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Dose-range Finding Study of BF2.649 Effect on Patients With Obstructive Sleep Apnea (OSA)

Phase 2
Completed
Conditions
Obstructive Sleep Apnoea
Excessive Daytime Sleepiness
Interventions
Drug: Placebo
Registration Number
NCT01620554
Lead Sponsor
Bioprojet
Brief Summary

Prospective, multicenter, double-blind, phase II, randomized, dose-response study in 5 parallel groups (dose-range).

Detailed Description

Obstructive sleep apnea (OSA) is a relatively common condition and is estimated to affect 2 to 4% of middle-aged adults

The study medication BF2.649 tested here is a novel, highly potent, selective, orally active inverse agonist at the histamine H3 receptor, therefore strengthens histaminergic transmission in the brain and increases wakefulness EDS is characterized by daytime somnolence and sudden sleep episodes. This problem has several consequences, e.g., an impairment of quality of life, an interference with activities of daily living and other handicaps in the management of social and family affairs.

The primary endpoint of this study will be measured by the change in the well-validated Epworth sleepiness scale (ESS). The ESS is a simple self-administered 8-item questionnaire. The outcome is to get an impression about the level of the daytime sleepiness in several real-life situations.

In this study, each patient will be treated during 2 weeks, and randomly assigned to one the 5 arms (BF2.649 at one of the 4 possible dosages or placebo).

The patient will then attend a end-of-treatment visit, in order to assess the particularly the ESS score.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
110
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
BF2.649 5mgBF2.649-
PlaceboPlacebo-
BF2.649 20mgBF2.649-
BF2.649 40mgBF2.649-
BF2.649 10mgBF2.649-
Primary Outcome Measures
NameTimeMethod
Change in Epworth Sleepiness Scale scores (ESS)change of ESS at 2 weeks

ESS value compared from baseline (Day 0) and End of treatment period (Day 14)

Secondary Outcome Measures
NameTimeMethod

Trial Locations

Locations (1)

CHU de Grenoble

🇫🇷

Grenoble, France

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