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Pharmacokinetic, Safety, Tolerability and Immunogenicity Study of SB4 in Healthy Male Subjects

Phase 1
Completed
Conditions
Healthy
Interventions
Biological: SB4
Biological: EU sourced Enbrel
Biological: US sourced Enbrel
Registration Number
NCT01865552
Lead Sponsor
Samsung Bioepis Co., Ltd.
Brief Summary

The purpose of this study is to compare the pharmacokinetics, safety and immunogenicity of SB4 and Enbrel (EU sourced Enbrel and US sourced Enbrel) in healthy male subjects.

Detailed Description

* Part A: Comparison between SB4 and EU sourced Enbrel

* Part B: Comparison between SB4 and US sourced Enbrel

* Part C: Comparison between EU sourced Enbrel and US sourced Enbrel

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
138
Inclusion Criteria
  • Healthy male subjects
  • Have a body weight between 60 and 94.9 kg and a body mass index between 20.0 and 29.9 kg/m², inclusive.
Exclusion Criteria
  • history and/or current presence of clinical significant atopic allergy, hypersensitivity or allergic reactions, also including known or suspected clinically relevant drug hypersensitivity to any components of the test and reference IP formulation or comparable drugs.
  • active or latent Tuberculosis or who have a history of TB.
  • history of invasive systemic fungal infections or other opportunistic infections
  • systemic or local infection, a known risk for developing sepsis and/or known active inflammatory process
  • serious infection associated with hospitalisation and/or which required intravenous antibiotics
  • history of and/or current cardiac disease
  • have received live vaccine(s) within 30 days prior to Screening or who will require live vaccine(s) between Screening and the final study visit.
  • Intake medication with a half-life > 24 h within 1 month or 10 half-lives of the medication prior to the first administration of IP.

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
US sourced Enbrel and SB4 in Part BSB4US sourced Enbrel followed by SB4
US and EU sourced Enbrel in Part CUS sourced EnbrelUS sourced Enbrel followed by EU sourced Enbrel
SB4 and US sourced Enbrel in Part BUS sourced EnbrelSB4 followed by US sourced Enbrel
EU and US sourced Enbrel in Part CEU sourced EnbrelEU sourced Enbrel followed by US sourced Enbrel
SB4 and EU sourced Enbrel in Part ASB4SB4 followed by EU sourced Enbrel
SB4 and EU sourced Enbrel in Part AEU sourced EnbrelSB4 followed by EU sourced Enbrel
EU sourced Enbrel and SB4 in Part ASB4EU sourced Enbrel followed by SB4
EU sourced Enbrel and SB4 in Part AEU sourced EnbrelEU sourced Enbrel followed by SB4
SB4 and US sourced Enbrel in Part BSB4SB4 followed by US sourced Enbrel
US sourced Enbrel and SB4 in Part BUS sourced EnbrelUS sourced Enbrel followed by SB4
EU and US sourced Enbrel in Part CUS sourced EnbrelEU sourced Enbrel followed by US sourced Enbrel
US and EU sourced Enbrel in Part CEU sourced EnbrelUS sourced Enbrel followed by EU sourced Enbrel
Primary Outcome Measures
NameTimeMethod
Area Under the Concentration-time Curve From Time Zero to Infinity (AUCinf)0 to 480 hours post-dose

pre-dose and at 6, 12, 24, 36, 48, 60, 72, 84, 96, 120, 144, 168, 216, 312 and 480 h post-dose

Maximum Serum Concentration (Cmax)0 to 480 hours post-dose

pre-dose (0 h) and at 6, 12, 24, 36, 48, 60, 72, 84, 96, 120, 144, 168, 216, 312 and 480 h post-dose.

Secondary Outcome Measures
NameTimeMethod
Area Under the Concentration-time Curve From Time Zero to the Last Quantifiable Concentration (AUClast)0 to 480 hours post-dose

pre-dose and at 6, 12, 24, 36, 48, 60, 72, 84, 96, 120, 144, 168, 216, 312 and 480 h post-dose

Time to Cmax (Tmax)0 to 480 hours post-dose

pre-dose and at 6, 12, 24, 36, 48, 60, 72, 84, 96, 120, 144, 168, 216, 312 and 480 h post-dose

Trial Locations

Locations (1)

Parexel International GmbH

🇩🇪

Berlin, Germany

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