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Effects of Sodium-glucose Co-transporter-2( SGLT-2 ) Inhibition on Sympathetic Nervous System Activity in Humans

Phase 4
Recruiting
Conditions
Metabolic Syndrome
Type 2 Diabetes Mellitus
Obesity
Interventions
Registration Number
NCT03912909
Lead Sponsor
Royal Perth Hospital
Brief Summary

This study is designed to investigate whether the sodium-glucose co-transporter-2 (SGLT-2) inhibitor Empagliflozin reduces sympathetic nervous system (SNS) activity in humans.

Detailed Description

This is a randomised, double-blind, placebo controlled, cross-over study. Participants will be randomly assigned to receive either Empagliflozin 10mg/daily or Placebo and will later receive the alternate treatment.

Comprehensive testing will occur after each 4 week treatment phase and will include assessment of muscle sympathetic nerve activity, cardiac and renal noradrenaline spillover to assess organ specific SNS activity.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
30
Inclusion Criteria
  • Age: 25 -65 years
  • (Body Mass Index) BMI≥30kg/m2
  • Currently weight stable (+/- 3% in previous 6-12 months and not on any specific exercise or dietary program)
  • Metabolic syndrome (defined as having: obesity (BMI ≥30kg/m2 ) plus any two of the following four factors: Elevated triglycerides (Triglyceride≥ 1.7mmol/L), Reduced HDL (High - density lipoprotein) cholesterol (<1.0mmol/L in males, <1.3mmol/L in females), Elevated clinic systolic (Blood Pressure) BP ≥130 or diastolic BP ≥85mmHg, Fasting glucose ≥5.6mmol/L or type 2 diabetes.
  • office BP for screening purposes ≤160/90mmHg
  • drug naïve for at least 6 weeks prior to baseline assessment
Exclusion Criteria
  • Grade 2-3 hypertension (systolic office BP >160, diastolic office BP >100 mmHg)
  • Secondary causes of hypertension
  • CKD (Chronic kidney disease) stage 4-5 {(estimated glomerular filtration) eGFR<30ml/min}
  • Heart failure NYHA (New York Heart Association) class II-IV
  • Recent CV (cardiovascular) event (acute myocardial infarction, acute coronary syndrome, stroke or transient ischaemic attack within the previous six months)
  • unstable psychiatric condition
  • medication such as corticosteroids, several antidepressants and antipsychotics
  • Female participants of childbearing potential must have a negative pregnancy test prior to treatment

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
Phase 1Placebo Oral TabletEmpagliflozin 10mg daily or placebo
Phase2Placebo Oral TabletEmpagliflozin 10mg daily or placebo
Phase 1Empagliflozin Oral Tablet [Jardiance]Empagliflozin 10mg daily or placebo
Phase2Empagliflozin Oral Tablet [Jardiance]Empagliflozin 10mg daily or placebo
Primary Outcome Measures
NameTimeMethod
Reduction in renal sympathetic nerve activity18 weeks

Renal sympathetic nerve activity assessed by renal noradrenaline spillover

Reduction in muscle sympathetic nerve activity18 weeks

Muscle sympathetic nerve activity assessed by microneurography

Reduction in cardiac sympathetic nerve activity18 weeks

Cardiac sympathetic nerve activity assessed by cardiac noradrenaline spillover

Secondary Outcome Measures
NameTimeMethod
Reduction in ambulatory BP (blood pressure)18 weeks

Blood Pressure assessed by ambulatory blood pressure monitoring

Change in urinary sodium excretion18 weeks

Urinary sodium excretion assessed in a 24 hour urine sample

Reduction in central Blood Pressure18 weeks

central Blood Pressure assessed by Sphygmocor XCEL

Change in glycemic control18 weeks

Glycemic control as assessed by an oral glucose tolerance test

Trial Locations

Locations (1)

Royal Perth Hospital

🇦🇺

Perth, Western Australia, Australia

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