmHg from baseline; DBP ≤50 mmHg and decreased ≥15 mmHg from baseline; Pulse rate (PR) ≥120 bpm and increased ≥15 bpm from baseline; PR≤50 bpm and decreased ≥15 bpm from baseline. Baseline was the baseline value of previous study ACP-2566-003.

Number (%) of Patients With Potentially Clinically Important Changes in Body Weight Post-baselineMean study drug exposure was 426 days, corresponding to 1.2 years

Potentially clinically important changes from baseline in body weight were defined as:

Weight increase ≥7% from baseline Weight decrease ≥7% from baseline

Number (%) of Patients With Potentially Clinically Important Changes in Laboratory Parameters Post-baselineMean study drug exposure was 426 days, corresponding to 1.2 years

Potentially clinically important changes in laboratory parameters were defined as: sodium ≤125 mmol/L; sodium ≥155 mmol/L; potassium ≤3.0 mmol/L ; potassium ≥5.5 mmol/L; chloride ≤85 mmol/L; chloride ≥120 mmol/L; calcium \<2.0 mmol/L; calcium \>2.75 mmol/L; blood urea nitrogen ≥10.71 mmol/L; creatinine \>1.5× upper limit of normal (ULN); uric acid ≥505.75 μmol/L; lactate dehydrogenase (LDH) ≥3×ULN; glucose ≤2.48 mmol/L; glucose ≥11 mmol/L; albumin ≤26 g/L; albumin ≥60 g/L; protein ≤50 g/L; protein ≥100 g/L; alanine transaminase (ALT) ≥3×ULN; aspartate transaminase (AST) ≥3×ULN; gamma glutamyl transferase (GGT) ≥3×ULN; alkaline phosphatase (ALP) ≥3×ULN; bilirubin ≥1.5×ULN

Secondary Outcome Measures
NameTimeMethod

Trial Locations

Locations (21)

Children's Hospital of Philadelphia

🇺🇸

Philadelphia, Pennsylvania, United States

UC Davis MIND Institute

🇺🇸

Sacramento, California, United States

Rush University Medical Center

🇺🇸

Chicago, Illinois, United States

Texas Children's Hospital

🇺🇸

Houston, Texas, United States

Seattle Children's Hospital

🇺🇸

Seattle, Washington, United States

University of California, San Diego

🇺🇸

La Jolla, California, United States

Children's Hospital Colorado Aurora

🇺🇸

Aurora, Colorado, United States

Kennedy Krieger Institute, John Hopkins School of Medicine

🇺🇸

Baltimore, Maryland, United States

Emory Genetics Clinical Trial Center

🇺🇸

Atlanta, Georgia, United States

Boston Children's Hospital Harvard Medical School

🇺🇸

Boston, Massachusetts, United States

Gillette Children's Specialty Healthcare

🇺🇸

Saint Paul, Minnesota, United States

The University of North Carolina at Chapel Hill

🇺🇸

Chapel Hill, North Carolina, United States

Cleveland Clinic

🇺🇸

Cleveland, Ohio, United States

Translational Genomics Research Institute (TGen)

🇺🇸

Phoenix, Arizona, United States

University of Alabama at Birmingham

🇺🇸

Birmingham, Alabama, United States

Cincinnati Children's Hospital Medical Center

🇺🇸

Cincinnati, Ohio, United States

Vanderbilt University Medical Center

🇺🇸

Nashville, Tennessee, United States

University of South Florida

🇺🇸

Tampa, Florida, United States

Greenwood Genetic Center

🇺🇸

Greenwood, South Carolina, United States

Washington University School of Medicine

🇺🇸

Saint Louis, Missouri, United States

Montefiore Medical Center

🇺🇸

Bronx, New York, United States

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