MedPath

An Evaluation of Sarilumab Plus Methotrexate Compared to Etanercept Plus Methotrexate in RA Patients Not Responding to Adalimumab Plus Methotrexate

Phase 3
Terminated
Conditions
Rheumatoid Arthritis
Interventions
Drug: Placebo (for etanercept)
Drug: Placebo (for sarilumab)
Registration Number
NCT01764997
Lead Sponsor
Sanofi
Brief Summary

Primary Objective:

To demonstrate the treatment effect of sarilumab and methotrexate (MTX) compared to etanercept and MTX in participants with rheumatoid arthritis (RA) and an inadequate response to adalimumab and MTX by evaluation of the Disease Activity Score for 28 joints (DAS28).

Secondary Objectives:

To assess the signs and symptoms of RA in participants taking sarilumab in combination with MTX.

To assess the quality of life of participants with RA taking sarilumab in combination with MTX.

To assess the safety and tolerability of sarilumab in combination with MTX in participants with RA.

Detailed Description

The maximum study duration per participant enrolled in the open label run-in phase and was eligible to enroll in the randomized phase of main study was 54 weeks:

* open label screening period of up to 4 weeks

* open-label treatment period of 16 weeks

* randomized screening period of 2 to 4 weeks

* randomized treatment post-treatment safety follow-up period of 6 weeks.

The maximum study duration per participant enrolled only in the open label run-in phase and was not eligible to enroll in the randomized phase of main study was 26 weeks:

* open label screening period of up to 4 weeks

* open-label treatment period of 16 weeks

* open label treatment post-treatment safety follow-up period of 6 weeks.

The maximum study duration per participant enrolled in the open label run-in phase and was eligible to enroll in the sarilumab sub-study was 82 weeks:

* open label screening period of up to 4 weeks

* open-label treatment period of 16 weeks

* screening period of 2 to 4 weeks

* sarilumab treatment period of 52 weeks

* sub-study post-treatment safety follow-up period of 6 weeks.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
776
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Sarilumab 150 mg + MTX (Randomized)SarilumabSarilumab 150 mg in combination with placebo for etanercept Q2W and placebo for etanercept on alternating weeks for 24 weeks added to stable dose of MTX.
Adalimumab Open Label run-inAdalimumabAdalimumab 40 mg every 2 weeks (Q2W) for 16 weeks added to stable dose of MTX.
Sarilumab 150 mg + MTX (Randomized)MethotrexateSarilumab 150 mg in combination with placebo for etanercept Q2W and placebo for etanercept on alternating weeks for 24 weeks added to stable dose of MTX.
Sarilumab 150 mg + MTX (Randomized)Placebo (for etanercept)Sarilumab 150 mg in combination with placebo for etanercept Q2W and placebo for etanercept on alternating weeks for 24 weeks added to stable dose of MTX.
Etanercept + MTX (Randomized)EtanerceptEtanercept 50 mg in combination with Placebo for sarilumab Q2W and etanercept 50 mg on alternating weeks for 24 weeks added to stable dose of MTX.
Etanercept + MTX (Randomized)MethotrexateEtanercept 50 mg in combination with Placebo for sarilumab Q2W and etanercept 50 mg on alternating weeks for 24 weeks added to stable dose of MTX.
Etanercept + MTX (Randomized)Placebo (for sarilumab)Etanercept 50 mg in combination with Placebo for sarilumab Q2W and etanercept 50 mg on alternating weeks for 24 weeks added to stable dose of MTX.
Sarilumab 200 mg + MTX (Randomized)Placebo (for etanercept)Sarilumab 200 mg in combination with placebo for etanercept Q2W and placebo for etanercept on alternating weeks for 24 weeks added to stable dose of MTX.
Sarilumab 150 mg + MTX Open Label Sub-studySarilumabSarilumab 150 mg Q2W for 52 weeks added to stable dose of MTX.
Adalimumab Open Label run-inMethotrexateAdalimumab 40 mg every 2 weeks (Q2W) for 16 weeks added to stable dose of MTX.
Sarilumab 200 mg + MTX (Randomized)SarilumabSarilumab 200 mg in combination with placebo for etanercept Q2W and placebo for etanercept on alternating weeks for 24 weeks added to stable dose of MTX.
Sarilumab 200 mg + MTX (Randomized)MethotrexateSarilumab 200 mg in combination with placebo for etanercept Q2W and placebo for etanercept on alternating weeks for 24 weeks added to stable dose of MTX.
Sarilumab 150 mg + MTX Open Label Sub-studyMethotrexateSarilumab 150 mg Q2W for 52 weeks added to stable dose of MTX.
Primary Outcome Measures
NameTimeMethod
Change From Baseline in Disease Activity Score for 28 Joints - C-Reactive Protein (DAS28-CRP) Score at Week 24Baseline, Week 24
Secondary Outcome Measures
NameTimeMethod
Number of Participants With at Least 20% Improvement in American College of Rheumatology (ACR20), at Least 50% Improvement in ACR (ACR50) and at Least 70% Improvement in ACR (ACR70) Efficacy Response Rates at Week 12 and Week 24Week 12 and Week 24
Percentage of Participants Achieving Clinical Remission Score (DAS28-CRP) <2.6 at Week 12 and Week 24Week 12 and Week 24
Change From Baseline in DAS28-CRP Score at Week 12Baseline, Week 12

Trial Locations

Locations (257)

Investigational Site Number 840203

🇺🇸

Washington, D.C., District of Columbia, United States

Investigational Site Number 032009

🇦🇷

Zarate, Argentina

Investigational Site Number 152018

🇨🇱

Santiago, Chile

Investigational Site Number 170041

🇨🇴

Medellin, Colombia

Investigational Site Number 840150

🇺🇸

Lansing, Michigan, United States

Investigational Site Number 840200

🇺🇸

Jackson, Mississippi, United States

Investigational Site Number 032053

🇦🇷

La Plata, Argentina

Investigational Site Number 076006

🇧🇷

Goiania, Brazil

Investigational Site Number 840210

🇺🇸

Clearwater, Florida, United States

Investigational Site Number 152015

🇨🇱

Temuco, Chile

Investigational Site Number 170040

🇨🇴

Bogotá, Colombia

Investigational Site Number 218001

🇪🇨

Guayaquil, Ecuador

Investigational Site Number 250006

🇫🇷

Strasbourg, France

Investigational Site Number 840060

🇺🇸

Sarasota, Florida, United States

Investigational Site Number 032050

🇦🇷

Buenos Aires, Argentina

Investigational Site Number 032013

🇦🇷

Rosario, Argentina

Investigational Site Number 032005

🇦🇷

Tucuman, Argentina

Investigational Site Number 840073

🇺🇸

Cumberland, Maryland, United States

Investigational Site Number 840025

🇺🇸

Jackson, Tennessee, United States

Investigational Site Number 840202

🇺🇸

Hagerstown, Maryland, United States

Investigational Site Number 840016

🇺🇸

North Charleston, South Carolina, United States

Investigational Site Number 076010

🇧🇷

Juiz De Fora, Brazil

Investigational Site Number 152001

🇨🇱

Santiago, Chile

Investigational Site Number 170007

🇨🇴

Bucaramanga, Colombia

Investigational Site Number 246001

🇫🇮

Helsinki, Finland

Investigational Site Number 250003

🇫🇷

Amiens Cedex 1, France

Investigational Site Number 840204

🇺🇸

Battle Creek, Michigan, United States

Investigational Site Number 032051

🇦🇷

San Miguel De Tucumán, Argentina

Investigational Site Number 076001

🇧🇷

Curitiba, Brazil

Investigational Site Number 152005

🇨🇱

Osorno, Chile

Investigational Site Number 152002

🇨🇱

Santiago, Chile

Investigational Site Number 170001

🇨🇴

Bogota, Colombia

Investigational Site Number 246030

🇫🇮

Oulu, Finland

Investigational Site Number 076016

🇧🇷

Curitiba, Brazil

Investigational Site Number 076005

🇧🇷

Rio De Janeiro, Brazil

Investigational Site Number 076013

🇧🇷

Vitoria, Brazil

Investigational Site Number 250005

🇫🇷

Paris, France

Investigational Site Number 152011

🇨🇱

Santiago, Chile

Investigational Site Number 170016

🇨🇴

Bogota, Colombia

Investigational Site Number 276056

🇩🇪

Dresden, Germany

Investigational Site Number 276053

🇩🇪

Ludwigsfelde, Germany

Investigational Site Number 300012

🇬🇷

Patras, Greece

Investigational Site Number 376010

🇮🇱

Haifa, Israel

Investigational Site Number 380002

🇮🇹

Firenze, Italy

Investigational Site Number 410016

🇰🇷

Seoul, Korea, Republic of

Investigational Site Number 250008

🇫🇷

Toulouse, France

Investigational Site Number 218002

🇪🇨

Quito, Ecuador

Investigational Site Number 250007

🇫🇷

Bobigny, France

Investigational Site Number 250004

🇫🇷

Paris Cedex 4, France

Investigational Site Number 276055

🇩🇪

Dresden, Germany

Investigational Site Number 276001

🇩🇪

Herne, Germany

Investigational Site Number 276050

🇩🇪

Rostock, Germany

Investigational Site Number 276057

🇩🇪

Berlin, Germany

Investigational Site Number 348001

🇭🇺

Budapest, Hungary

Investigational Site Number 246032

🇫🇮

Tampere, Finland

Investigational Site Number 300010

🇬🇷

Athens, Greece

Investigational Site Number 376034

🇮🇱

Tel Hashomer, Israel

Investigational Site Number 380005

🇮🇹

Genova, Italy

Investigational Site Number 410020

🇰🇷

Busan, Korea, Republic of

Investigational Site Number 410005

🇰🇷

Daejeon, Korea, Republic of

Investigational Site Number 428001

🇱🇻

Riga, Latvia

Investigational Site Number 458001

🇲🇾

Ipoh, Malaysia

Investigational Site Number 276007

🇩🇪

Berlin, Germany

Investigational Site Number 410022

🇰🇷

Seoul, Korea, Republic of

Investigational Site Number 410023

🇰🇷

Seoul, Korea, Republic of

Investigational Site Number 250001

🇫🇷

La Roche Sur Yon Cedex 9, France

Investigational Site Number 250002

🇫🇷

Montpellier, France

Investigational Site Number 276051

🇩🇪

Erlangen, Germany

Investigational Site Number 348021

🇭🇺

Esztergom, Hungary

Investigational Site Number 376011

🇮🇱

Tel Aviv, Israel

Investigational Site Number 616018

🇵🇱

Poznan, Poland

Investigational Site Number 616016

🇵🇱

Szczecin, Poland

Investigational Site Number 616058

🇵🇱

Ustron, Poland

Investigational Site Number 410015

🇰🇷

Seoul, Korea, Republic of

Investigational Site Number 410021

🇰🇷

Seoul, Korea, Republic of

Investigational Site Number 276013

🇩🇪

Hamburg, Germany

Investigational Site Number 276058

🇩🇪

Koeln, Germany

Investigational Site Number 380042

🇮🇹

Valeggio Sul Mincio, Italy

Investigational Site Number 410011

🇰🇷

Jeonju, Korea, Republic of

Investigational Site Number 428003

🇱🇻

Ventspils, Latvia

Investigational Site Number 554011

🇳🇿

Nelson, New Zealand

Investigational Site Number 616054

🇵🇱

Bytom, Poland

Investigational Site Number 616013

🇵🇱

Sosnowiec, Poland

Investigational Site Number 300014

🇬🇷

N. Efkarpia, Greece

Investigational Site Number 376001

🇮🇱

Haifa, Israel

Investigational Site Number 376035

🇮🇱

Jerusalem, Israel

Investigational Site Number 376030

🇮🇱

Ramat Gan, Israel

Investigational Site Number 410008

🇰🇷

Suwon, Korea, Republic of

Investigational Site Number 428002

🇱🇻

Liepaja, Latvia

Investigational Site Number 440005

🇱🇹

Kaunas, Lithuania

Investigational Site Number 840124

🇺🇸

Clarksburg, West Virginia, United States

Investigational Site Number 440011

🇱🇹

Vilnius, Lithuania

Investigational Site Number 616015

🇵🇱

Elblag, Poland

Investigational Site Number 616061

🇵🇱

Krakow, Poland

Investigational Site Number 616056

🇵🇱

Starachowice, Poland

Investigational Site Number 642023

🇷🇴

Bucharest, Romania

Investigational Site Number 642040

🇷🇴

Bucuresti, Romania

Investigational Site Number 616052

🇵🇱

Dzialdowo, Poland

Investigational Site Number 616059

🇵🇱

Krakow, Poland

Investigational Site Number 616005

🇵🇱

Lublin, Poland

Investigational Site Number 616051

🇵🇱

Warszawa, Poland

Investigational Site Number 642005

🇷🇴

Galati, Romania

Investigational Site Number 642013

🇷🇴

Iasi, Romania

Investigational Site Number 642004

🇷🇴

Bucharest, Romania

Investigational Site Number 642002

🇷🇴

Bucuresti, Romania

Investigational Site Number 642001

🇷🇴

Bucuresti, Romania

Investigational Site Number 643022

🇷🇺

Novosibirsk, Russian Federation

Investigational Site Number 643010

🇷🇺

Samara, Russian Federation

Investigational Site Number 643011

🇷🇺

Saratov, Russian Federation

Investigational Site Number 642042

🇷🇴

Bucuresti, Romania

Investigational Site Number 642022

🇷🇴

Targoviste, Romania

Investigational Site Number 643051

🇷🇺

Yaroslavl, Russian Federation

Investigational Site Number 643031

🇷🇺

Moscow, Russian Federation

Investigational Site Number 642014

🇷🇴

Iasi, Romania

Investigational Site Number 643006

🇷🇺

Kemerovo, Russian Federation

Investigational Site Number 158010

🇨🇳

Changhua, Taiwan

Investigational Site Number 643052

🇷🇺

Moscow, Russian Federation

Investigational Site Number 643021

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Moscow, Russian Federation

Investigational Site Number 643008

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St-Petersburg, Russian Federation

Investigational Site Number 158012

🇨🇳

Kaohsiung, Taiwan

Investigational Site Number 158011

🇨🇳

Kaohsiung, Taiwan

Investigational Site Number 804022

🇺🇦

Odesa, Ukraine

Investigational Site Number 643030

🇷🇺

Moscow, Russian Federation

Investigational Site Number 643059

🇷🇺

Smolensk, Russian Federation

Investigational Site Number 643058

🇷🇺

St. Peterburg, Russian Federation

Investigational Site Number 643013

🇷🇺

Ufa, Russian Federation

Investigational Site Number 643050

🇷🇺

Voronezh, Russian Federation

Investigational Site Number 804001

🇺🇦

Kharkov, Ukraine

Investigational Site Number 804023

🇺🇦

Kyiv, Ukraine

Investigational Site Number 804030

🇺🇦

Lutsk, Ukraine

Investigational Site Number 643057

🇷🇺

Yaroslavl, Russian Federation

Investigational Site Number 764011

🇹🇭

Khon Kaen, Thailand

Investigational Site Number 158006

🇨🇳

Taipei, Taiwan

Investigational Site Number 158004

🇨🇳

Chia-Yi, Taiwan

Investigational Site Number 764003

🇹🇭

Bangkok-Noi, Thailand

Investigational Site Number 764010

🇹🇭

Bangkok, Thailand

Investigational Site Number 804010

🇺🇦

Kharkiv, Ukraine

Investigational Site Number 804025

🇺🇦

Kiev, Ukraine

Investigational Site Number 804020

🇺🇦

Lviv, Ukraine

Investigational Site Number 804002

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Donetsk, Ukraine

Investigational Site Number 804024

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Donetsk, Ukraine

Investigational Site Number 804014

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Kyiv, Ukraine

Investigational Site Number 804029

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Ivano-Frankivsk, Ukraine

Investigational Site Number 804027

🇺🇦

Kyiv, Ukraine

Investigational Site Number 804012

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Odessa, Ukraine

Investigational Site Number 804028

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Zaporozhye, Ukraine

Investigational Site Number 804031

🇺🇦

Zhytomyr, Ukraine

Investigational Site Number 804011

🇺🇦

Kyiv, Ukraine

Investigational Site Number 804005

🇺🇦

Lviv, Ukraine

Investigational Site Number 804033

🇺🇦

Lviv, Ukraine

Investigational Site Number 840128

🇺🇸

Ormond Beach, Florida, United States

Investigational Site Number 840056

🇺🇸

New York, New York, United States

Investigational Site Number 840018

🇺🇸

Idaho Falls, Idaho, United States

Investigational Site Number 840074

🇺🇸

Mesquite, Texas, United States

Investigational Site Number 840037

🇺🇸

Tupelo, Mississippi, United States

Investigational Site Number 840112

🇺🇸

Lincoln, Nebraska, United States

Investigational Site Number 203030

🇨🇿

Praha 4, Czechia

Investigational Site Number 203006

🇨🇿

Zlin, Czechia

Investigational Site Number 840061

🇺🇸

Tacoma, Washington, United States

Investigational Site Number 036020

🇦🇺

Camperdown, Australia

Investigational Site Number 036007

🇦🇺

Woodville, Australia

Investigational Site Number 203004

🇨🇿

Ostrava, Czechia

Investigational Site Number 840209

🇺🇸

Danbury, Connecticut, United States

Investigational Site Number 840205

🇺🇸

Victorville, California, United States

Investigational Site Number 840109

🇺🇸

Lake Charles, Louisiana, United States

Investigational Site Number 032052

🇦🇷

Buenos Aires, Argentina

Investigational Site Number 840117

🇺🇸

Pittsburgh, Pennsylvania, United States

Investigational Site Number 203031

🇨🇿

Praha 4, Czechia

Investigational Site Number 036004

🇦🇺

Heidelberg West, Australia

Investigational Site Number 036014

🇦🇺

Victoria Park, Australia

Investigational Site Number 348013

🇭🇺

Gy?r, Hungary

Investigational Site Number 170009

🇨🇴

Bucaramanga, Colombia

Investigational Site Number 203001

🇨🇿

Praha 2, Czechia

Investigational Site Number 203002

🇨🇿

Uherske Hradiste, Czechia

Investigational Site Number 218003

🇪🇨

Cuenca, Ecuador

Investigational Site Number 246002

🇫🇮

Hyvinkää, Finland

Investigational Site Number 246003

🇫🇮

Pori, Finland

Investigational Site Number 203033

🇨🇿

Praha 4, Czechia

Investigational Site Number 203032

🇨🇿

Praha, Czechia

Investigational Site Number 376032

🇮🇱

Ashkelon, Israel

Investigational Site Number 380004

🇮🇹

Genova, Italy

Investigational Site Number 380041

🇮🇹

L'Aquila, Italy

Investigational Site Number 724042

🇪🇸

Madrid, Spain

Investigational Site Number 710008

🇿🇦

Pretoria, South Africa

Investigational Site Number 724001

🇪🇸

Málaga, Spain

Investigational Site Number 724011

🇪🇸

Sabadell, Spain

Investigational Site Number 616053

🇵🇱

Zyrardow, Poland

Investigational Site Number 826021

🇬🇧

Dudley, United Kingdom

Investigational Site Number 826020

🇬🇧

Harlow, United Kingdom

Investigational Site Number 724040

🇪🇸

Madrid, Spain

Investigational Site Number 642012

🇷🇴

Bucharest, Romania

Investigational Site Number 826025

🇬🇧

Wigan, United Kingdom

Investigational Site Number 724009

🇪🇸

La Coruña, Spain

Investigational Site Number 710010

🇿🇦

Stellenbsoch, South Africa

Investigational Site Number 724041

🇪🇸

Madrid, Spain

Investigational Site Number 724043

🇪🇸

Córdoba, Spain

Investigational Site Number 643056

🇷🇺

Krasnoyarsk, Russian Federation

Investigational Site Number 826022

🇬🇧

Birmingham, United Kingdom

Investigational Site Number 724012

🇪🇸

Santiago De Compostela, Spain

Investigational Site Number 710011

🇿🇦

Cape Town, South Africa

Investigational Site Number 710006

🇿🇦

Pretoria, South Africa

Investigational Site Number 826026

🇬🇧

Durham, United Kingdom

Investigational Site Number 840004

🇺🇸

Birmingham, Alabama, United States

Investigational Site Number 840213

🇺🇸

Indianapolis, Indiana, United States

Investigational Site Number 840201

🇺🇸

Denver, Colorado, United States

Investigational Site Number 840207

🇺🇸

Tampa, Florida, United States

Investigational Site Number 840212

🇺🇸

Glendale, California, United States

Investigational Site Number 840211

🇺🇸

Thousand Oaks, California, United States

Investigational Site Number 840049

🇺🇸

Upland, California, United States

Investigational Site Number 300002

🇬🇷

Heraklion, Greece

Investigational Site Number 348010

🇭🇺

Debrecen, Hungary

Investigational Site Number 348008

🇭🇺

Gyula, Hungary

Investigational Site Number 376031

🇮🇱

Haifa, Israel

Investigational Site Number 410006

🇰🇷

Busan, Korea, Republic of

Investigational Site Number 410013

🇰🇷

Daegu, Korea, Republic of

Investigational Site Number 440006

🇱🇹

Klaipeda, Lithuania

Investigational Site Number 440010

🇱🇹

Panevezys, Lithuania

Investigational Site Number 458012

🇲🇾

Batu Caves, Malaysia

Investigational Site Number 458014

🇲🇾

Georgetown, Malaysia

Investigational Site Number 458013

🇲🇾

Kota Bharu, Malaysia

Investigational Site Number 458002

🇲🇾

Kuching, Malaysia

Investigational Site Number 458010

🇲🇾

Melaka, Malaysia

Investigational Site Number 458011

🇲🇾

Seremban, Malaysia

Investigational Site Number 484027

🇲🇽

Cd. Obregon, Mexico

Investigational Site Number 484023

🇲🇽

Chihuahua, Mexico

Investigational Site Number 484029

🇲🇽

Deleg. Benito Juárez, Mexico

Investigational Site Number 484013

🇲🇽

Guadalajara, Mexico

Investigational Site Number 484018

🇲🇽

Guadalajara, Mexico

Investigational Site Number 484004

🇲🇽

Merida, Mexico

Investigational Site Number 484052

🇲🇽

Mexico City, Mexico

Investigational Site Number 484010

🇲🇽

Mexicali, Mexico

Investigational Site Number 484026

🇲🇽

Mexicali, Mexico

Investigational Site Number 484017

🇲🇽

México, Mexico

Investigational Site Number 484051

🇲🇽

Tijuana, Mexico

Investigational Site Number 484025

🇲🇽

San Luis, Mexico

Investigational Site Number 554010

🇳🇿

Dunedin, New Zealand

Investigational Site Number 554007

🇳🇿

Auckland, New Zealand

Investigational Site Number 554005

🇳🇿

Hamilton, New Zealand

Investigational Site Number 604001

🇵🇪

Lima, Peru

Investigational Site Number 604009

🇵🇪

Lima, Peru

Investigational Site Number 604010

🇵🇪

Lima, Peru

Investigational Site Number 604012

🇵🇪

Lima, Peru

Investigational Site Number 604007

🇵🇪

Lima, Peru

Investigational Site Number 604005

🇵🇪

Lima, Peru

Investigational Site Number 604020

🇵🇪

Lima, Peru

Investigational Site Number 616019

🇵🇱

Bydgoszcz, Poland

Investigational Site Number 616057

🇵🇱

Krakow, Poland

Investigational Site Number 616063

🇵🇱

Myslenice, Poland

Investigational Site Number 642041

🇷🇴

Bacau, Romania

Investigational Site Number 710007

🇿🇦

Cape Town, South Africa

Investigational Site Number 764002

🇹🇭

Bangkok, Thailand

Investigational Site Number 804003

🇺🇦

Dnipropetrovsk, Ukraine

Investigational Site Number 804021

🇺🇦

Simferopol, Ukraine

Investigational Site Number 826023

🇬🇧

Barnsley, United Kingdom

Investigational Site Number 804032

🇺🇦

Odesa, Ukraine

Investigational Site Number 826027

🇬🇧

Durham, United Kingdom

Investigational Site Number 840063

🇺🇸

Palm Harbor, Florida, United States

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