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A Study of LY3484356 in Women With Breast Cancer Before Having Surgery

Phase 1
Completed
Conditions
Breast Cancer
Interventions
Registration Number
NCT04647487
Lead Sponsor
Eli Lilly and Company
Brief Summary

The purpose for this study is to see if the study drug, LY3484356, is safe and to determine what effects it has on breast cancer in participants with Estrogen Receptor Positive (ER+), HER2 Negative (HER2-) early stage (stage I-III) breast cancer, when given prior to surgery. Participation in this study could last up to 2.5 months.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
Female
Target Recruitment
86
Inclusion Criteria
  • Have histologically confirmed invasive ER+, HER2- breast carcinoma
  • Be willing and able to provide pre- and on-treatment tumor samples
  • Have a performance status of 0 or 1 on the Eastern Cooperative Oncology Group scale
  • Have adequate organ function
  • Be able to swallow capsules
  • Be a postmenopausal woman
Exclusion Criteria
  • Have bilateral invasive breast cancer
  • Have metastatic breast cancer
  • Plan to receive concurrent neoadjuvant therapy with any other non-protocol anti-cancer therapy
  • Have had prior therapy (of any kind) for an invasive or non-invasive breast cancer
  • Have had prior radiotherapy to the ipsilateral chest wall for any malignancy
  • Have had prior anti-estrogen therapy with raloxifene, tamoxifen, aromatase inhibitor, or other selective estrogen receptor modulator (SERM), either for osteoporosis or prevention of breast cancer
  • Have had prior hormone-replacement therapy within 4 weeks of the start of study treatment
  • Have had major surgery within 28 days prior to randomization to allow for post-operative healing of the surgical wound and site(s)
  • Have certain infections such as hepatitis or tuberculosis or HIV that are not well controlled
  • Have another serious medical condition
  • Have a history of any other cancer (except nonmelanoma skin cancer or carcinoma in-situ of the cervix), unless in complete remission with no therapy for a minimum of 3 years

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
LY3484356 Dose Level 1LY3484356Administered orally.
LY3484356 Dose Level 2LY3484356Administered orally.
LY3484356 Dose Level 3LY3484356Administered orally.
Primary Outcome Measures
NameTimeMethod
Change from Baseline in ER ExpressionBaseline, Day 15

ER expression measured by H-score immunohistochemistry (IHC)

Secondary Outcome Measures
NameTimeMethod
Change from Baseline in Ki-67 IndexBaseline, Day 15

Ki-67 index measured by percentage positive scoring by IHC

Change from Baseline in Progesterone Receptor (PR) ExpressionBaseline, Day 15

PR expression measured by H-score IHC

PK: Plasma Concentration of LY3484356Baseline through follow-up at Day 15

Trial Locations

Locations (19)

Northwestern Memorial Hosptial

🇺🇸

Chicago, Illinois, United States

Baylor College of Medicine

🇺🇸

Houston, Texas, United States

University of Texas MD Anderson Cancer Center

🇺🇸

Houston, Texas, United States

University of Vermont Medical Center

🇺🇸

Burlington, Vermont, United States

Massachusetts General Hospital

🇺🇸

Boston, Massachusetts, United States

Winship Cancer Center Emory University

🇺🇸

Atlanta, Georgia, United States

The Royal Cornwall Hospital

🇬🇧

Truro, Cornwall, United Kingdom

Sarah Cannon Research Institute SCRI

🇺🇸

Nashville, Tennessee, United States

Helios Kliniken Schwerin

🇩🇪

Schwerin, Mecklenburg-Vorpommern, Germany

Universitaire Ziekenhuizen Leuven - Campus Gasthuisberg

🇧🇪

Leuven, Belgium

Institut Jules Bordet

🇧🇪

Brussel - Capital, Belgium

Universitätsklinikum Erlangen

🇩🇪

Erlangen, Bayern, Germany

Klinikum der Universitaet Muenchen

🇩🇪

Muenchen, Germany

Hospital Clinic I Provincial

🇪🇸

Barcelona, Spain

Hospital General Universitario Gregorio Marañon

🇪🇸

Madrid, Spain

Barts Cancer Institute

🇬🇧

London, London City, United Kingdom

Washington University School of Medicine

🇺🇸

Saint Louis, Missouri, United States

Hospital Madrid Norte Sanchinarro

🇪🇸

Madrid, Spain

Hôpital René Huguenin

🇫🇷

Saint-Cloud, Hauts-de-Seine, France

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