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BGJ398 for Patients With Tumors With FGFR Genetic Alterations

Phase 2
Terminated
Conditions
Solid Tumor
Hematologic Malignancies
Interventions
Registration Number
NCT02160041
Lead Sponsor
Novartis Pharmaceuticals
Brief Summary

The purpose of this signal seeking study was to determine whether treatment with BGJ398 demonstrates sufficient efficacy in select FGFR pathway-regulated solid tumors and/or hematologic malignancies to warrant further study.

Detailed Description

Not available

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
84
Inclusion Criteria

Patient has a confirmed diagnosis of a select solid tumor (except with a primary diagnosis of Urothelial cell carcinoma, Cholangiocarcinoma, Endometrial cancer, and Glioblastoma multiforme) or hematologic malignancies and is in need of treatment because of progression or relapse.

Patient's tumor has been evaluated and pre-identified as having a tumor with a FGFR genetic alteration. The qualifying alteration must be assessed and reported by a CLIA-certified laboratory.

Patient must have received at least one prior treatment for recurrent, metastatic and /or locally advanced disease and for whom no standard therapy options are anticipated to result in a durable remission.

Patient must have progressive and measurable disease per RECIST 1.1. or other appropriate hematological response criteria.

Patient has an Eastern Cooperative Oncology Group (ECOG) performance status ≤ 1

Exclusion Criteria

Patient has received prior treatment with BGJ398

Patients with Central Nervous System (CNS) metastasis or leptomeningeal carcinomatosis

Patient has received chemotherapy or other anticancer therapy ≤ 4 weeks (6 weeks for nitrosourea, antibodies or mitomycin-C) prior to starting study drug.

Patients with acute or chronic pancreatitis

Patients with impaired cardiac function or clinically significant cardiac diseases

History and/or current evidence of extensive tissue calcification

Use of medications that increase serum levels of phosphorus and/or calcium

Current evidence of corneal or retinal disorder/keratopathy

History and/or current evidence of renal or endocrine alterations of calcium/phosphate homeostasis

Patients with another primary malignancy within 3 years prior to starting study treatment, with the exception of adequately treated basal cell carcinoma, squamous cell carcinoma or other non-melanomatous skin cancer, or in-situ carcinoma of the uterine cervix

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
BGJ398BGJ398BGJ398 was dosed on a flat scale of 125 mg (e.g., 1 x 100 mg and 1 x 25 mg capsules) once daily for the first 21 days of the 28-day cycle (3 weeks on, 1 week off in a cycle). A complete treatment cycle is defined as 28 days.
Primary Outcome Measures
NameTimeMethod
Clinical Benefit Rate (CBR) Associated With BGJ398 Treatment16 weeks

Tumor Response: Overall response rate (ORR) and clinical benefit rate (CBR) for solid tumor (non-lymphoma) which excludes 3 TIO and 1 Lymphoma patients (hence 80 patients and not 84)

Clinical benefit rate for patients with solid tumors were assessed using RECIST 1.1 and include responses of CR or PR or SD. For hematologic tumors other appropriate hematological response criteria may apply

Per Response Evaluation Criteria In Solid Tumors Criteria (RECIST v1.0) for target lesions and assessed by MRI: Complete Response (CR), Disappearance of all target lesions; Partial Response (PR), \>=30% decrease in the sum of the longest diameter of target lesions; Overall Response (OR) = CR + PR

Secondary Outcome Measures
NameTimeMethod
Kaplan-Meier Estimates of Survival Rate, % (95% CI)months 3, 6, 9, 12, 24

Overall survival (OS) is the time from the date of start of treatment to date of death due to any cause. If a patient was not known to have died, survival was censored at the date of last contact.

Progression-Free Survival (PFS)every 8 weeks until death, assessed up to 24 months

Kaplan-Meier estimates of PFS timing, months

Progression free survival (PFS) is defined as the time from the date of first dose to the date of first documented disease progression or relapse or death due to any cause

Overall Survival (OS)every 8 weeks until death, assessed up to 36 months

Overall survival (OS) is defined as the time from the date of first dose to the date of death due to any cause

Overall Response (OR) or Partial Response (PR) or Greaterbaseline and every 8 weeks until disease progression or end of treatment, assessed up to 24 months

The key secondary endpoint, OR, was determined by Investigator assessment for each tumor assessment and defined as responses of CR and PR per RECIST version 1.1.

Per Response Evaluation Criteria In Solid Tumors Criteria (RECIST v1.0) for target lesions and assessed by MRI: Complete Response (CR), Disappearance of all target lesions; Partial Response (PR), \>=30% decrease in the sum of the longest diameter of target lesions; Overall Response (OR) = CR + PR

Kaplan-Meier Estimates of PFS Rate, % (95% CI)Months 1, 2, 3, 4, 5, 6, 12, 18, 24
Number of Participants With 99 Day Minimum Duration of Response (DOR)baseline and every 8 weeks until disease progression or end of treatment, assessed up to 24 months

The duration of response (PR or greater) applies only to patients whose best response was PR or greater. It is defined as the Ttime from the first documented response to the date first documented disease progression or relapse or death due to any cause

Trial Locations

Locations (56)

Alabama Oncology St. Vincent's Birmingham

🇺🇸

Birmingham, Alabama, United States

North County Oncology Medical Clinic Inc

🇺🇸

Oceanside, California, United States

San Francisco General Hospital San Francisco Gen Hosp (7)

🇺🇸

San Francisco, California, United States

Rocky Mountain Cancer Centers Rocky Mountain Cancer Ctr (50)

🇺🇸

Greenwood Village, Colorado, United States

Norwalk Hospital

🇺🇸

Norwalk, Connecticut, United States

Florida Cancer Specialists Florida Cancer Specialists 36

🇺🇸

Fort Myers, Florida, United States

University of Miami Sylvester Comprehensive Cancer

🇺🇸

Miami, Florida, United States

NorthWest Georgia Oncology Centers NW Georgia Oncology

🇺🇸

Marietta, Georgia, United States

Harbin Clinic Medical Oncology Clin. Res.

🇺🇸

Rome, Georgia, United States

Illinois Cancer Specialists

🇺🇸

Arlington Heights, Illinois, United States

Scroll for more (46 remaining)
Alabama Oncology St. Vincent's Birmingham
🇺🇸Birmingham, Alabama, United States

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