MedPath

A Study to Evaluate the Efficacy, Safety, and Pharmacokinetics of UTTR1147A Compared With Placebo and With Vedolizumab in Participants With Moderate to Severe Ulcerative Colitis (UC)

Phase 2
Completed
Conditions
Ulcerative Colitis
Interventions
Drug: UTTR1147A
Drug: UTTR1147A Placebo
Registration Number
NCT03558152
Lead Sponsor
Genentech, Inc.
Brief Summary

This study is designed to evaluate the efficacy, safety, and pharmacokinetics of UTTR1147A compared with vedolizumab and with placebo in the treatment of participants with moderate to severe UC. This study will consist of two parts, Part A and Part B. Part A will test the induction of clinical remission and Part B will test the durability of clinical remission.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
195
Inclusion Criteria
  • Diagnosis of UC
  • Confirmation of moderately to severely active UC, defined by the Mayo Clinic Score
  • Inadequate response, loss of response, or intolerance to prior immunosuppressant treatment (i.e., azathioprine, 6-mercaptopurine, methotrexate, or tumor necrosis factor [TNF] inhibitors [maximum of 2 prior TNF inhibitors]) and/or corticosteroid treatment
  • Use of highly effective contraception as defined by the protocol
Exclusion Criteria
  • History of psoriasis or psoriatic arthritis; any other inflammatory skin disorders requiring oral corticosteroids, immunosuppressants, or biological therapy within the previous year; or primary sclerosing cholangitis
  • History of cancer as defined by the protocol
  • Significant uncontrolled comorbidity, such as cardiac, pulmonary, renal, hepatic, endocrine, or gastrointestinal disorders (excluding UC)
  • Prior extensive colonic resection, subtotal or total colectomy, or proctocolectomy, or planned surgery for UC
  • Diagnosis of indeterminate colitis or granulomatous (Crohn's) colitis or toxic megacolon within 12 months prior to screening
  • Suspicion of ischemic colitis, radiation colitis, or microscopic colitis
  • Current fistula or history of fistula, pericolonic abscess and stricture (stenosis) of the colon
  • History or current evidence of unresectable colonic mucosal dysplasia or history of high-grade colonic mucosal dysplasia
  • Prior treatment with UTTR1147A
  • Prior treatment with vedolizumab, etrolizumab, natalizumab, efalizumab, or any other anti-integrin agents
  • Prior treatment with rituximab
  • Use of prohibited therapies, as defined by the protocol, prior to randomization
  • Congenital or acquired immune deficiency
  • Evidence or treatment of infections or history of infections, as defined by the protocol

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Arm 3a: UTTR1147A Dose Level 3 (Part A) + UTTR1147A (Part B)Vedolizumab PlaceboPart A: UTTR1147A dose level 3 and Vedolizumab Placebo. Part B: UTTR1147A maintenance dose and Vedolizumab Placebo.
Arm 3b: UTTR1147A Dose Level 3 (Part A) + Placebo (Part B)Vedolizumab PlaceboPart A: UTTR1147A dose level 3 and Vedolizumab Placebo. Part B: UTTR1147A Placebo and Vedolizumab Placebo.
Arm 1a: UTTR1147A Dose Level 1 (Part A) + UTTR1147A (Part B)UTTR1147APart A: UTTR1147A dose level 1 and Vedolizumab Placebo. Part B: UTTR1147A maintenance dose and Vedolizumab Placebo.
Arm 1a: UTTR1147A Dose Level 1 (Part A) + UTTR1147A (Part B)Vedolizumab PlaceboPart A: UTTR1147A dose level 1 and Vedolizumab Placebo. Part B: UTTR1147A maintenance dose and Vedolizumab Placebo.
Arm 1b: UTTR1147A Dose Level 1 (Part A) + Placebo (Part B)UTTR1147APart A: UTTR1147A dose level 1 and Vedolizumab Placebo. Part B: UTTR1147A Placebo and Vedolizumab Placebo.
Arm 1b: UTTR1147A Dose Level 1 (Part A) + Placebo (Part B)UTTR1147A PlaceboPart A: UTTR1147A dose level 1 and Vedolizumab Placebo. Part B: UTTR1147A Placebo and Vedolizumab Placebo.
Arm 1b: UTTR1147A Dose Level 1 (Part A) + Placebo (Part B)Vedolizumab PlaceboPart A: UTTR1147A dose level 1 and Vedolizumab Placebo. Part B: UTTR1147A Placebo and Vedolizumab Placebo.
Arm 2a: UTTR1147A Dose Level 2 (Part A) + UTTR1147A (Part B)UTTR1147APart A: UTTR1147A dose level 2 and Vedolizumab Placebo. Part B: UTTR1147A maintenance dose and Vedolizumab Placebo.
Arm 2a: UTTR1147A Dose Level 2 (Part A) + UTTR1147A (Part B)Vedolizumab PlaceboPart A: UTTR1147A dose level 2 and Vedolizumab Placebo. Part B: UTTR1147A maintenance dose and Vedolizumab Placebo.
Arm 2b: UTTR1147A Dose Level 2 (Part A) + Placebo (Part B)UTTR1147APart A: UTTR1147A dose level 2 and Vedolizumab Placebo. Part B: UTTR1147A Placebo and Vedolizumab Placebo.
Arm 2b: UTTR1147A Dose Level 2 (Part A) + Placebo (Part B)UTTR1147A PlaceboPart A: UTTR1147A dose level 2 and Vedolizumab Placebo. Part B: UTTR1147A Placebo and Vedolizumab Placebo.
Arm 2b: UTTR1147A Dose Level 2 (Part A) + Placebo (Part B)Vedolizumab PlaceboPart A: UTTR1147A dose level 2 and Vedolizumab Placebo. Part B: UTTR1147A Placebo and Vedolizumab Placebo.
Arm 3a: UTTR1147A Dose Level 3 (Part A) + UTTR1147A (Part B)UTTR1147APart A: UTTR1147A dose level 3 and Vedolizumab Placebo. Part B: UTTR1147A maintenance dose and Vedolizumab Placebo.
Arm 3b: UTTR1147A Dose Level 3 (Part A) + Placebo (Part B)UTTR1147APart A: UTTR1147A dose level 3 and Vedolizumab Placebo. Part B: UTTR1147A Placebo and Vedolizumab Placebo.
Arm 3b: UTTR1147A Dose Level 3 (Part A) + Placebo (Part B)UTTR1147A PlaceboPart A: UTTR1147A dose level 3 and Vedolizumab Placebo. Part B: UTTR1147A Placebo and Vedolizumab Placebo.
Arm 4: VedolizumabUTTR1147A PlaceboParts A and B: Vedolizumab and UTTR1147A Placebo.
Arm 5: PlaceboUTTR1147A PlaceboParts A and B: UTTR1147A Placebo and Vedolizumab Placebo.
Arm 5: PlaceboVedolizumab PlaceboParts A and B: UTTR1147A Placebo and Vedolizumab Placebo.
Arm 4: VedolizumabVedolizumabParts A and B: Vedolizumab and UTTR1147A Placebo.
Primary Outcome Measures
NameTimeMethod
Percentage of Participants With Clinical Remission at Week 88 weeks

Clinical remission is defined as modified Mayo Clinic Score (mMCS) \<= 2 with Mayo rectal bleeding subscore = 0, Mayo stool frequency subscore \<=1 and Centrally read endoscopic score \<= 1. Patients were classified as Non-Remitters if Week 8 assessments were missing or patient received permitted/ prohibited Rescue Therapy prior to assessment.

Secondary Outcome Measures
NameTimeMethod
Percentage of Participants With Sustained RemissionAt Weeks 8 and 30

Sustained remission is defined as clinical remission at both Week 8 and Week 30, where clinical remission is defined as modified Mayo Clinic Score (mMCS) \<= 2 with Mayo rectal bleeding subscore = 0, Mayo stool frequency subscore \<=1 and Centrally read endoscopic score \<= 1.

Patients were classified as Non-Remitters at Week 8 or at Week 30 if assessments were missing or patient received permitted/prohibited Rescue Therapy prior to assessment

Maximum Serum Concentration (Cmax) of UTTR1147ADays 1 - 29, Visit: Day 57
Percentage of Participants With Endoscopic Remission at Week 30At Week 30

Endoscopic remission is defined as a Mayo endoscopic subscore of 0. Patients were classified as Non-Responders if assessments were missing or patient received permitted/prohibited Rescue Therapy prior to assessment.

Change From Baseline in UC Bowel Movement Signs and Symptoms at Week 8, as Assessed by Ulcerative Colitis Patient-Reported Outcome Signs and Symptoms (UC-PRO/SS) ScoreAt Week 8

The UC-PRO is being reported in three domains; two domains are key endpoints and reported as UC-PRO Signs and Symptoms (UC-PRO/SS). The bowel domain score ranges from 0-27, with a higher score indicating a worse disease state.

Change From Baseline in UC Abdominal Signs and Symptoms at Week 8, as Assessed by Ulcerative Colitis Patient-Reported Outcome Signs and Symptoms (UC-PRO/SS) ScoreAt Week 8

The UC-PRO is being reported in three domains; two domains are key endpoints and reported as UC-PRO Signs and Symptoms (UC-PRO/SS). The functional (abdominal symptoms) domain score ranges from 0-12, with a higher score indicating a worse disease state.

Percentage of Participants With Clinical Response at Week 8At Week 8

Clinical response is defined as achieving clinical remission or as meeting both of the following criteria: A \>= 3-point decrease from baseline in modified Mayo Clinic Score (mMCS); A \>= 1-point decrease from baseline in rectal bleeding subscore or a rectal bleeding subscore of 0 or 1.

Patients were classified as Non-Responders if assessments were missing or patient received permitted/prohibited Rescue Therapy prior to assessment.

NOTE: An Outcome Measure Description has not been entered.

Percentage of Participants With Clinical Response at Week 30At Week 30

Clinical response is defined as achieving clinical remission or as meeting both of the following criteria: A \>= 3-point decrease from baseline in modified Mayo Clinic Score (mMCS); A \>= 1-point decrease from baseline in rectal bleeding subscore or a rectal bleeding subscore of 0 or 1.

Patients were classified as Non-Responders if assessments were missing or patient received permitted/prohibited Rescue Therapy prior to assessment.

Minimum Serum Concentration (Cmin) of UTTR1147ADays 1 - 29, Visit: Day 57
Percentage of Participants With Endoscopic Healing at Week 30At Week 30

Endoscopic healing is defined as a Mayo endoscopic subscore \<= 1. Patients were classified as Non-Responders if assessments were missing or patient received permitted/prohibited Rescue Therapy prior to assessment.

Percentage of Participants With Endoscopic Healing at Week 8At Week 8

Endoscopic healing is defined as a Mayo endoscopic subscore \<= 1. Patients were classified as Non-Responders if assessments were missing or patient received permitted/prohibited Rescue Therapy prior to assessment.

Change From Baseline in UC Bowel Movement Signs and Symptoms at Week 30, as Assessed by Ulcerative Colitis Patient-Reported Outcome Signs and Symptoms (UC-PRO/SS) ScoreAt Week 30

The UC-PRO is being reported in three domains; two domains are key endpoints and reported as UC-PRO Signs and Symptoms (UC-PRO/SS). The bowel domain score ranges from 0-27, with a higher score indicating a worse disease state.

Percentage of Participants With Endoscopic Remission at Week 8At Week 8

Endoscopic remission is defined as a Mayo endoscopic subscore of 0. Patients were classified as Non-Responders if assessments were missing or patient received permitted/prohibited Rescue Therapy prior to assessment.

Change From Baseline in UC Abdominal Signs and Symptoms at Week 30, as Assessed by Ulcerative Colitis Patient-Reported Outcome Signs and Symptoms (UC-PRO/SS) ScoreAt Week 30

The UC-PRO is being reported in three domains; two domains are key endpoints and reported as UC-PRO Signs and Symptoms (UC-PRO/SS). The functional (abdominal symptoms) domain score ranges from 0-12, with a higher score indicating a worse disease state.

Change From Baseline in Patient-Reported Inflammatory Bowel Disease Questionnaire (IBDQ) Score at Week 8At Week 8

The IBDQ score is a Total Score summed up from across all 32 questions on the questionnaire. The Total Score range is from 32 to 224 with higher scores representing a better quality of life.

Change From Baseline in Patient-Reported Inflammatory Bowel Disease Questionnaire (IBDQ) Score at Week 30At Week 30

The IBDQ score is a Total Score summed up from across all 32 questions on the questionnaire. The Total Score range is from 32 to 224 with higher scores representing a better quality of life.

Percentage of Participants With Adverse EventsUp to 30 weeks
Percentage of Participants With Presence of Anti-Drug Antibodies (ADA) at Baseline and After Drug AdministrationBaseline up to 30

Trial Locations

Locations (72)

Synexus Polska Sp. z o.o. Oddzial w Gdansku

🇵🇱

Gda?sk, Poland

Clinical Hospital Center Zvezdara

🇷🇸

Belgrade, Serbia

Klimed Marek Klimkiewicz

🇵🇱

Piotrków Trybunalski, Poland

Gastromed Kopon Zmudzinski i

🇵🇱

Toru?, Poland

Complesso Integrato Columbus

🇮🇹

Roma, Lazio, Italy

Synexus Polska Sp. z o.o. Oddzial w Czestochowie

🇵🇱

Cz?stochowa, Poland

Synexus Polska Sp. z o.o. Oddzial we Wroclawiu

🇵🇱

Wroc?aw, Poland

Melita Medical

🇵🇱

Wroc?aw, Poland

Portiuncula Hospital, Ballinasloe

🇮🇪

Co Galway, Ireland

Policlinico Universitario Campus Biomedico Di Roma

🇮🇹

Roma, Lazio, Italy

Synexus - Katowice

🇵🇱

Katowice, Poland

Synexus Polska Sp. z o.o. Oddzial w Poznaniu

🇵🇱

Pozna?, Poland

Clinical Hospital Centre Zemun

🇷🇸

Zemun, Serbia

Clinical Center Kragujevac; Clinic Of Psychiatry

🇷🇸

Kragujevac, Serbia

General Hospital Vrsac

🇷🇸

Vrsac, Serbia

Medical University Reaviz

🇷🇺

Samara, Russian Federation

Universitätsklinikum Ulm; Klinik für Innere Medizin II

🇩🇪

Ulm, Germany

Carolina Digestive Diseases

🇺🇸

Greenville, North Carolina, United States

University of Utah School of Medicine; Gastroenterology Division

🇺🇸

Salt Lake City, Utah, United States

MHAT Saint Karidad EAD

🇧🇬

Plovdiv, Bulgaria

LLC ARENSIA Exploratory Medicine

🇬🇪

Tbilisi, Georgia

Multiprofile Hospital for Active Treatment Hadji Dimitar OOD

🇧🇬

Sliven, Bulgaria

Gastroenterologische Spezialpraxis-Berlin-Karlshorst

🇩🇪

Berlin, Germany

Universitaetsklinikum Carl Gustav Carus TU Dresden

🇩🇪

Dresden, Germany

St. Marien Krankenhaus; Med. Klinik

🇩🇪

Ludwigshafen, Germany

Universitatsklinikum Schleswig-Holstein

🇩🇪

Lubeck, Germany

Iatriko Palaiou Falirou; Gastrointestinal Department

🇬🇷

Palaio Faliro, Greece

Shaare Zedek Medical Center; Bait Vagan

🇮🇱

Jerusalem, Israel

Magyar Honvédség Egészségügyi Központ; Országos Haemophilia Központ

🇭🇺

Budapest, Hungary

EUROMEDICA General Clinic of Thessaloniki; Gastroenterology Department

🇬🇷

Thessaloniki, Greece

ASST di Monza - Azienda Ospedaliera San Gerardo; U.O. Farmacia -Settore A - Corpo Posteriore

🇮🇹

Monza, Lombardia, Italy

Istituto Clinico Humanitas

🇮🇹

Rozzano (MI), Lombardia, Italy

Azienda Ospedaliera Di Padova

🇮🇹

Padova, Veneto, Italy

ICS ARENSIA Exploratory Medicine

🇲🇩

Chisinau, Moldova, Republic of

SPZOZ Uniwersytecki SK nr 1 im N. Barlickiego UM w Lodzi; Oddz. Klin. Gastroenter. Og. i Onk.

🇵🇱

?ód?, Poland

Szpital Uniwersytecki Nr 2 im. Dr Jana Biziela w Bydgoszczy; Centrum Endoskopii Zabiegowej

🇵🇱

Bydgoszcz, Poland

ETG Kielce

🇵🇱

Kielce, Poland

Economicus - NZOZ ALL-MEDICUS; Zaklad Gastroenterologii

🇵🇱

Katowice, Poland

Gastromed SPK Niepubliczny Zaklad Opieki Zdrowotnej

🇵🇱

Lublin, Poland

Clinical Research Center Sp. z o.o. MEDIC-R Spó?ka Komandytowa

🇵🇱

Pozna?, Poland

Endoskopia Sp. z o.o.

🇵🇱

Sopot, Poland

Centrum Zdrowia MDM

🇵🇱

Warszawa, Poland

Jaroslaw Kierkus Prywatna Prakyka Lekarska

🇵🇱

Warszawa, Poland

Przychodnia EuroMediCare

🇵🇱

Wroc?aw, Poland

Irkutsk Research Centre Hospital of Siberian department of Russian Academy of Science

🇷🇺

Irkutsk, Russian Federation

Saint Martyr Elizabeth City Hospital

🇷🇺

Sankt-peterburg, Sankt Petersburg, Russian Federation

Rostov State Medical University; Cardiorheumatology Department

🇷🇺

Rostov-na-Donu, Russian Federation

North-West State Medical University n.a. I.I. Mechnikov

🇷🇺

St. Petersburg, Russian Federation

KBC Dr Dragisa Misovic Dedinje

🇷🇸

Belgrade, Serbia

University Hospital Medical Center Bezanijska kosa

🇷🇸

Belgrade, Serbia

General Hospital Djordje Joanovic - Zrenjanin

🇷🇸

Zrenjanin, Serbia

Hospital de Gran Canaria Dr. Negrin; Servicio de Aparato Digestivo

🇪🇸

Las Palmas de Gran Canaria, LAS Palmas, Spain

Ternopil University Hospital; Regional Center of Gastroenterology with Hepatology

🇺🇦

Ternopil, Katerynoslav Governorate, Ukraine

Hospital Universitario de Torrejon

🇪🇸

Torrejon de Ardoz, Madrid, Spain

Regional Municipal Institution Chernivtsi Regional Clinical Hospital; Gastroenterology department

🇺🇦

Chernivtsi, Chernihiv Governorate, Ukraine

Medical Centre of PE First Private Clinic

🇺🇦

Zhytomir, Crimean Regional Governmenta, Ukraine

City Clinical Hospital #1; Department of Gastroenterology

🇺🇦

Vinnytsia, Kharkiv Governorate, Ukraine

ME Dnipropetrovsk Regional Clinical Hospital n.a. I.I Mechnykov Dnipropetrovsk Regional Council

🇺🇦

Dnipro, KIEV Governorate, Ukraine

Medical Center of LLC Medical Center Dopomoga Plus

🇺🇦

Kyiv, KIEV Governorate, Ukraine

Synexus Affiliate - MC of LLC Medbud-Clinic

🇺🇦

Kyiv, KIEV Governorate, Ukraine

Medical Center of LLC Diaservis

🇺🇦

Zaporizhzhia, KIEV Governorate, Ukraine

Clinic of SRI of Invalid Rehab. (ESTC) of VNMU n.a. M.I.Pyrohov

🇺🇦

Vinnytsia, Podolia Governorate, Ukraine

Medical Center of LLC Medical Center Family Medicine Clinic; Endoscopy & Gastroenterology

🇺🇦

Dnipr, Polissya Okruha, Ukraine

Transcarpathian Regional Clinical Hospital n.a. A. Novak; Rheumatology Department

🇺🇦

Uzhgorod, Ukraine

Kings College Hospital

🇬🇧

London, United Kingdom

Medical Center of Diaservice LLC; Division of clinical trials conduct, Department #3

🇺🇦

Zaporizhzhia, Ukraine

Medical Center of LLC Medical Clinic Blagomed

🇺🇦

Kyiv, KIEV Governorate, Ukraine

Med Center of International Institute of Clinical Trials LLC; Medical Center "OK!Clinic+"

🇺🇦

Kyiv, KIEV Governorate, Ukraine

Municipal Institution Zaporizhzhia Regional Clinical Hospital of Zaporizhzhia Regional Council

🇺🇦

Zaporizhzhia, Kharkiv Governorate, Ukraine

Treatment and Diagnostic Center of LLC MRT Elit

🇺🇦

Kropyvnytskyi, KIEV Governorate, Ukraine

Medical Center of Limited Liability Company ?Harmoniya krasy?

🇺🇦

Kyiv, KIEV Governorate, Ukraine

Medical Center of Edelweiss Medics LLC

🇺🇦

Kyiv, KIEV Governorate, Ukraine

© Copyright 2025. All Rights Reserved by MedPath