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A Phase 2 Study to Evaluate the Efficacy and Safety of 60mg of MM-093 in Patients With Active Rheumatoid Arthritis

Phase 2
Completed
Conditions
Rheumatoid Arthritis
Interventions
Registration Number
NCT00458146
Lead Sponsor
Merrimack Pharmaceuticals
Brief Summary

The purpose of this study is to determine whether MM-093 is safe and effective in the treatment of RA.

Detailed Description

To evaluate the safety and tolerability of 60 mg of MM-093 in patients who have active RA despite MTX background therapy.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
100
Inclusion Criteria
  • Meet American College of Rheumatology (ACR) criteria for RA.
  • Have active RA consisting of > or equal to 6 tender joints and > or equal to 6 swollen joints and one of the following:CRP or ESR levels of ULN
  • Have an ACR functional class of I-III.
  • Have had RA for at least 6 months.
  • Had disease onset at > 16 years of age.
  • Aged 18 - 80 years.
  • Currently being treated with a stable, well tolerated weekly dose of MTX between 10-25 mg for at least 6 consecutive prior to screening visit.
  • Currently being treated with folic/folinic acid in conjunction with their MTX treatment.

(Note: Patients may begin folic/folinic acid treatment after their screening visit, but must remain on stable dose for two weeks before undergoing the Day 1 assessments.)

  • Willing to remain on a constant, weekly dose of MTX and folic/folinic acid through out the duration of the study.
  • Understand, sign, and date the written, voluntary informed consent form at the screening visit prior to any protocol - specific procedures being performed.
  • Be able and willing to comply with study visits and procedures per protocol.
  • Women of childbearing potential must use a medically acceptable means of birth control in an effective manner and agree to continue its use during the study and for 4 weeks after the last dose of study drug. Women who have had a complete surgical hysterectomy or are postmenopausal (absence of menstrual period for at least one year or > 52 years old) are exempt from this requirement. Medically acceptable forms of birth control include oral contraceptives, injectable or implantable methods, intrauterine devices, tubal ligation (if performed more than 1 year before screening), or properly used barrier contraception. Additionally, the use of condoms is suggested as an adjunct to the methods previously addressed to protect against sexually transmitted diseases and to provide additional protection against accidental pregnancy.
  • Sexually active men must agree to use a medically acceptable form of contraception during the study and continue for 4 weeks after the last dose of study drug.
  • Able to store patient kit/cooler containing drug in a refrigerator at home.
Exclusion Criteria
  • Patient will be excluded if any of the following prior medications are currently being used or have used within the designated time interval before the screening visit:

    1. Any B - cell or antibody depleting therapy , including plasmaphoresis or Prosorba columns (6 months)
    2. Leflunomide, Adalimumab (Humira)(3 months)
    3. Investigational biologics (2 months)
    4. Infliximab (Remicade) (2 months)
    5. Cyclosporine, sulphasalazine, auranofin, intramuscular gold, azathioprine, D-penicillamine, tacrolimus (6 weeks)
    6. Investigational small molecules (e.g. NSAIDS or Cox-2 inhibitors)(4 weeks)
    7. Use more than 10mg/day of prednisone or equivalent (4 weeks)
    8. Bolus intramuscular/intravenous (IM/IV) treatment with corticosteroids (>20 mg prednisone or equivalent)(4 weeks)
    9. Intra-articular corticosteroid injection (4 weeks)
    10. Etanercept (Enbrel) (4 weeks)
    11. Anakinra (Kineret) (2 weeks)
    12. Use of more than one NSAID (current)
    13. Dose of NSAID greater than maximum recommended dose in the product information (current)
  • Significant concurrent medical diseases including:

    1. Cancer, or a history of cancer (other than successfully resected cutaneous basal and squamous cell carcinoma) within 5 years before the screening visit.
    2. Any condition for which participation in this study is judged by the physician to be detrimental to the patient, such as history of significant or unstable cardiac, pulmonary, gastrointestinal, neurological, or psychiatric disease, or a DMARD-related severe, potentially life threatening AE.
    3. Significant ongoing infection requiring systemic antibiotic, antifungal, antiviral, or anti-myobacterial therapy.
  • Autoimmune or connective tissue disorder other than rheumatoid arthritis (e.g. Systemic Lupus Erythematosis, Scleroderma, or Psoriatic Arthritis)

  • Grade 2 or above leukopenia (i.e. white blood cells < 3000/mm^3 [SI units: < 3.0 x 10^9/L)

  • Thrombocytopenia or thrombocytosis (platelets > 125,000/mm^3 or > 1,000,000/mm^3 [SI units: < 125 x 10^9/L or > 1,000 x 10^9/L]), respectively.

  • Grade 2 or above liver function abnormality(i.e. total bilirubin .1.5 x the upper limit of normal; or aspartate aminotransfersate [AST/SGOT] or alanine aminotransferase [ALT/SGPT]> 2.5 x upper limit of normal.

  • Renal disease (including serum creatinine level > 1.5 x the upper limit of normal).

  • Any history of immunodeficiency syndromes or infection with human immunodeficiency virus (HIV), or a history of hepatitis C or chronic hepatitis B.

  • Pregnant or breastfeeding women or women planning to become pregnant during the study or within 4 weeks after the last dose of study drug.

  • Any major surgery, including joint surgery, within 3 months before the screening visit.

  • Scheduled elective surgery during the study participation.

  • Participated in any previous clinical trial using MM-093 or have any prior exposure to MM-093.

  • History of severe hypersensitivity to goat, sheep, or cow milk. (Patients who are lactose intolerant are not excluded).

  • Any other condition that the investigator feels would jeopardize the integrity of the study (e.g. a CTCAE grade 2 or above clinical finding or laboratory result).

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
1MM-093MM-093
2MM-093Placebo
Primary Outcome Measures
NameTimeMethod
Evaluate the efficacy of MM-093 using ACR20 response rateAfter three months of treatment
Secondary Outcome Measures
NameTimeMethod
Evaluate the efficacy of MM-093 using DAS-28 and EULARAfter three months of treatment

Trial Locations

Locations (20)

East Valley Rheumatology & Osteoporosis

🇺🇸

Gilbert, Arizona, United States

Arthritis and Rheumatic Disease Specialties

🇺🇸

Aventura, Florida, United States

Montgomery Rheumatology Associates

🇺🇸

Montgomery, Alabama, United States

New England Research Associates

🇺🇸

Trumbull, Connecticut, United States

Arthritis Center of Nebraska

🇺🇸

Lincoln, Nebraska, United States

East Pennsylvania Rheumatology Association

🇺🇸

Bethlehem, Pennsylvania, United States

Wichita Clinic

🇺🇸

Wichita, Kansas, United States

Illinois Bone & Joint Institute

🇺🇸

Morton Grove, Illinois, United States

National Jewish Medical and Research Center

🇺🇸

Denver, Colorado, United States

Denver Arthritis Clinic

🇺🇸

Denver, Colorado, United States

University of Utah Division of Rheumatology

🇺🇸

Salt Lake City, Utah, United States

Sarasota Arthritis Research Center

🇺🇸

Sarasota, Florida, United States

Arthritis Research of Florida, Inc.

🇺🇸

Palm Harbor, Florida, United States

Paddock Park Clinical Research

🇺🇸

Ocala, Florida, United States

Arthritis Center of Reno

🇺🇸

Reno, Nevada, United States

Arthritis Center and Carolina Bone and Joint

🇺🇸

Charlotte, North Carolina, United States

Rheumatology and Internal Medicine

🇺🇸

Amarillo, Texas, United States

Altoona Center for Clinical Research

🇺🇸

Duncansville, Pennsylvania, United States

Arthritis Medical Center of the Central Coast

🇺🇸

Santa Maria, California, United States

Radiant Research

🇺🇸

Scottsdale, Arizona, United States

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