MedPath

A Placebo-Controlled, Double-Blind Study to Confirm the Reversal of Hepatorenal Syndrome Type 1 With Terlipressin

Phase 3
Completed
Conditions
Hepatorenal Syndrome
Interventions
Drug: Placebo
Registration Number
NCT01143246
Lead Sponsor
Mallinckrodt
Brief Summary

This study is designed to evaluate the efficacy and safety of intravenous terlipressin versus placebo for the treatment of type 1 hepatorenal syndrome (HRS) in participants receiving standard of care albumin therapy.

Detailed Description

Hepatorenal syndrome is a rare syndrome of marked renal dysfunction in patients with cirrhosis, decompensated liver disease, and portal hypertension. Hepatorenal syndrome type 1 is characterized by a rapid progressive renal impairment and has a very poor prognosis with \> 80% mortality within 3 months. At present, there are no approved drug therapies for HRS type 1 in the US, Australia, or Canada. The only curative treatment for HRS type 1 and the underlying end-stage cirrhosis is liver transplantation. However, many patients will not survive long enough to receive a liver transplant and therapy, which may provide a bridge to transplantation, is badly needed. Increased understanding of the pathophysiology of HRS type 1 has demonstrated that vasoconstrictive drug therapy may reverse HRS type 1. Substantial data available from many published clinical investigations in the literature provide compelling evidence suggesting that administration of terlipressin improves renal function in patients with HRS.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
196
Inclusion Criteria
  1. Written informed consent by subject or legally authorized representative

  2. At least 18 years of age

  3. Cirrhosis and ascites

  4. Rapidly progressive reduction in renal function characterized by:

    • Serum creatinine (SCr) ≥ 2.5 mg/dL
    • Doubling of SCr within 2 weeks (or for observations of shorter duration, SCr values over time meeting slope-based criteria for proportional increases likely to be representative of at least a doubling within 2 weeks
  5. No sustained improvement in renal function (< 20% decrease in SCr and SCr ≥ 2.25 mg/dL) 48 hours after both diuretic withdrawal and the beginning of plasma volume expansion with albumin:

Note: Albumin doses recommended by the International Ascites Club (IAC) are 1 g/kg on the first day (Maximum 100 g) and 20 - 40 g/day thereafter as clinically indicated. It is recommended (if clinically appropriate) that the albumin dose is kept constant during the study drug administration period.

Note: The qualifying SCr value is the SCr value at least 48 hrs after both diuretic withdrawal (if applicable) and the beginning of albumin fluid challenge. The qualifying SCr value must be ≥ 2.25 mg/dL AND at least 80% of the diagnostic (pre-fluid challenge) SCr value.

Exclusion Criteria
  1. SCr > 7 mg/dL

  2. Shock Note: Hypotension (Mean Arterial Pressure < 70 mm Hg or a decrease > 40 mm Hg in systolic blood pressure from baseline) with evidence of hypoperfusion abnormalities despite adequate fluid resuscitation.

  3. Sepsis or systemic inflammatory response syndrome (SIRS)

    Note: SIRS: Presence of 2 or more of the following findings:

    Temperature > 38°C or < 36°C; heart rate > 90/min; respiratory rate of > 20/min or a PaCO2 of < 32 mm Hg; white blood cell count of > 12,000 cells/µL or < 4,000/ µL.

    Note: Sepsis: Documented infection and systemic inflammatory response syndrome.

  4. < 2 days anti-infective therapy for documented or suspected infection

  5. Proteinuria > 500 mg/day

  6. Hematuria or microhematuria (> 50 red blood cells per high power field)

  7. Clinically significant casts on urinalysis, including granular casts Note: Urine sediment examination is required to exclude presence of granular casts and other clinically significant casts [e.g., red blood cell (RBC) casts].

  8. Evidence of intrinsic or parenchymal renal disease (including acute tubular necrosis)

  9. Obstructive uropathy or other renal pathology on ultrasound or other medical imaging

  10. Current or recent treatment (within 4 weeks) with nephrotoxic drugs, e.g., aminoglycosides, nonsteroidal anti-inflammatory drugs (NSAID) Note: Up to 3 doses of an NSAID within the prior month (prescription or over the counter) is acceptable Note: Use of short-term (< 2 weeks) oral neomycin for acute encephalopathy is acceptable.

  11. Current or recent (within 4 weeks) renal replacement therapy

  12. Superimposed acute liver failure/injury due to factors other than alcoholic hepatitis, including acute viral hepatitis, drugs, medications (e.g., acetaminophen), or other toxins (e.g., mushroom [Amanita] poisoning)

  13. Current or recent treatment (within 48 hours) with octreotide, midodrine, vasopressin, dopamine or other vasopressors

  14. Severe cardiovascular disease as judged by investigator

  15. Estimated life expectancy of less than 3 days

  16. Confirmed pregnancy

  17. Known allergy or sensitivity to terlipressin or another component of the study treatment

  18. Participation in other clinical research studies involving the evaluation of other investigational drugs or devices within 30 days of randomization

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
PlaceboPlaceboParticipants receive matching placebo intravenously as a bolus injection, followed by a saline flush. Dose, duration, retreatment and/or discontinuation may be modified by the investigator, per protocol.
TerlipressinTerlipressinParticipants receive terlipressin intravenously as a bolus injection, followed by a saline flush. Dose, duration, retreatment and/or discontinuation may be modified by the investigator, per protocol.
Primary Outcome Measures
NameTimeMethod
Percentage of Participants With Confirmed Hepatorenal Syndrome (HRS) Reversalwithin 14 days

Confirmed HRS Reversal: The percentage of participants with two serum creatinine (SCr) values of ≤ 1.5 mg/dL at least 48 hours apart, on treatment, and without intervening renal replacement therapy or liver transplant.

Secondary Outcome Measures
NameTimeMethod
Percentage of Participants With Transplant-free SurvivalUp to 90 days

Transplant-Free Survival up to 90 days, defined as the time (in days) that each participant survives without liver transplantation from the day of randomization.

Percentage of Participants With HRS Reversalwithin 14 days

HRS reversal is defined as at least one SCr value of ≤ 1.5 mg/dL on treatment (up to 24 hours after the last dose of study medication).

Percentage of Participants With Serious Adverse EventsUp to 30 days post treatment (within 44 days)

Clinically significant changes in vital signs, height, weight, immunogenicity and laboratory assessments which qualified for the definition of serious adverse event are reported.

Percentage of Participants With Overall SurvivalUp to 90 days

Overall Survival up to 90 days, defined as the time (in days) that each participant survives from the day of randomization.

Trial Locations

Locations (73)

Scripps Clinic

🇺🇸

La Jolla, California, United States

University of Kentucky Chandler Medical Center

🇺🇸

Lexington, Kentucky, United States

Iowa City VA Health Care System

🇺🇸

Iowa City, Iowa, United States

New York Medical College/Westchester Medical Center

🇺🇸

Valhalla, New York, United States

UT Southwestern Medical Center

🇺🇸

Dallas, Texas, United States

Tulane Medical Center

🇺🇸

New Orleans, Louisiana, United States

University of Massachusetts Medical Center

🇺🇸

Worcester, Massachusetts, United States

NYU Langhorn Medical Center

🇺🇸

New York, New York, United States

Temple University Hospital

🇺🇸

Philadelphia, Pennsylvania, United States

Mount Sinai Medical Center

🇺🇸

New York, New York, United States

Carolinas Medical Center

🇺🇸

Charlotte, North Carolina, United States

SCTI Research Foundation

🇺🇸

Coronado, California, United States

University of Maryland

🇺🇸

Baltimore, Maryland, United States

Saint Louis University

🇺🇸

Saint Louis, Missouri, United States

Toronto General Hospital

🇨🇦

Toronto, Ontario, Canada

Columbia University Medical Center

🇺🇸

New York, New York, United States

Northwestern University

🇺🇸

Chicago, Illinois, United States

Beth Lsrael Deaconess Medical Center

🇺🇸

Boston, Massachusetts, United States

Cleveland Clinic

🇺🇸

Cleveland, Ohio, United States

Indiana University Health - University Hospital

🇺🇸

Indianapolis, Indiana, United States

Veteran's Administration Medical Center

🇺🇸

San Diego, California, United States

University of Cincinnati, Internal Medicine-Digestive Diseases

🇺🇸

Cincinnati, Ohio, United States

Washington University School of Medicine

🇺🇸

Saint Louis, Missouri, United States

California Pacific Medical Center

🇺🇸

San Francisco, California, United States

University of Minnesota

🇺🇸

Minneapolis, Minnesota, United States

Vanderbilt Medical Center

🇺🇸

Nashville, Tennessee, United States

The University of Texas Health Science Center at San Antonio

🇺🇸

San Antonio, Texas, United States

University of Texas Health Science Center

🇺🇸

San Antonio, Texas, United States

University of Utah

🇺🇸

Salt Lake City, Utah, United States

University of Arizona Medical Center South Campus

🇺🇸

Tucson, Arizona, United States

University of Arizona Liver Research Institute

🇺🇸

Tucson, Arizona, United States

Mayo Clinic

🇺🇸

Jacksonville, Florida, United States

Georgetown University Hospital

🇺🇸

Washington, District of Columbia, United States

CHUM, Hopital St-Luc

🇨🇦

Montreal, Quebec, Canada

University of Miami

🇺🇸

Miami, Florida, United States

Hartford Hospital

🇺🇸

Hartford, Connecticut, United States

University of Alabama at Birmingham

🇺🇸

Birmingham, Alabama, United States

Banner Good Samaritan Medical Center/Liver Disease Center

🇺🇸

Phoenix, Arizona, United States

Mayo Clinic Arizona

🇺🇸

Phoenix, Arizona, United States

University of Colorado Denver

🇺🇸

Aurora, Colorado, United States

Henry Ford Hospital

🇺🇸

Detroit, Michigan, United States

University of Nebraska Medical Center

🇺🇸

Omaha, Nebraska, United States

INTEGRIS Baptist Medical Center

🇺🇸

Oklahoma City, Oklahoma, United States

Orgeon Health & Science University

🇺🇸

Portland, Oregon, United States

Emory University Hospital

🇺🇸

Atlanta, Georgia, United States

VA Pittsburgh Healthcare System

🇺🇸

Pittsburgh, Pennsylvania, United States

Baylor University Medical Center

🇺🇸

Dallas, Texas, United States

The University of Texas Medical Branch at Galveston

🇺🇸

Galveston, Texas, United States

St. Luke's Advanced Liver Therapies

🇺🇸

Houston, Texas, United States

Baylor All Saints Medical Center

🇺🇸

Fort Worth, Texas, United States

The Methodist Hospital

🇺🇸

Houston, Texas, United States

Methodist Specialty Transplant Hospital Lab

🇺🇸

San Antonio, Texas, United States

Virginia Commonwealth University Health System

🇺🇸

Richmond, Virginia, United States

UC Davis Medical Center

🇺🇸

Sacramento, California, United States

University of Chicago

🇺🇸

Chicago, Illinois, United States

University of Wisconsin

🇺🇸

Madison, Wisconsin, United States

Virginia Mason Medical Center

🇺🇸

Seattle, Washington, United States

USC University Hospital

🇺🇸

Los Angeles, California, United States

Arrowhead Regional Medical Center

🇺🇸

Colton, California, United States

Loyola University Medical Center

🇺🇸

Maywood, Illinois, United States

Lahey Clinic Medical Center

🇺🇸

Burlington, Massachusetts, United States

Bellevue Hospital

🇺🇸

New York, New York, United States

Drexel University College of Medicine

🇺🇸

Philadelphia, Pennsylvania, United States

University of Pennsylvania

🇺🇸

Philadelphia, Pennsylvania, United States

Albert Einstein Medical Center

🇺🇸

Philadelphia, Pennsylvania, United States

WJB Dorn VA Medical Center

🇺🇸

Columbia, South Carolina, United States

Dallas VA Medical Center

🇺🇸

Dallas, Texas, United States

University of Texas Health Science Center at Houston - Memorial Hermann Hospital

🇺🇸

Houston, Texas, United States

McGuire DVAMC

🇺🇸

Richmond, Virginia, United States

Yale University School of Medicine

🇺🇸

New Haven, Connecticut, United States

University of Louisville

🇺🇸

Louisville, Kentucky, United States

Saint Luke's Hospital

🇺🇸

Kansas City, Missouri, United States

University of Kansas Medical Center

🇺🇸

Kansas City, Kansas, United States

© Copyright 2025. All Rights Reserved by MedPath