Cabotegravir
- Generic Name
- Cabotegravir
- Brand Names
- Apretude, Vocabria
- Drug Type
- Small Molecule
- Chemical Formula
- C19H17F2N3O5
- CAS Number
- 1051375-10-0
- Unique Ingredient Identifier
- HMH0132Z1Q
- Background
Cabotegravir, or GSK1265744, is an HIV-1 integrase inhibitor that is prescribed with the non-nucleoside reverse transcriptase inhibitor, rilpivirine. Early research into cabotegravir showed it had lower oral bioavailability than dolutegravir, which resulted in the development of long acting monthly intramuscular injection formulation for cabotegravir.
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- Indication
Oral cabotegravir is indicated in combination with rilpivirine for the short-term treatment of HIV-1 in virologically suppressed adults with no history of treatment failure to assess tolerability of cabotegravir or who have missed an injected dose of cabotegravir. Intramuscular extended-release cabotegravir in combination with rilpivirine is indicated as a c...
- Associated Conditions
- Human Immunodeficiency Virus Type 1 (HIV-1), Human Immunodeficiency Virus Type 1 (HIV-1) Infection
- Associated Therapies
- Oral Therapies
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