Lenacapavir

Generic Name
Lenacapavir
Brand Names
Sunlenca
Drug Type
Small Molecule
Chemical Formula
C39H32ClF10N7O5S2
CAS Number
2189684-44-2
Unique Ingredient Identifier
A9A0O6FB4H
Background

HIV/AIDS remains an area of concern despite the introduction of numerous successful therapies, mainly due to the emergence of multidrug resistance and patient difficulty in adhering to treatment regimens. Lenacapavir is a first-in-class capsid inhibitor that demonstrates picomolar HIV-1 inhibition as a monotherapy in vitro, little to no cross-resistance with...

Indication

Lenacapavir, in combination with other antiretroviral(s), is indicated for the treatment of multidrug-resistant human immunodeficiency virus type 1 (HIV-1) infection in heavily treatment-experienced adults who are experiencing a failure of their current antiretroviral regimen due to resistance, intolerance, or safety considerations.

Associated Conditions
Multidrug resistant HIV-1 infection
Associated Therapies
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