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A Study of Once-Daily Oral Orforglipron (LY3502970) in Japanese Adult Participants With Obesity Disease

Phase 3
Active, not recruiting
Conditions
Obesity
Interventions
Drug: Placebo
Registration Number
NCT05931380
Lead Sponsor
Eli Lilly and Company
Brief Summary

The main purpose of this study is to investigate the efficacy and safety of oral orforglipron in participants with obesity disease with obesity-related health problems.

Detailed Description

Not available

Recruitment & Eligibility

Status
ACTIVE_NOT_RECRUITING
Sex
All
Target Recruitment
236
Inclusion Criteria
  • Participants with a BMI ≥27 kg/m² and <35 kg/m² and at least 2 obesity-related health problems (treated or untreated), OR a BMI ≥35 kg/m² and at least 1 obesity-related health problem (treated or untreated). At least one obesity-related health problem should be hypertension, dyslipidemia or T2D (approximately 25% of participants).
  • Have a history of at least one self-reported unsuccessful dietary effort to lose body weight.
  • Males and females may participate in this trial. Female participants must not be pregnant, intending to be pregnant, breastfeeding, or intending to breastfeed.
  • Contraceptive use by participants should be consistent with local regulations regarding the methods of contraception for those participating in clinical studies.
  • No male contraception is required except in compliance with specific local government study requirements.
Exclusion Criteria
  • For participants with Type 2 Diabetes (T2D):

    • Have Type 1 Diabetes (T1D), history of ketoacidosis or hyperosmolar state/coma, or any other types of diabetes except T2D.
    • Have had 1 or more episode of severe hypoglycemia and/or 1 or more episode of hypoglycemia unawareness within the 180 days prior to screening.
  • Have renal impairment measured as estimated glomerular filtration rate (eGFR) <15 mL/min/1.73 m², calculated by Japanese Society of Nephrology coefficient-modified chronic kidney disease-epidemiology equation during screening.

  • Have a known clinically significant gastric emptying abnormality.

  • For participants without Type 2 diabetes (T2D): Have any type of diabetes with hemoglobin A1c (HbA1c) ≥6.5 %.

  • Have a self-reported change in body weight >5 kg (11 pounds) within 90 days prior to screening.

  • Have chronic kidney disease.

  • Have lupus or rheumatoid arthritis.

  • Have the following cardiovascular conditions within 90 days prior to screening.

  • Have acute or chronic hepatitis.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
PlaceboPlaceboParticipants will receive placebo.
Orforglipron Dose 1OrforglipronParticipants will receive orforglipron orally.
Orforglipron Dose 2OrforglipronParticipants will receive orforglipron orally.
Orforglipron Dose 3OrforglipronParticipants will receive orforglipron orally.
Primary Outcome Measures
NameTimeMethod
Mean Percent Change in Body WeightBaseline, Week 72
Percentage of Participants Who Achieve ≥5% Body Weight ReductionBaseline to Week 72
Secondary Outcome Measures
NameTimeMethod
Mean Change from Baseline in HDLBaseline, Week 72
Mean Change from Baseline in TriglyceridesBaseline, Week 72
Mean Change from Baseline in Fasting GlucoseBaseline, Week 72
Percentage of Participants Who Achieve ≥10% Body Weight ReductionBaseline to Week 72
Percentage of Participants Who Achieve ≥15% Body Weight ReductionBaseline to Week 72
Percentage of Participants Who Achieve ≥20% Body Weight ReductionBaseline to Week 72
Mean Change from Baseline in Body Mass Index (BMI)Baseline, Week 72
Percentage of Participants Who Had Improvements in HypertensionBaseline to Week 72
Percentage of Participants Who Had Improvements in Dyslipidemia (only for participants with Dyslipidemia at baseline)Baseline to Week 72
Percentage of Participants Who Achieve HbA1c Target value (<6.5% (48 mmol/mol) at Week 72 (only T2D at Baseline):Baseline to Week 72
Mean Change from Baseline in Visceral Adipose Tissue (VAT)Baseline, Week 72
Mean Change from Baseline in Waist Circumference at Umbilical LevelBaseline, Week 72
Mean Change from Baseline in Systolic Blood Pressure (SBP)Baseline, Week 72
Mean Change from Baseline in Hemoglobin A1c (HbA1c)Baseline, Week 72
Mean Change from Baseline in non-High Density Lipoprotein (HDL)Baseline, Week 72
Mean Change from Baseline in High-sensitivity C-reactive ProteinBaseline, Week 72
Mean Change from Baseline in Short Form 36 Version 2 (SF-36v2) Acute Form Domain ScoresBaseline, Week 72
Mean Change from Baseline in IMPACT of Weight on Quality-of-Life Lite Clinical Trials Version (IWQOL-Lite-CT) Physical Function, Physical, and Psychosocial Composite ScoreBaseline, Week 72
Time to Onset of Type 2 Diabetes (T2D) (only non T2D at Baseline)Baseline to Week 72
Pharmacokinetics (PK): Plasma Concentration of OrforglipronBaseline to Week 72

Trial Locations

Locations (16)

Nihonbashi Sakura Clinic

🇯🇵

Chuo-ku, Tokyo, Japan

Heishinkai Medical Group ToCROM Clinic

🇯🇵

Shinjuku-ku, Tokyo, Japan

Fukuwa Clinic

🇯🇵

Chuo-ku, Tokyo, Japan

Tokyo-Eki Center-building Clinic

🇯🇵

Chuo-ku, Tokyo, Japan

Shiraiwa Medical Clinic

🇯🇵

Kashiwara, Osaka, Japan

Hiroshima Station Clinic

🇯🇵

Hiroshima, Japan

Osaka Nishiumeda Clinic

🇯🇵

Osaka, Japan

Takai Internal Medicine Clinic

🇯🇵

Kamakura-shi, Kanagawa, Japan

Ohishi Internal Medicine Clinic

🇯🇵

Tsuchiura, Ibaraki, Japan

Nishiyamadou Keiwa Hospital

🇯🇵

Naka, Ibaraki, Japan

Tsuchiura Beryl Clinic

🇯🇵

Tsuchiura, Ibaraki, Japan

Medical Corporation Yuga Higashirinkan Kaneshiro Diabetes Clinic

🇯🇵

Sagamihara, Kanagawa, Japan

Medical Corporation Heishinkai OCROM Clinic

🇯🇵

Suita-shi, Osaka, Japan

Shonan Takai Clinic

🇯🇵

Kamakura, Kanagawa, Japan

Sugiura Clinic

🇯🇵

Kawaguchi, Saitama, Japan

Yotsuya Medical Cube

🇯🇵

Chiyoda, Tokyo, Japan

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