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TA-8995: Its Use in Patients With Mild Dyslipidaemia (TULIP)

Phase 2
Completed
Conditions
Dyslipidemia
Interventions
Drug: TA-8995 0mg (placebo)
Drug: Placebo Statin
Registration Number
NCT01970215
Lead Sponsor
Xention Ltd
Brief Summary

The primary objective of this study is to evaluate the efficacy of different doses of TA-8995, a cholesteryl ester transfer protein (CETP) inhibitor, on the elevation of high-density lipoprotein cholesterol (HDL-C) and reduction of low-density lipoprotein cholesterol (LDL-C), alone and in combination with statin therapy.

The secondary objectives of this study are to determine the safety and tolerability of TA-8995 in patients with mild dyslipidaemia.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
364
Inclusion Criteria
  • Fasting LDL-C levels >2.5 mmol/L and <4.5 mmol/L, HDL-C levels <1.8 mmol/L and >0.8 mmol/L, and TG levels <4.5 mmol/L after run in or washout of existing therapies
  • Not on lipid-altering therapy at screening or on lipid-altering treatment regimens at screening
Exclusion Criteria
  • Body mass index >32 kg/m2;
  • Participation in another clinical study involving an investigational or marketed drug within 30 days prior to enrolment (Visit 2);
  • Any clinical manifestation of atherosclerotic vascular disease;
  • Diagnosis of type 1 diabetes;
  • Uncontrolled type 2 diabetes: haemoglobin A1c >8%;
  • Uncontrolled hypertension: sitting systolic blood pressure >160 mmHg and/or sitting diastolic blood pressure >90 mmHg;
  • History of hyperaldosteronism;
  • Active muscle disease or persistent creatine kinase concentration >3 × the upper limit of normal (ULN). One retest will be allowed after 1 week to verify the result;

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Group 3Placebo StatinTA-8995 2.5mg \& placebo statin
Group 5TA-8995TA-8995 10mg \& placebo statin
Group 4Placebo StatinTA-8995 5mg \& placebo statin
Group 1Placebo StatinTA-8995 0mg (placebo) \& placebo statin
Group 1TA-8995 0mg (placebo)TA-8995 0mg (placebo) \& placebo statin
Group 2Placebo StatinTA-8995 1mg \& placebo statin
Group 2TA-8995TA-8995 1mg \& placebo statin
Group 9TA-8995TA-8995 10mg \& rosuvastatin 10mg
Group 9RosuvastatinTA-8995 10mg \& rosuvastatin 10mg
Group 6TA-8995 0mg (placebo)TA-8995 0mg (placebo) \& atorvastatin 20mg
Group 7TA-8995TA-8995 10mg \& atorvastatin 20mg
Group 5Placebo StatinTA-8995 10mg \& placebo statin
Group 8TA-8995 0mg (placebo)TA-8995 0mg (placebo) \& rosuvastatin 10mg
Group 3TA-8995TA-8995 2.5mg \& placebo statin
Group 4TA-8995TA-8995 5mg \& placebo statin
Group 6AtorvastatinTA-8995 0mg (placebo) \& atorvastatin 20mg
Group 7AtorvastatinTA-8995 10mg \& atorvastatin 20mg
Group 8RosuvastatinTA-8995 0mg (placebo) \& rosuvastatin 10mg
Primary Outcome Measures
NameTimeMethod
The co-primary efficacy endpoints are the percentage changes in both HDL-C and LDL-C levels at Week 12 compared to baseline.12 weeks
Secondary Outcome Measures
NameTimeMethod

Trial Locations

Locations (17)

Albert Schweitzer Ziekenhuis

🇳🇱

Sliedrecht, Netherlands

Andromed Zoetermeer

🇳🇱

Leiderdorp, Netherlands

Andromed Breda B.V

🇳🇱

Breda, Netherlands

Andromed Rotterdam BV

🇳🇱

Rotterdam, Netherlands

Sydvestjysk Sygehus

🇩🇰

Esbjerg, Denmark

H:S Amager Hospital

🇩🇰

Copenhagen, Denmark

Herlev University Hospital

🇩🇰

Herlev, Denmark

EB FlevoResearch B.V

🇳🇱

Almere, Netherlands

Hvidovre Hospital

🇩🇰

Hvidovre, Denmark

Andromed Leiden

🇳🇱

Amsterdam, Netherlands

Regionshopitalet - Silkeborg

🇩🇰

Silkeborg, Denmark

Andromed Amsterdam

🇳🇱

Amsterdam, Netherlands

Academic Medical Centre

🇳🇱

Amsterdam-Zuidoost, Netherlands

Andromed Eindhoven

🇳🇱

Eindhoven, Netherlands

Andromed Noord B.V

🇳🇱

Groningen, Netherlands

Praktijk Zwijndrecht

🇳🇱

Zwijndrecht, Netherlands

Andromed Oost

🇳🇱

Velp, Netherlands

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