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The Interaction Between Metformin and Acute Exercise

Not Applicable
Completed
Conditions
Impaired Glucose Tolerance
Diabetes Mellitus, Type 2
Interventions
Drug: Placebo treatment
Registration Number
NCT03329651
Lead Sponsor
Kristian Karstoft
Brief Summary

Physical activity is a first line treatment for patients with type 2 diabetes (T2D), however, the vast majority of patients with T2D do not achieve satisfying glycemic control with physical activity alone, which is why pharmacological treatment with metformin is most often initiated.

It is known that metformin and exercise both activates 5' adenosine monophosphate-activated protein kinase (AMPK) in skeletal muscle and liver, and the activation of AMPK results in many different metabolic effects, including improvements in glycemic control. Because of this similarity in mechanism of action, an interaction between metformin and exercise is plausible, but knowledge in the area is sparse. Thus, the aim of this study is to assess the effects of acute physical activity with and without concomitant metformin treatment, in order to investigate whether an interaction between the two occur.

Subjects with impaired glucose tolerance will be randomized (1:1) to metformin/placebo treatment in a double-blinded way. Following a treatment run-in period of 17 days, two experimental days (one with acute exercise and one without acute exercise), separated by one week, will be performed in each subject.

This registration concerns a sub-study of another study which has previously been registrered at ClinicalTrials.gov (Unique Protocol ID: H-17012307). The specific outcomes in this registration have not previously been registered.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
34
Inclusion Criteria
  • Glucose-lowering-medication naïve T2D and/or subjects with impaired glucose tolerance defined as: 2-h plasma glucose (PG) in the 75-g OGTT (7.8-11.0 mmol/L) and/or HbA1c (39-47 mmol/mol)
  • Caucasian
  • BMI > 25 but < 40 kg/m2
  • Low to moderate physically active (≤90 min of structured physical activity/week)
Exclusion Criteria
  • Pregnancy
  • Smoking
  • Glucose-lowering treatment
  • Treatment with steroids and other immunomodulating drugs
  • Contraindication to increased levels of physical activity
  • Liver disease (ALAT elevated more than 3 times above upper normal limit, or reduced levels of the liver function markers albumin and KF II+VII+X)
  • Renal insufficiency (eGFR<60 ml/min)
  • Prior history of lactic acidosis
  • HbA1c >55 mmol/mol and/or 2-hPG in the 75-g OGTT > 15 mmol/L

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Metformin treatmentMetformin treatment-
Placebo treatmentPlacebo treatment-
Primary Outcome Measures
NameTimeMethod
Difference in postprandial glycemic control as assessed by mean blood glucose concentration during a 4 hour mixed-meal tolerance testDay 17 (no acute exercise [control day]) and 24 (following an acute exercise bout)
Secondary Outcome Measures
NameTimeMethod
Difference in exogenous glucose uptake as assessed by rate of ingested glucose tracer appearance in bloodDay 17 (no acute exercise [control day]) and 24 (following an acute exercise bout)
Difference in endogenous glucose production as assessed by rate of infused glucose tracer appearance in bloodDay 17 (no acute exercise [control day]) and 24 (following an acute exercise bout)
Difference in peripheral glucose uptake as assessed by rate of glucose disappearance from bloodDay 17 (no acute exercise [control day]) and 24 (following an acute exercise bout)

Trial Locations

Locations (1)

Center for aktiv sundhed

🇩🇰

Copenhagen, Copenhagen N, Denmark

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