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The Effect of Acipimox on GLP (Glucagon-like Peptide)-1 Secretion

Not Applicable
Completed
Conditions
Diabetes Mellitus Type 2
Interventions
Registration Number
NCT02796950
Lead Sponsor
University of Aarhus
Brief Summary

Glucagon like peptide 1 is produced in enteroendocrine L cells in the small intestine stimulated by peroral food intake. GLP-1 induces insulin secretion, and analogues are used in the treatment of DM2 (type 2 diabetes mellitus). Recently it was found, that levels of GLP-1 are increased in response to acipimox. The hypothesis is that G protein coupled receptors on enteroendocrine L cells bind acipimox and thereby induce GLP-1 secretion.

In a controlled, open, randomized experiment, eight healthy, overweight men will be studied on an intervention day, where they receive acipimox, and on a control day. The study day includes an OGTT (oral glucose tolerance test), blood samples before and after the OGTT and a biopsy from adipose tissue.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
8
Inclusion Criteria
  • Adult men
  • Healthy
  • BMI 25-35
Exclusion Criteria
  • Known DM2
  • Receiving hypolipidemic drugs

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
AcipimoxAcipimoxAdministration of acipimox 250 mg p.o.
Primary Outcome Measures
NameTimeMethod
Levels of GLP-1 in plasma9 months
Secondary Outcome Measures
NameTimeMethod
Lipolytic activity in adipose tissue by measuring FFA (free fatty acid) levels9 months
Insulin sensitivity by measuring blood glucose after an OGTT5 months

Trial Locations

Locations (1)

University Hospital of Aarhus

🇩🇰

Aarhus, Denmark

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