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Monoclonal Antibody Against PCSK9 to Reduce Elevated LDL-C in Subjects Currently Not Receiving Drug Therapy for Easing Lipid Levels-2

Phase 3
Completed
Conditions
Hyperlipidemia
Interventions
Biological: Placebo to Evolocumab
Biological: Evolocumab
Drug: Ezetimibe
Other: Placebo to Ezetimibe
Registration Number
NCT01763827
Lead Sponsor
Amgen
Brief Summary

The primary objective was to evaluate the effect of 12 weeks of evolocumab subcutaneous (SC) monotherapy every 2 weeks (Q2W) and monthly (QM), compared with placebo and ezetimibe, on percent change from baseline in low-density lipoprotein cholesterol (LDL-C) in adults with a 10-year Framingham risk score of 10% or less.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
615
Inclusion Criteria
  • Male or female ≥ 18 to ≤ 80 years of age
  • National Cholesterol Education Program Adult Treatment Panel III (NCEP ATP III) Framingham risk score of 10% or less
  • Fasting LDL-C ≥ 100 mg/dL (2.6 mmol/L) and <190 mg/dL
  • Fasting triglycerides ≤ 400 mg/dL (4.5 mmol/L)
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Exclusion Criteria
  • History of coronary heart disease
  • New York Heart Association (NYHA) III or IV heart failure
  • Uncontrolled cardiac arrhythmia
  • Uncontrolled hypertension
  • Diabetes mellitus (Type 1 diabetes, poorly controlled type 2 diabetes)
  • Uncontrolled hypothyroidism or hyperthyroidism
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Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Placebo Q2WPlacebo to EvolocumabParticipants received placebo subcutaneous injection once every 2 weeks (Q2W) and placebo tablets once a day for up to 12 weeks.
Placebo Q2WPlacebo to EzetimibeParticipants received placebo subcutaneous injection once every 2 weeks (Q2W) and placebo tablets once a day for up to 12 weeks.
Placebo QMPlacebo to EvolocumabParticipants received placebo subcutaneous injection once every month (QM) and placebo tablets once a day for up to 12 weeks.
Placebo QMPlacebo to EzetimibeParticipants received placebo subcutaneous injection once every month (QM) and placebo tablets once a day for up to 12 weeks.
Ezetimibe (Q2W)Placebo to EvolocumabParticipants received placebo subcutaneous injection once every 2 weeks and 10 mg ezetimibe orally once a day for up to 12 weeks.
Ezetimibe (QM)Placebo to EvolocumabParticipants received placebo subcutaneous injection once a month and 10 mg ezetimibe orally once a day for up to 12 weeks.
Evolocumab Q2WEvolocumabParticipants received 140 mg evolocumab by subcutaneous injection once every 2 weeks and placebo tablets once a day for up to 12 weeks.
Evolocumab Q2WPlacebo to EzetimibeParticipants received 140 mg evolocumab by subcutaneous injection once every 2 weeks and placebo tablets once a day for up to 12 weeks.
Evolocumab QMEvolocumabParticipants received 420 mg evolocumab by subcutaneous injection once a month and placebo tablets once a day for up to 12 weeks.
Evolocumab QMPlacebo to EzetimibeParticipants received 420 mg evolocumab by subcutaneous injection once a month and placebo tablets once a day for up to 12 weeks.
Ezetimibe (QM)EzetimibeParticipants received placebo subcutaneous injection once a month and 10 mg ezetimibe orally once a day for up to 12 weeks.
Ezetimibe (Q2W)EzetimibeParticipants received placebo subcutaneous injection once every 2 weeks and 10 mg ezetimibe orally once a day for up to 12 weeks.
Primary Outcome Measures
NameTimeMethod
Percent Change From Baseline in Low-density Lipoprotein Cholesterol (LDL-C) at Week 12Baseline and Week 12
Percent Change From Baseline in LDL-C at the Mean of Weeks 10 and 12Baseline and Weeks 10 and 12
Secondary Outcome Measures
NameTimeMethod
Percent Change From Baseline in Lipoprotein (a) at the Mean of Weeks 10 and 12Baseline and Weeks 10 and 12
Percent Change From Baseline in Lipoprotein (a) at Week 12Baseline and Week 12
Percent Change From Baseline in Triglycerides at the Mean of Weeks 10 and 12Baseline and Weeks 10 and 12
Change From Baseline in LDL-C at Week 12Baseline and Week 12
Percent Change From Baseline in Non-HDL-C at Week 12Baseline and Week 12
Percent Change From Baseline in Apolipoprotein B at the Mean of Weeks 10 and 12Baseline and Weeks 10 and 12
Percent Change From Baseline in Apolipoprotein B at Week 12Baseline and Week 12
Percent Change From Baseline in Total Cholesterol/High Density Lipoprotein-cholesterol Ratio at the Mean of Weeks 10 and 12Baseline and Weeks 10 and 12
Percent Change From Baseline in Total Cholesterol/High Density Lipoprotein-cholesterol Ratio at Week 12Baseline and Week 12
Percent Change From Baseline in Apolipoprotein B/Apolipoprotein A1 Ratio at the Mean of Weeks 10 and 12Baseline and Weeks 10 and 12
Percent Change From Baseline in Apolipoprotein B/Apolipoprotein A1 Ratio at Week 12Baseline and Week 12
Percent Change From Baseline in Triglycerides at Week 12Baseline and Week 12
Percent Change From Baseline in Very Low Density Lipoprotein Cholesterol (VLDL-C) at the Mean of Weeks 10 and 12Baseline and Weeks 10 and 12
Percent Change From Baseline in VLDL-C at Week 12Baseline and Week 12
Percent Change From Baseline in High-density Lipoprotein Cholesterol (HDL-C) at the Mean of Weeks 10 and 12Baseline and Weeks 10 and 12
Percent Change From Baseline in HDL-C at Week 12Baseline and Week 12
Change From Baseline in LDL-C at the Mean of Weeks 10 and 12Baseline and Weeks 10 and 12
Percentage of Participants Who Achieved a Mean LDL-C at Weeks 10 and 12 of Less Than 70 mg/dLWeeks 10 and 12
Percentage of Participants Who Achieved LDL-C < 70 mg/dL at Week 12Week 12
Percent Change From Baseline in Non-high-density Lipoprotein Cholesterol (Non-HDL-C) at the Mean of Weeks 10 and 12Baseline and Weeks 10 and 12

Trial Locations

Locations (1)

Research Site

🇹🇷

Istanbul, Turkey

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