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biased agonists
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biased agonists
biased agonists
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摘要
临床试验
审批记录
专利
每项发明一条,涵盖美国、欧洲、PCT 与中国的同族专利。
HETEROCYCLIC COMPOUNDS AS 5HT2A BIASED AGONISTS
EP 4447954 A1
申请人: ICAHN SCHOOL MED MOUNT SINAI
优先权: 2021
EP
US
WO
3 件公开
WO 2026136510 A1
申请人: ICAHN SCHOOL MED MOUNT SINAI
优先权: 2024
WO
BETA CARBOLINE ANALOGUES AS SELECTIVE AND BIASED KAPPA OPIOID RECEPTORS AGONISTS FOR TREATING VARIOUS ASSOCIATED PATHOPHYSIOLOGICAL CONDITIONS
EP 4543880 A4
申请人: COUNCIL SCIENT IND RES
优先权: 2022
EP
US
WO
3 件公开
PREPARATION OF 3,4,5-TRISUBSTITUTED TRIAZOLES AND METHODS OF USING THE SAME
EP 4673133 A2
申请人: UNIV FLORIDA
优先权: 2023
EP
US
WO
3 件公开
Methods and compositions related to GPCR agonist polypeptides
US 10745456 B2
申请人: SCRIPPS RESEARCH INST
优先权: 2015
CN
US
2 件公开
HETEROCYCLE FUSED GAMMA-CARBOLINES ACTING ON THE SEROTONINE 5-HT2A RECEPTOR
EP 4642458 A1
申请人: INTRA CELLULAR THERAPIES INC
优先权: 2022
EP
WO
2 件公开
HIGHLY POTENT KAPPA OPIOID RECEPTOR AGONISTS AND METHOD OF USE THEREOF
EP 4798582 A1
申请人: UNIV NORTH CAROLINA CHAPEL HILL
优先权: 2023
EP
WO
2 件公开
Beta-arrestin-biased cannabinoid CB1 receptor agonists and methods for making and using them
US 10118914 B2
申请人: THE UNIV OF NORTH CAROLINA AT GREENSBORO
优先权: 2016
US
2 件公开
Biarylmethyl heterocycles
US 11407733 B2
申请人: UNIV MONTREAL
优先权: 2017
US
2 件公开
Substituted benzimidazoles as nociceptin receptor modulators
US 9656994 B2
申请人: SCRIPPS RESEARCH INST
优先权: 2014
US
Signaling-biased mu opioid receptor agonists
US 10751335 B2
申请人: SCRIPPS RESEARCH INST
优先权: 2017
US
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