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Clinical Trials/NCT07259512
NCT07259512
Recruiting
Phase 4

Comparative Effects of Single Versus Twice-Daily Ramipril Dosing on Renal Function in Patients With Chronic Kidney Disease and Heart Failure With Reduced Ejection Fraction: Evaluation of Plasma Renin Activity, Malondialdehyde, Interleukin-6, Albuminuria, and Cystatin C

Evi Liliek Wulandari1 site in 1 country80 target enrollmentStarted: June 30, 2025Last updated:
InterventionsRamipril

Overview

Phase
Phase 4
Status
Recruiting
Sponsor
Evi Liliek Wulandari
Enrollment
80
Locations
1
Primary Endpoint
Change in Plasma Renin Activity (PRA)

Overview

Brief Summary

This study compares the effects of once-daily versus twice-daily ramipril dosing on renal function in chronic kidney disease (CKD) patients with heart failure with reduced ejection fraction (HFrEF). Outcomes include changes in plasma renin activity, malondialdehyde, interleukin-6, albuminuria, and cystatin C after 30 days of therapy.

Detailed Description

Chronic kidney disease (CKD) frequently coexists with heart failure with reduced ejection fraction (HFrEF), characterized by neurohormonal activation, inflammation, oxidative stress, and progressive renal deterioration. Activation of the renin-angiotensin-aldosterone system (RAAS) contributes significantly to both renal and cardiac dysfunction. Ramipril, an ACE inhibitor, is widely recommended for CKD with albuminuria and HFrEF. However, discrepancies exist in guidelines regarding once-daily versus twice-daily administration. These differences may influence RAAS suppression effectiveness and patient adherence.

This randomized, double-blind, parallel assignment clinical trial investigates the impact of once-daily (10 mg every 24 hours) versus twice-daily (5 mg every 12 hours) ramipril dosing on renal biomarkers in CKD patients with HFrEF. Outcomes include plasma renin activity (PRA), malondialdehyde (MDA), interleukin-6 (IL-6), albuminuria, and cystatin C measured over a 30-day treatment period. The study aims to provide scientific evidence to support optimal ramipril dosing strategies that improve renal outcomes among patients with CKD and reduced ejection fraction heart failure.

Study Design

Study Type
Interventional
Allocation
Randomized
Intervention Model
Parallel
Primary Purpose
Treatment
Masking
Triple (Participant, Care Provider, Outcomes Assessor)

Eligibility Criteria

Ages
18 Years to — (Adult, Older Adult)
Sex
All
Accepts Healthy Volunteers
No

Inclusion Criteria

  • Female or Male with age \>18 years old
  • Patients with a diagnosis of CKD stage 3-5 non-dialysis with low ejection fraction heart failure (ejection fraction \< 40%)

Exclusion Criteria

  • Receiving hemodialysis therapy
  • History of intolerance to ACE inhibitors
  • Refractory hyperkalemia
  • Pregnancy
  • History of angioedema to ACE inhibitors
  • Receiving sacubitril-valsartan therapy
  • Receiving ARB therapy
  • Hypotension with blood pressure \<90/60, or patients in shock.

Arms & Interventions

Once-Daily Ramipril

Experimental

Participants receive ramipril 10 mg once daily for 30 days

Intervention: Ramipril (Drug)

Twice-Daily Ramipril

Experimental

Participants receive ramipril 5 mg twice daily for 30 days

Intervention: Ramipril (Drug)

Outcomes

Primary Outcomes

Change in Plasma Renin Activity (PRA)

Time Frame: 30 days

Change in plasma renin activity from baseline to day 30.

Change in Malondialdehyde (MDA)

Time Frame: 30 days

Change in plasma MDA levels as a biomarker of oxidative stress

Change in Interleukin-6 (IL-6)

Time Frame: 30 days

Change in serum IL-6 levels as a marker of systemic inflammation

Change in Albuminuria

Time Frame: 30 days

Change in albumin-creatinine ratio (ACR) from baseline to day 30

Change in Cystatin C

Time Frame: 30 days

Change in serum cystatin C levels as a marker of glomerular filtration

Secondary Outcomes

  • Change in Serum Creatinine(30 days)
  • Change in Estimated Glomerular Filtration Rate (eGFR)(30 days)
  • Change in Blood Pressure (Systolic and Diastolic)(30 days)
  • Incidence of Treatment-Related Adverse Events(30 days)

Investigators

Sponsor
Evi Liliek Wulandari
Sponsor Class
Other
Responsible Party
Sponsor Investigator
Principal Investigator

Evi Liliek Wulandari

Principal Investigator, Consultant Internist (Internal Medicine Specialist)

Universitas Sebelas Maret

Study Sites (1)

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