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To Investigate the Safety, Tolerability and Pharmacokinetics of AZD2516 After Multiple Dosing in Healthy Volunteers

Phase 1
Completed
Conditions
Part A Healthy Young Males and Non-fertile Female Volunteers Aged 20 to 45 Years.
Part B Healthy Young Males and Non-fertile Female Volunteers Aged 20 to 45 and Elderly Volunteers Aged 60 to 80
Interventions
Drug: Placebo
Registration Number
NCT01148095
Lead Sponsor
AstraZeneca
Brief Summary

AZD2516 is being developed for the oral treatment of chronic neuropathic pain. This study is split in to two parts. Part A will measure the effect of food and a new formulation of the drug in the blood and see how well it is tolerated. Part B will commence after the completion of Part A and will investigate the safety and tolerability of daily dosing with AZD2516.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
6
Inclusion Criteria
  • Have a body mass index (BMI) between 18 and 30 kg/m2 and weigh at least 50 kg and no more than 100 kg
  • Healthy volunteers able and willing to comply with all study requirements.
Exclusion Criteria
  • An ongoing or history of a medical or psychiatric disease/condition which may put the healthy volunteer at risk or interfere with the study objectives because of participation in the study, as judged by the investigator(s).
  • History of psychotic disorder among first degree relatives.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
1AZD2516AZD2516 (dose escalating)
2PlaceboPlacebo
Primary Outcome Measures
NameTimeMethod
Adverse Events, vital signsDay -1 until follow-up
Secondary Outcome Measures
NameTimeMethod
Maximum plasma concentration (Cmax)Day 1 - Day 12
Time to Cmax (tmax)Day 1 - Day 12
Terminal rate constant (λz)Day 1 - Day 12

Trial Locations

Locations (1)

Research Site

🇬🇧

London, United Kingdom

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