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Xylocaine

Xylocaine® (lidocaine HCl Injection, USP) Xylocaine® (lidocaine HCl and epinephrine Injection, USP)

Approved
Approval ID

ba082c2f-64f4-419d-9c88-74f203316e17

Product Type

HUMAN PRESCRIPTION DRUG LABEL

Effective Date

Aug 25, 2021

Manufacturers
FDA

Fresenius Kabi USA, LLC

DUNS: 608775388

Products 10

Detailed information about drug products covered under this FDA approval, including NDC codes, dosage forms, ingredients, and administration routes.

LIDOCAINE HYDROCHLORIDE,EPINEPHRINE BITARTRATE

Product Details

FDA regulatory identification and product classification information

FDA Identifiers
NDC Product Code63323-489
Application NumberNDA006488
Product Classification
M
Marketing Category
C73594
G
Generic Name
LIDOCAINE HYDROCHLORIDE,EPINEPHRINE BITARTRATE
Product Specifications
Route of AdministrationINFILTRATION, PERINEURAL, INTRACAUDAL, EPIDURAL
Effective DateAugust 28, 2020
FDA Product Classification

INGREDIENTS (7)

SODIUM CHLORIDEInactive
Quantity: 6 mg in 1 mL
Code: 451W47IQ8X
Classification: IACT
CITRIC ACID MONOHYDRATEInactive
Quantity: 0.2 mg in 1 mL
Code: 2968PHW8QP
Classification: IACT
SODIUM METABISULFITEInactive
Quantity: 0.5 mg in 1 mL
Code: 4VON5FNS3C
Classification: IACT
SODIUM HYDROXIDEInactive
Code: 55X04QC32I
Classification: IACT
HYDROCHLORIC ACIDInactive
Code: QTT17582CB
Classification: IACT
EPINEPHRINE BITARTRATEActive
Quantity: 0.005 mg in 1 mL
Code: 30Q7KI53AK
Classification: ACTIM
LIDOCAINE HYDROCHLORIDE ANHYDROUSActive
Quantity: 20 mg in 1 mL
Code: EC2CNF7XFP
Classification: ACTIB

LIDOCAINE HYDROCHLORIDE,EPINEPHRINE BITARTRATE

Product Details

FDA regulatory identification and product classification information

FDA Identifiers
NDC Product Code63323-482
Application NumberNDA006488
Product Classification
M
Marketing Category
C73594
G
Generic Name
LIDOCAINE HYDROCHLORIDE,EPINEPHRINE BITARTRATE
Product Specifications
Route of AdministrationINFILTRATION, PERINEURAL
Effective DateAugust 28, 2020
FDA Product Classification

INGREDIENTS (8)

SODIUM METABISULFITEInactive
Quantity: 0.5 mg in 1 mL
Code: 4VON5FNS3C
Classification: IACT
SODIUM HYDROXIDEInactive
Code: 55X04QC32I
Classification: IACT
HYDROCHLORIC ACIDInactive
Code: QTT17582CB
Classification: IACT
EPINEPHRINE BITARTRATEActive
Quantity: 0.01 mg in 1 mL
Code: 30Q7KI53AK
Classification: ACTIM
CITRIC ACID MONOHYDRATEInactive
Quantity: 0.2 mg in 1 mL
Code: 2968PHW8QP
Classification: IACT
SODIUM CHLORIDEInactive
Quantity: 7 mg in 1 mL
Code: 451W47IQ8X
Classification: IACT
METHYLPARABENInactive
Quantity: 1 mg in 1 mL
Code: A2I8C7HI9T
Classification: IACT
LIDOCAINE HYDROCHLORIDE ANHYDROUSActive
Quantity: 10 mg in 1 mL
Code: EC2CNF7XFP
Classification: ACTIB

LIDOCAINE HYDROCHLORIDE,EPINEPHRINE BITARTRATE

Product Details

FDA regulatory identification and product classification information

FDA Identifiers
NDC Product Code63323-481
Application NumberNDA006488
Product Classification
M
Marketing Category
C73594
G
Generic Name
LIDOCAINE HYDROCHLORIDE,EPINEPHRINE BITARTRATE
Product Specifications
Route of AdministrationINFILTRATION, PERINEURAL
Effective DateAugust 28, 2020
FDA Product Classification

INGREDIENTS (8)

CITRIC ACID MONOHYDRATEInactive
Quantity: 0.2 mg in 1 mL
Code: 2968PHW8QP
Classification: IACT
SODIUM CHLORIDEInactive
Quantity: 8 mg in 1 mL
Code: 451W47IQ8X
Classification: IACT
SODIUM METABISULFITEInactive
Quantity: 0.5 mg in 1 mL
Code: 4VON5FNS3C
Classification: IACT
METHYLPARABENInactive
Quantity: 1 mg in 1 mL
Code: A2I8C7HI9T
Classification: IACT
SODIUM HYDROXIDEInactive
Code: 55X04QC32I
Classification: IACT
HYDROCHLORIC ACIDInactive
Code: QTT17582CB
Classification: IACT
EPINEPHRINE BITARTRATEActive
Quantity: 0.005 mg in 1 mL
Code: 30Q7KI53AK
Classification: ACTIM
LIDOCAINE HYDROCHLORIDE ANHYDROUSActive
Quantity: 5 mg in 1 mL
Code: EC2CNF7XFP
Classification: ACTIB

LIDOCAINE HYDROCHLORIDE

Product Details

FDA regulatory identification and product classification information

FDA Identifiers
NDC Product Code63323-487
Application NumberNDA006488
Product Classification
M
Marketing Category
C73594
G
Generic Name
LIDOCAINE HYDROCHLORIDE
Product Specifications
Route of AdministrationINFILTRATION, PERINEURAL, INTRACAUDAL, EPIDURAL
Effective DateAugust 28, 2020
FDA Product Classification

INGREDIENTS (7)

SODIUM CHLORIDEInactive
Quantity: 7 mg in 1 mL
Code: 451W47IQ8X
Classification: IACT
SODIUM METABISULFITEInactive
Quantity: 0.5 mg in 1 mL
Code: 4VON5FNS3C
Classification: IACT
HYDROCHLORIC ACIDInactive
Code: QTT17582CB
Classification: IACT
SODIUM HYDROXIDEInactive
Code: 55X04QC32I
Classification: IACT
CITRIC ACID MONOHYDRATEInactive
Quantity: 0.2 mg in 1 mL
Code: 2968PHW8QP
Classification: IACT
EPINEPHRINE BITARTRATEActive
Quantity: 0.005 mg in 1 mL
Code: 30Q7KI53AK
Classification: ACTIM
LIDOCAINE HYDROCHLORIDE ANHYDROUSActive
Quantity: 10 mg in 1 mL
Code: EC2CNF7XFP
Classification: ACTIB

LIDOCAINE HYDROCHLORIDE

Product Details

FDA regulatory identification and product classification information

FDA Identifiers
NDC Product Code63323-491
Application NumberNDA006488
Product Classification
M
Marketing Category
C73594
G
Generic Name
LIDOCAINE HYDROCHLORIDE
Product Specifications
Route of AdministrationINFILTRATION
Effective DateAugust 28, 2020
FDA Product Classification

INGREDIENTS (4)

SODIUM CHLORIDEInactive
Quantity: 8 mg in 1 mL
Code: 451W47IQ8X
Classification: IACT
SODIUM HYDROXIDEInactive
Code: 55X04QC32I
Classification: IACT
HYDROCHLORIC ACIDInactive
Code: QTT17582CB
Classification: IACT
LIDOCAINE HYDROCHLORIDE ANHYDROUSActive
Quantity: 5 mg in 1 mL
Code: EC2CNF7XFP
Classification: ACTIB

LIDOCAINE HYDROCHLORIDE

Product Details

FDA regulatory identification and product classification information

FDA Identifiers
NDC Product Code63323-492
Application NumberNDA006488
Product Classification
M
Marketing Category
C73594
G
Generic Name
LIDOCAINE HYDROCHLORIDE
Product Specifications
Route of AdministrationINFILTRATION, PERINEURAL, INTRACAUDAL, EPIDURAL
Effective DateAugust 28, 2020
FDA Product Classification

INGREDIENTS (4)

HYDROCHLORIC ACIDInactive
Code: QTT17582CB
Classification: IACT
SODIUM CHLORIDEInactive
Quantity: 7 mg in 1 mL
Code: 451W47IQ8X
Classification: IACT
SODIUM HYDROXIDEInactive
Code: 55X04QC32I
Classification: IACT
LIDOCAINE HYDROCHLORIDE ANHYDROUSActive
Quantity: 10 mg in 1 mL
Code: EC2CNF7XFP
Classification: ACTIB

LIDOCAINE HYDROCHLORIDE

Product Details

FDA regulatory identification and product classification information

FDA Identifiers
NDC Product Code63323-485
Application NumberNDA006488
Product Classification
M
Marketing Category
C73594
G
Generic Name
LIDOCAINE HYDROCHLORIDE
Product Specifications
Route of AdministrationINFILTRATION, PERINEURAL
Effective DateAugust 28, 2020
FDA Product Classification

INGREDIENTS (5)

SODIUM CHLORIDEInactive
Quantity: 7 mg in 1 mL
Code: 451W47IQ8X
Classification: IACT
SODIUM HYDROXIDEInactive
Code: 55X04QC32I
Classification: IACT
METHYLPARABENInactive
Quantity: 1 mg in 1 mL
Code: A2I8C7HI9T
Classification: IACT
HYDROCHLORIC ACIDInactive
Code: QTT17582CB
Classification: IACT
LIDOCAINE HYDROCHLORIDE ANHYDROUSActive
Quantity: 10 mg in 1 mL
Code: EC2CNF7XFP
Classification: ACTIB

LIDOCAINE HYDROCHLORIDE

Product Details

FDA regulatory identification and product classification information

FDA Identifiers
NDC Product Code63323-495
Application NumberNDA006488
Product Classification
M
Marketing Category
C73594
G
Generic Name
LIDOCAINE HYDROCHLORIDE
Product Specifications
Route of AdministrationINFILTRATION, PERINEURAL, INTRACAUDAL, EPIDURAL
Effective DateAugust 28, 2020
FDA Product Classification

INGREDIENTS (4)

SODIUM CHLORIDEInactive
Quantity: 6 mg in 1 mL
Code: 451W47IQ8X
Classification: IACT
SODIUM HYDROXIDEInactive
Code: 55X04QC32I
Classification: IACT
HYDROCHLORIC ACIDInactive
Code: QTT17582CB
Classification: IACT
LIDOCAINE HYDROCHLORIDE ANHYDROUSActive
Quantity: 20 mg in 1 mL
Code: EC2CNF7XFP
Classification: ACTIB

LIDOCAINE HYDROCHLORIDE,EPINEPHRINE BITARTRATE

Product Details

FDA regulatory identification and product classification information

FDA Identifiers
NDC Product Code63323-488
Application NumberNDA006488
Product Classification
M
Marketing Category
C73594
G
Generic Name
LIDOCAINE HYDROCHLORIDE,EPINEPHRINE BITARTRATE
Product Specifications
Route of AdministrationINFILTRATION, PERINEURAL, INTRACAUDAL, EPIDURAL
Effective DateAugust 28, 2020
FDA Product Classification

INGREDIENTS (7)

SODIUM CHLORIDEInactive
Quantity: 6.5 mg in 1 mL
Code: 451W47IQ8X
Classification: IACT
SODIUM METABISULFITEInactive
Quantity: 0.5 mg in 1 mL
Code: 4VON5FNS3C
Classification: IACT
HYDROCHLORIC ACIDInactive
Code: QTT17582CB
Classification: IACT
SODIUM HYDROXIDEInactive
Code: 55X04QC32I
Classification: IACT
EPINEPHRINE BITARTRATEActive
Quantity: 0.005 mg in 1 mL
Code: 30Q7KI53AK
Classification: ACTIM
CITRIC ACID MONOHYDRATEInactive
Quantity: 0.2 mg in 1 mL
Code: 2968PHW8QP
Classification: IACT
LIDOCAINE HYDROCHLORIDE ANHYDROUSActive
Quantity: 15 mg in 1 mL
Code: EC2CNF7XFP
Classification: ACTIB

LIDOCAINE HYDROCHLORIDE,EPINEPHRINE BITARTRATE

Product Details

FDA regulatory identification and product classification information

FDA Identifiers
NDC Product Code63323-483
Application NumberNDA006488
Product Classification
M
Marketing Category
C73594
G
Generic Name
LIDOCAINE HYDROCHLORIDE,EPINEPHRINE BITARTRATE
Product Specifications
Route of AdministrationINFILTRATION, PERINEURAL
Effective DateAugust 28, 2020
FDA Product Classification

INGREDIENTS (8)

CITRIC ACID MONOHYDRATEInactive
Quantity: 0.2 mg in 1 mL
Code: 2968PHW8QP
Classification: IACT
SODIUM CHLORIDEInactive
Quantity: 6 mg in 1 mL
Code: 451W47IQ8X
Classification: IACT
METHYLPARABENInactive
Quantity: 1 mg in 1 mL
Code: A2I8C7HI9T
Classification: IACT
SODIUM HYDROXIDEInactive
Code: 55X04QC32I
Classification: IACT
HYDROCHLORIC ACIDInactive
Code: QTT17582CB
Classification: IACT
EPINEPHRINE BITARTRATEActive
Quantity: 0.01 mg in 1 mL
Code: 30Q7KI53AK
Classification: ACTIM
SODIUM METABISULFITEInactive
Quantity: 0.5 mg in 1 mL
Code: 4VON5FNS3C
Classification: IACT
LIDOCAINE HYDROCHLORIDE ANHYDROUSActive
Quantity: 20 mg in 1 mL
Code: EC2CNF7XFP
Classification: ACTIB

Drug Labeling Information

DESCRIPTION SECTION

LOINC: 34089-3Updated: 8/28/2020

DESCRIPTION

Xylocaine (lidocaine HCl) Injections are sterile, nonpyrogenic, aqueous solutions that contain a local anesthetic agent with or without epinephrine and are administered parenterally by injection. SeeINDICATIONS AND USAGE section for specific uses.

Xylocaine solutions contain lidocaine HCl, which is chemically designated as acetamide, 2-(diethylamino)-N-(2,6-dimethylphenyl)-, monohydrochloride and has the molecular wt. 270.8. Lidocaine HCl (C14H22N2O • HCl) has the following structural formula:

structure 1

Epinephrine is (-) -3, 4-Dihydroxy-α-[(methylamino) methyl] benzyl alcohol and has the molecular wt. 183.21. Epinephrine (C9H13NO3) has the following structural formula:

structure 2

Dosage forms listed as Xylocaine-MPF indicate single dose solutions that are MethylParabenFree (MPF).

Xylocaine MPF is a sterile, nonpyrogenic, isotonic solution containing sodium chloride. Xylocaine in multiple dose vials: Each mL also contains 1 mg methyl­paraben as antiseptic preservative. The pH of these solutions is adjusted to approximately 6.5 (5.0 to 7.0) with sodium hydroxide and/or hydrochloric acid.

Xylocaine MPF with Epinephrine is a sterile, nonpyrogenic, isotonic solution containing sodium chloride. Each mL contains lidocaine hydrochloride and epinephrine, with 0.5 mg sodium metabisulfite as an antioxidant and 0.2 mg citric acid as a stabilizer. Xylocaine with Epinephrine in multiple dose vials: Each mL also contains 1 mg methylparaben as antiseptic preservative. The pH of these solutions is adjusted to approximately 4.5 (3.3 to 5.5) with sodium hydroxide and/or hydrochloric acid. Filled under nitrogen.

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