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Pimasertib

Generic Name
Pimasertib
Drug Type
Small Molecule
Chemical Formula
C15H15FIN3O3
CAS Number
1236699-92-5
Unique Ingredient Identifier
6ON9RK82AL
Background

Pimasertib is under investigation in clinical trial NCT01378377 (Combination Trial of Pimasertib (MSC1936369B) With Temsirolimus).

Oral SAR245408 (XL147) and Oral MSC1936369B in Patients With Locally Advanced or Metastatic Solid Tumors

Phase 1
Completed
Conditions
Solid Tumors
Interventions
Drug: SAR245408 (XL147)
First Posted Date
2011-05-20
Last Posted Date
2016-04-01
Lead Sponsor
Sanofi
Target Recruit Count
18
Registration Number
NCT01357330
Locations
🇺🇸

Investigational Site Number 840001, Boston, Massachusetts, United States

🇺🇸

Investigational Site Number 840002, Boston, Massachusetts, United States

🇺🇸

Investigational Site Number 840003, Nashville, Tennessee, United States

MEK Inhibitor MSC1936369B Plus FOLFIRI in Second Line K-Ras Mutated Metastatic Colorectal Cancer (mCRC)

Phase 1
Terminated
Conditions
Metastatic Colorectal Cancer
Interventions
Drug: Placebo
Drug: FOLFIRI
First Posted Date
2010-03-11
Last Posted Date
2016-10-19
Lead Sponsor
EMD Serono
Target Recruit Count
16
Registration Number
NCT01085331
Locations
🇪🇸

Research Site, Barcelona, Spain

Trial of Gemcitabine With or Without MSC1936369B in Pancreatic Cancer

Phase 1
Completed
Conditions
Pancreatic Adenocarcinoma
Interventions
First Posted Date
2009-11-19
Last Posted Date
2017-07-13
Lead Sponsor
EMD Serono
Target Recruit Count
141
Registration Number
NCT01016483
Locations
🇺🇸

For Recruiting Locations in the United States, please Contact U.S. Medical Information, Rockland, Massachusetts, United States

🇩🇪

For Recruiting Locations outside the United States, Please contact the Merck KGaA Communication Center, Darmstadt, Germany

Trial of MSC1936369B in Subjects With Solid Tumors

Phase 1
Completed
Conditions
Solid Tumors
Cancer
Interventions
First Posted Date
2009-09-23
Last Posted Date
2018-10-23
Lead Sponsor
Merck KGaA, Darmstadt, Germany
Target Recruit Count
182
Registration Number
NCT00982865
Locations
🇫🇷

Hopital Saint Louis, Paris, France

🇦🇺

Westmead Hospital, Westmead, Australia

🇫🇷

Centre Eugène Marquis, Rennes, France

and more 6 locations

Trial of Pimasertib in Hematological Malignancies

Phase 2
Terminated
Conditions
Leukemia, Myeloid, Acute
Hematologic Neoplasms
Interventions
First Posted Date
2009-08-12
Last Posted Date
2017-08-21
Lead Sponsor
EMD Serono
Target Recruit Count
81
Registration Number
NCT00957580
Locations
🇺🇸

Northwestern University, Chicago, Illinois, United States

🇺🇸

Dana Farber Cancer Institute, Boston, Massachusetts, United States

🇺🇸

Sidney Kimmel Comprehensive Cancer Center at Johns Hopkins, Baltimore, Maryland, United States

and more 6 locations
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