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Multi-center, Open-label, Phase 1b Study in Patients With Relapsed/Refractory Multiple Myeloma (RRMM)

Phase 1
Completed
Conditions
Multiple Myeloma
Interventions
Registration Number
NCT04045795
Lead Sponsor
Sanofi
Brief Summary

Primary Objectives:

* To evaluate the safety and tolerability of isatuximab administered subcutaneously (SC) versus intravenously (IV)

* To assess the safety and tolerability (including local injection site tolerability) of isatuximab using the (investigational) isatuximab injector device

* To evaluate the pharmacokinetics (PK) of SC and IV isatuximab

Secondary Objectives:

* To estimate absolute bioavailability of SC and IV isatuximab

* To measure receptor occupancy (RO) after isatuximab SC versus IV administration

* To assess efficacy of isatuximab after SC and IV administration

* To assess patient expectations prior to and patient experience and satisfaction after SC administration

* To evaluate potential immunogenicity of SC or IV isatuximab

Detailed Description

Total study duration is variable depending on treatment and follow-up periods, including 21 days of screening, and treatment period until disease progression, unacceptable adverse reaction or other reason for discontinuation. End of treatment will be 30 days after last administration of investigational medicinal product, or before further anti-myeloma therapy, whichever comes first; approximately 14 months after first study treatment administration.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
56
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
Dose regimen 1isatuximab SAR650984 SCIsatuximab SC administration dose level 1 once weekly for 4 weeks (Cycle 1) and on Day 1 and Day 15 of each subsequent cycle
Dose regimen 3Investigational injector deviceIsatuximab SC administration dose level 3 using the investigational injector device once weekly for 4 weeks (Cycle 1) and on Day 1 and Day 15 of each subsequent cycle
Dose regimen 4isatuximab SAR650984 IVIsatuximab IV administration once weekly for 4 weeks (Cycle 1) and on Day 1 and Day 15 of each subsequent cycle
Dose regimen 5dexamethasoneIsatuximab IV administration once weekly for 4 weeks (Cycle 1) and on Day 1 and Day 15 of each subsequent cycle
Dose regimen 3isatuximab SAR650984 SCIsatuximab SC administration dose level 3 using the investigational injector device once weekly for 4 weeks (Cycle 1) and on Day 1 and Day 15 of each subsequent cycle
Dose regimen 5pomalidomideIsatuximab IV administration once weekly for 4 weeks (Cycle 1) and on Day 1 and Day 15 of each subsequent cycle
Dose regimen 2isatuximab SAR650984 SCIsatuximab SC administration dose level 2 once weekly for 4 weeks (Cycle 1) and on Day 1 and Day 15 of each subsequent cycle
Dose regimen 5isatuximab SAR650984 IVIsatuximab IV administration once weekly for 4 weeks (Cycle 1) and on Day 1 and Day 15 of each subsequent cycle
Dose regimen 1pomalidomideIsatuximab SC administration dose level 1 once weekly for 4 weeks (Cycle 1) and on Day 1 and Day 15 of each subsequent cycle
Dose regimen 1dexamethasoneIsatuximab SC administration dose level 1 once weekly for 4 weeks (Cycle 1) and on Day 1 and Day 15 of each subsequent cycle
Dose regimen 2pomalidomideIsatuximab SC administration dose level 2 once weekly for 4 weeks (Cycle 1) and on Day 1 and Day 15 of each subsequent cycle
Dose regimen 2dexamethasoneIsatuximab SC administration dose level 2 once weekly for 4 weeks (Cycle 1) and on Day 1 and Day 15 of each subsequent cycle
Dose regimen 3dexamethasoneIsatuximab SC administration dose level 3 using the investigational injector device once weekly for 4 weeks (Cycle 1) and on Day 1 and Day 15 of each subsequent cycle
Dose regimen 3pomalidomideIsatuximab SC administration dose level 3 using the investigational injector device once weekly for 4 weeks (Cycle 1) and on Day 1 and Day 15 of each subsequent cycle
Dose regimen 4dexamethasoneIsatuximab IV administration once weekly for 4 weeks (Cycle 1) and on Day 1 and Day 15 of each subsequent cycle
Dose regimen 4pomalidomideIsatuximab IV administration once weekly for 4 weeks (Cycle 1) and on Day 1 and Day 15 of each subsequent cycle
Primary Outcome Measures
NameTimeMethod
PK assessment: CtroughBaseline to EOT after isatuximab SC and to Cycle 10 after IV (28 days per Cycle)

Concentration observed just before treatment administration during repeated dosing (Ctrough)

PK assessment: AUClastBaseline to EOT after isatuximab SC and to Cycle 10 after IV (28 days per Cycle)

Area under the plasma concentration versus time curve calculated using the trapezoidal method from time zero to time of the last concentration observed above the lower limit of quantification (ie, Clast) (AUClast)

Assessment of adverse events (AEs)Baseline to 30 days after last study treatment administration (up to approximately 14 months after first study treatment administration)

Number of participants with adverse events

PK assessment: ClastBaseline to EOT after isatuximab SC and to Cycle 10 after IV (28 days per Cycle)

Last concentration observed above the lower limit of quantification after the first infusion (Clast)

Pharmacokinetic (PK) assessment: CeoiBaseline to end of treatment (EOT) after isatuximab SC and to Cycle 10 after IV (28 days per Cycle)

Concentration observed at the end of infusion (Ceoi)

PK assessment: CmaxBaseline to EOT after isatuximab SC and to Cycle 10 after IV (28 days per Cycle)

Maximum concentration observed after the first infusion (Cmax)

PK assessment: tlastBaseline to EOT after isatuximab SC and to Cycle 10 after IV (28 days per Cycle)

Time of Clast (tlast)

PK assessment: AUC0 TBaseline to EOT after isatuximab SC and to Cycle 10 after IV (28 days per Cycle)

Area under the plasma concentration versus time curve calculated over the dosing interval T (168h or 336h) (AUC0 T)

PK assessment: tmaxBaseline to EOT after isatuximab SC and to Cycle 10 after IV (28 days per Cycle)

Time to reach Cmax (tmax)

Secondary Outcome Measures
NameTimeMethod
Overall response rate (ORR)From day -21 to day 60 after last study treatment (up to approximately 14 months after first study treatment administration)

ORR is the proportion of patients with stringent complete response (sCR), complete response (CR), very good partial response (VGPR), and partial response (PR) using the IMWG response criteria

Duration of response (DOR)From day -21 to day 60 after last study treatment (up to approximately 14 months after first study treatment administration)

Time from the date of the first response to the date of first progressive disease (PD) or death, whichever happens first

Time to response (TTR)From day -21 to day 60 after last study treatment (up to approximately 14 months after first study treatment administration)

Time from the date of first study treatment to the first response

Immunogenicity: Anti drug antibody levelsBaseline to EOT after isatuximab SC and to Cycle 10 after IV (28 days per Cycle)

Incidence of patients with anti drug antibodies against isatuximab

Estimation of absolute bioavailability of isatuximabDay 8

Absolute bioavailability of isatuximab SC, expressed as a percentage, estimated from AUC0-168h obtained after intravenous (IV) and extravascular (EV) administration

Clinical benefit rate (CBR)From day -21 to day 60 after last study treatment (up to approximately 14 months after first study treatment administration)

Proportion of patients with sCR, CR, VGPR, PR or minimal response (MR) according to IMWG criteria

Time to progression (TTP)From day -21 to day 60 after last study treatment (up to approximately 14 months after first study treatment administration)

Time from date of first study treatment to date of first documentation of progressive disease

Progression free survival (PFS)From day -21 to day 60 after last study treatment (up to approximately 14 months after first study treatment administration)

Time from date of first study treatment to date of first documentation of progressive disease or death

Comparison of patient expectations and satisfaction: Patient Expectations and Satisfaction QuestionnairesCycles 1 and 2 (28 days per Cycle), and 30 days after last isatuximab administration (up to approximately 14 months after first study treatment administration)

Comparison of patient expectations and satisfaction will be assessed using Patient Expectations and Satisfaction Questionnaires before and after subcutaneous (SC) administration, where a score of 1 = not satisfied and a score of 5 = extremely satisfied

Overall survival (OS)From day -21 to day 60 after last study treatment (up to approximately 14 months after first study treatment administration)

Time from the date of first study treatment to date of death from any cause

Biomarker: Change in CD38 receptor occupancyAt screening and at Day 1 of Cycle 2 (28 days per Cycle) (predose); to be stopped once the isatuximab SC dose has been selected.

Change in CD38 receptor occupancy from baseline

Trial Locations

Locations (14)

Investigational Site Number : 0360004

🇦🇺

Fitzroy, Victoria, Australia

~Banner MD Anderson Cancer Center Site Number : 8400005

🇺🇸

Gilbert, Arizona, United States

Investigational Site Number : 3920002

🇯🇵

Okayama-shi, Okayama, Japan

Investigational Site Number : 0360003

🇦🇺

Richmond, Victoria, Australia

Investigational Site Number : 0560001

🇧🇪

Leuven, Belgium

City of Hope Site Number : 8400002

🇺🇸

Duarte, California, United States

Gabrail Cancer Center Site Number : 8400001

🇺🇸

Canton, Ohio, United States

Investigational Site Number : 0360001

🇦🇺

Wollongong, New South Wales, Australia

Investigational Site Number : 0360002

🇦🇺

Blacktown, New South Wales, Australia

Investigational Site Number : 2500002

🇫🇷

TOULOUSE Cedex 9, France

Investigational Site Number : 2500001

🇫🇷

Nantes, France

Investigational Site Number : 3920001

🇯🇵

Shibuya-ku, Tokyo, Japan

Investigational Site Number : 7240002

🇪🇸

Santander, Cantabria, Spain

Investigational Site Number : 7240001

🇪🇸

Badalona, Catalunya [Cataluña], Spain

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