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Efficacy Study Exploring the Effect of Lu AE58054 as Augmentation Therapy in Patients With Schizophrenia

Phase 2
Completed
Conditions
Schizophrenia
Cognition
Interventions
Drug: Placebo
Registration Number
NCT00810667
Lead Sponsor
H. Lundbeck A/S
Brief Summary

The objective of this study is to explore the efficacy, safety and cognitive properties of Lu AE58054 as augmentation therapy to risperidone in patients with schizophrenia.

Detailed Description

Lu AE58054 is a selective 5-HT6 antagonist that is currently being investigated for treatment of conditions of cognitive impairment associated with schizophrenia. Substantial experimental evidence suggests that selective 5-HT6 receptor antagonists may be effective in treating cognitive deficits since they have been shown to improve performance in various animal models of cognitive function and are known to enhance cholinergic and glutaminergic neuronal function.

Lu AE58054 has been investigated in healthy volunteers and patients with schizophrenia, is generally well tolerated and has a benign side-effect profile. Moreover, no safety concerns or issues have been identified to date.

The study is designed to provide data on the efficacy, safety and cognitive properties of Lu AE58054 as augmentation therapy to risperidone in patients with schizophrenia. Efficacy will be assessed in patients who are in a stable phase of their illness, but with a predefined minimum and maximum level of symptoms that will allow them to be included in the study. Patients will be randomly assigned to receive either the investigational medicinal product (IMP) or placebo as add-on therapy to their existing risperidone treatment.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
124
Inclusion Criteria
  • Primary diagnosis of schizophrenia
  • Man or woman, aged between 18-65
  • Patient is on an optimised dose of risperidone (within 4-8 mg/day) for the treatment of schizophrenia for a minimum of 4 weeks prior to screening
  • The patient has a PANSS total score between 70 and 100 (extremes included) at screening
Exclusion Criteria
  • Primary psychiatric diagnosis other than schizophrenia
  • Acute exacerbation requiring hospitalisation within the last 3 months
  • Clinically significant extrapyramidal symptoms
  • Clinically significant cardiovascular disease, congestive heart failure, cardiac hypertrophy, arrhythmia or bradycardia
  • Significant ECG abnormalities
  • In concurrent treatment with drugs inhibiting the P450 enzymes system CYP2D6 and other CYP Isozymes
  • Failed to respond to adequate courses of treatment with risperidone
  • Treated with an antipsychotic other than risperidone within 4 weeks prior to screening

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Lu AE58054Lu AE58054-
PlaceboPlacebo-
Primary Outcome Measures
NameTimeMethod
Efficacy effect of treatment based on the PANSS total score12 weeks
Secondary Outcome Measures
NameTimeMethod
PANSS subscales scores, CGI-S and CGI-I scores, CDSS scores, S-QoL scores, BACS, Abnormal movement scales (AIMS, BARS, SAS), ECGs, serum prolactin, pharmacokinetic assessments12 weeks

Trial Locations

Locations (25)

PL012

🇵🇱

Lodz, Poland

PL009

🇵🇱

Belchatow, Poland

BE001

🇧🇪

Liege, Belgium

BE005

🇧🇪

Liege, Belgium

FR002

🇫🇷

Bordeaux, France

FR003

🇫🇷

Brumath, France

FR001

🇫🇷

Nimes, France

FR006

🇫🇷

Toulouse, France

DE002

🇩🇪

Dresden, Germany

IT003

🇮🇹

Brescia, Italy

IT004

🇮🇹

Napoli, Italy

HK001

🇭🇰

Hong Kong, Hong Kong

PL006

🇵🇱

Bialystok, Poland

PL003

🇵🇱

Lublin, Poland

PL002

🇵🇱

Leszno, Poland

PL001

🇵🇱

Lublin, Poland

PL010

🇵🇱

Piekary Slaskie, Poland

PL008

🇵🇱

Torun, Poland

PL004

🇵🇱

Skorzewo, Poland

PL011

🇵🇱

Warszawa, Poland

PL007

🇵🇱

Wrzesnia, Poland

TW001

🇨🇳

Hualien, Taiwan

TW003

🇨🇳

Keelung, Taiwan

TW004

🇨🇳

Tainan, Taiwan

TH002

🇹🇭

Chiang Mai, Thailand

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