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Extracorporeal Photopheresis of Patients With Crohn's Disease Using 5-aminolevulinic Acid

Phase 1
Completed
Conditions
Crohn Disease
Interventions
Procedure: Blue light photopheresis
Procedure: Transfusion
Procedure: Continuous Mononuclear Cell Collection (CMNC)
Registration Number
NCT04164849
Lead Sponsor
University Hospital, Akershus
Brief Summary

In the clinical trial the investigators will assess efficacy, safety and tolerability after single and multiple doses of 3 millimolar 5 aminolevulinic acid (Gliolan®) in combination with blue-light (405 nanometer) photopheresis in patients with active crohns disease. The study is a proof-of-concept pilot with up to 10 included patients where every patient will get active treatment. The use of 5-aminolevulinic acid in combination with blue-light photopheresis is a first-in-human trial. Primary endpoints include clinical response and adverse events (safety). Secondary endpoints include endoscopic improvement, quality of life questionnaires, faecal calprotectin, C-reactive protein and mechanisms of action (differences in t-cells and other cells before and after treatment). All patients will get treatment every 2 weeks for 10 weeks (6 treatments-induction) with evaluation at week 13. If any effect on week 13 eligible for study extension with treatment every 4 weeks for up to 12 months for the first 5 patients. The latter 5 patients will be referred to standard of care on the week 13 visit. Through the study the investigators will see if this kind of photopheresis is safe and can be an option for a larger randomized-controlled-trial. In addition the investigators will see if photopheresis as an option can be further developed for other diseases as well (ie other T-cell mediated diseases or patients already receiving photopheresis as a treatment).

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
7
Inclusion Criteria
  1. Provision of informed consent

  2. Age above 18

  3. Male or female patient with active Crohn's disease (6)

  4. Women of childbearing potential (WOCBP) will have to use highly effective methods of contraception throughout the entire study.

  5. Inadequate response (a) or intolerance to biological therapy

    a. Inadequate response on ongoing treatment is defined as: i. Progressive disease: increasing Harvey Bradshaw Index/Calprotectin/Simple Endoscopic Score for Crohns Disease and/or worsening of radiologic images after 6 months.

    ii. Stable disease: no-response after 6 months

  6. Active inflammation in the gut documented by

    1. Harvey Bradshaw Index >5 and
    2. Endoscopy with Simple Endoscopic Score for Crohns Disease equal to or above 6 points or equal to or above 4 points if only isolated ileitis is present and/or
    3. Inflammatory marker; fecal calprotectin > 250 and/or C reactive protein > 5
Exclusion Criteria
  1. Photosensitive comorbidities, porphyria or known hypersensitivity to 5-aminolevulinic acid or porphyrins
  2. Patients with aphakia
  3. Pregnant or breast-feeding women. A negative urine pregnancy test must be demonstrated in female patients of child-bearing potential at the Screening Visit and before every treatment.
  4. Ongoing cardiac and pulmonary diseases or aspartate transaminase alanine aminotransferase, Bilirubin or International Normalized Ratio value ≥ 3x upper limit of normal or clinically significant electrocardiogram findings
  5. Subjects with polyneuropathy
  6. Uncontrolled infection or fever
  7. History of heparin-induced thrombocytopenia, absolute neutrophil count <1x109, platelet count <20x10 9
  8. Body weight below 40 kg
  9. Investigator considers subject unlikely to comply with study procedures, restrictions and requirements.
  10. Presence of other gastrointestinal diseases potentially influencing the study endpoints
  11. History of any clinically significant disease or disorder which in the opinion of the investigator, may either put the patient at risk because of participation in the study, or influence the result or the patient's ability to participate in the study.

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
5-ALA photopheresis5-aminolevulinic acidAll patients will receive 5-aminolevulinic acid (5-ALA) in combination with blue light photopheresis. The investigators will collect mononuclear cells by connecting patient to Spectra Optia with CMNC (continuous mononuclear cell collection protocol), and these cells will include active T-lymphocytes. 5-ALA will be incubated for 1 hour to produce photoactive protoporphyrin-IX (PpIX) before light exposure.
5-ALA photopheresisBlue light photopheresisAll patients will receive 5-aminolevulinic acid (5-ALA) in combination with blue light photopheresis. The investigators will collect mononuclear cells by connecting patient to Spectra Optia with CMNC (continuous mononuclear cell collection protocol), and these cells will include active T-lymphocytes. 5-ALA will be incubated for 1 hour to produce photoactive protoporphyrin-IX (PpIX) before light exposure.
5-ALA photopheresisTransfusionAll patients will receive 5-aminolevulinic acid (5-ALA) in combination with blue light photopheresis. The investigators will collect mononuclear cells by connecting patient to Spectra Optia with CMNC (continuous mononuclear cell collection protocol), and these cells will include active T-lymphocytes. 5-ALA will be incubated for 1 hour to produce photoactive protoporphyrin-IX (PpIX) before light exposure.
5-ALA photopheresisContinuous Mononuclear Cell Collection (CMNC)All patients will receive 5-aminolevulinic acid (5-ALA) in combination with blue light photopheresis. The investigators will collect mononuclear cells by connecting patient to Spectra Optia with CMNC (continuous mononuclear cell collection protocol), and these cells will include active T-lymphocytes. 5-ALA will be incubated for 1 hour to produce photoactive protoporphyrin-IX (PpIX) before light exposure.
Primary Outcome Measures
NameTimeMethod
Clinical responseWeek 13, 26 (28 for patients not eligible for study extension and the latter 5 patients), 38, 50, 64 and 3 months after last treatment

Clinical response (Harvey Bradshaw Index change \> 3 from baseline or less than 4 points)

Safety and tolerability Electrocardiogram-PR segmentBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in PR segment before and after treatment

Safety and tolerability Electrocardiogram-T waveBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in T wave before and after treatment

Safety and tolerability Electrocardiogram-QRS complexBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in QRS complex before and after treatment

Alkaline phosphataseBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in serum alkaline phosphatase (U/L) before and after treatment

BilirubinBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Serum Bilirubin (micromol/L) before and after treatment

Safety and tolerability adverse eventsBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Frequency, seriousness and intensity of adverse events

Safety and tolerability Electrocardiogram-QT intervalBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in QT interval before and after treatment

Safety and tolerability Electrocardiogram-PR intervalBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in PR interval before and after treatment

Alanine aminotransferaseBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in serum alanine aminotransferase (U/L) before and after treatment

AlbuminBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Serum Albumin (g/L) before and after treatment

Safety and tolerability blood pressureBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Vital signs (systolic and diastolic blood pressure) before and after treatment

Aspartate transferaseBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in serum aspartate transferase(U/L) before and after treatment

White cell countBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Blood White cell count (10\^9/L) before and after treatment

Safety and tolerability Electrocardiogram-ST segmentBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in ST segment before and after treatment

Safety and tolerability vital signsBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Vital signs (heart rate) before and after treatment

Gamma glutamyltransferaseBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Serum gamma glutamyltransferase (U/L) before and after treatment

Neutrophil granulocytesBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Blood neutrophil granulocytes (10\^9/L) before and after treatment

LymphocytesBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Blood Lymphocytes (10\^9/L) before and after treatment

MonocytesBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Blood Monocytes (10\^9/L) before and after treatment

Eosinophile granulocytesBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Blood Eosinophile granulocytes (10\^9/L) before and after treatment

Basophile granulocytesBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Blood Basophile granulocytes (10\^9/L) before and after treatment

Platelet countBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Blood Platelet count (10\^9/L) before and after treatment

Mean Cell VolumeBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Blood Mean Cell Volume (fL) before and after treatment

Mean Cell hemoglobinBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Blood Mean Cell hemoglobin (picogram) before and after treatment

International Normalized RatioBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Blood International Normalized Ratio (0,8-1,2) before and after treatment

HemoglobinBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Blood Hemoglobin (g/dL) before and after treatment

CalciumBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Serum Calcium (millimol/L) before and after treatment

PotassiumBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Serum Potassium (millimol/L) before and after treatment

SodiumBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Serum Sodium (millimol/L) before and after treatment

CreatininBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Serum Creatinine (micromol/L) before and after treatment

Total ProteinBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Serum Total Protein (g/L) before and after treatment

Lactate DehydrogenaseBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Serum Lactate Dehydrogenase (U/L) before and after treatment

CholesterolBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Serum Cholesterol (millimol/L) before and after treatment

CarbamideBefore every treatment visit (every second week from week 0-10, every 4th week from week 14-62, week 28 for patients not eligible for study extension and latter 5 patients) in addition to week 64 and 3 months after last treatment.

Changes in Serum Carbamide (millimol/L) before and after treatment

Secondary Outcome Measures
NameTimeMethod
Quality of life questionnaire Short-Form 36 (SF-36)Week 13, 26 (28 for patients not eligible for study extension and the latter 5 patients), 38, 50, 64 and/or 3 months after last treatment

Change of both total and subscores of SF-36 from baseline. Min 0 Max 100. Higher value is better quality of life.

Quality of life questionnaire Inflammatory Bowel Disease Questionnaire (IBDQ)Week 13, 26 (28 for patients not eligible for study extension and the latter 5 patients), 38, 50, 64 and/or 3 months after last treatment

Change of both total and subscores of IBDQ from baseline. Min 32 Max 224. Higher value is better quality of life.

CD4+ and CD8+ T cell subpopulationsWeek 0, 10 (all patients) and 50 (patients of the first 5 subjects eligible for study extension)

Number of CD4+ and CD8+ T cell subpopulations before and after treatment assessed by flow cytometry.

Endoscopic efficacyWeek 13 (all patients) and 64 (patients of the first 5 subjects eligible for study extension) with baseline visit as reference.

Simple Endoscopic Score for Crohns Disease \>49 % improvement or \< 3 (endoscopic remission)

Faecal calprotectinWeek 13, 26 (28 for patients not eligible for study extension and the latter 5 patients), 38, 50, 64 and/or 3 months after last treatment

Change from baseline

Concentration of C reactive protein in bloodWeek 13, 26 (28 for patients not eligible for study extension and the latter 5 patients), 38, 50, 64 and/or 3 months after last treatment

Change from baseline

Apoptosis and necrosisWeek 0, 10 (all patients) and 50 (patients of the first 5 subjects eligible for study extension)

Number of cells in apoptosis or necrosis before and after treatment assessed by flow cytometry

Clinical remissionWeek 13 and/or sustained/delayed response in week 26 (28 for patients not eligible for study extension and the latter 5 patients), 38, 50, 64 and 3 months after last treatment.

Harvey Bradshaw Index \< 5 points

Trial Locations

Locations (1)

Akershus University Hospital

🇳🇴

Lorenskog, Akershus, Norway

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