Tolperisone
- Generic Name
- Tolperisone
- Drug Type
- Small Molecule
- Chemical Formula
- C16H23NO
- CAS Number
- 728-88-1
- Unique Ingredient Identifier
- F5EOM0LD8E
Overview
Tolperisone is an oral, centrally acting muscle relaxant. Its precise mechanism is not completely understood, though it blocks sodium and calcium channels. It possesses a high affinity for nervous system tissue, reaching highest concentrations in brain stem, spinal cord and peripheral nerves. Based on existing clinical data, Tolperisone is not sedating and does not interact with alcohol.
Background
Tolperisone is an oral, centrally acting muscle relaxant. Its precise mechanism is not completely understood, though it blocks sodium and calcium channels. It possesses a high affinity for nervous system tissue, reaching highest concentrations in brain stem, spinal cord and peripheral nerves. Based on existing clinical data, Tolperisone is not sedating and does not interact with alcohol.
Indication
Investigated for use/treatment in neurologic disorders, spinal cord injuries, muscle spasm, back pain, and multiple sclerosis.
Associated Conditions
- Spasticity
Clinical Trials
FDA Approved Products
Singapore Approved Products
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