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Safety and Efficacy Study of IFX-1 in add-on to Standard of Care in GPA and MPA

Phase 2
Terminated
Conditions
Granulomatosis With Polyangiitis (GPA)
Microscopic Polyangiitis (MPA)
Interventions
Registration Number
NCT03712345
Lead Sponsor
InflaRx GmbH
Brief Summary

The purpose of this study is to investigate the safety and tolerability of two dose regimens of IFX-1 as add-on to standard of care (SOC) in subjects with GPA and MPA compared with placebo.

Detailed Description

Granulomatosis with polyangiitis (GPA) and microscopic polyangiitis (MPA) are related systemic v anti-neutrophil cytoplasmic antibody (ANCA)-associated vasculitis (AAV), a potentially life-threatening disease.

GPA is a necrotizing vasculitis predominantly involving small- to medium-sized vessels (e.g., capillaries, venules, arterioles, arteries, and veins). MPA is a necrotizing vasculitis that primarily affects capillaries, venules, or arterioles, most commonly manifesting as necrotizing glomerulonephritis and/or pulmonary capillaritis. MPA.

Primed neutrophils are activated by ANCA and generate C5a that engages C5a receptors on neutrophils. Therefore, patients with ANCA-related disease have elevated plasma and urine levels of C5a in active disease and not in remission.

IFX-1 is a monoclonal antibody specifically binding to the soluble human complement split product C5a and the resulting nearly complete blockade of C5a-induced biological effects may be effective in the treatment of subjects with AAV.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
20
Inclusion Criteria
  1. Male or female, ≥18 years of age.
  2. Diagnosis of GPA or MPA according to the definitions of the Chapel Hill Consensus Conference.
  3. Have at least one "major" item, or at least three other items, or at least two renal items on the Birmingham Vasculitis Activity Score (BVAS) Version 3.0.
  4. New or relapsed GPA or MPA that require treatment with CYC or RTX plus GCs.
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Exclusion Criteria
  1. Any other multisystem autoimmune disease
  2. Requires mechanical ventilation because of alveolar hemorrhage at Screening.
  3. Human immunodeficiency virus, hepatitis B, or hepatitis C viral screening test showing evidence of active or chronic viral infection at Screening or a documented history of the human immunodeficiency virus, hepatitis B, or hepatitis C.
  4. Received CYC or RTX 12 weeks before Screening; if on azathioprine (AZA), methotrexate (MTX), mycophenolate mofetil (MMF), or mycophenolate sodium (MPS) at the time of Screening, these drugs must be withdrawn prior to receiving CYC or RTX.
  5. Received more than 3 g cumulative high dose intravenous GCs within 4 weeks before Screening.
  6. On an oral dose of a GC of more than 10 mg prednisone equivalent at Screening or for more than 6 weeks before Screening.
  7. Received a CD20 inhibitor, anti-tumor necrosis factor treatment, abatacept, alemtuzumab, any other experimental or biological therapy, intravenous immunoglobulin or plasma exchange, antithymocyte globulin, or required dialysis within 12 weeks before Screening.
  8. Received a live vaccination within 4 weeks before Screening or planned between Screening and Week 24.
  9. Female subjects of childbearing potential unwilling or unable to use a highly effective method of contraception (pearl index <1%) such as complete sexual abstinence, combined oral contraceptive, vaginal hormone ring, transdermal contraceptive patch, contraceptive implant, or depot contraceptive injection in combination with a second method of contraception such as condom, cervical cap, or diaphragm with spermicide during the study and for at least 4 weeks after last administration of IFX-1 (timeframes for SOC have to be considered as described in the respective Prescribing Information).
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Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
IFX-1 high doseIFX-1 high doseWill receive IFX-1 high dose regimen diluted in sodium chloride solution
PlaceboPlaceboWill receive placebo
IFX-1 low doseIFX-1 low doseWill receive IFX-1 low dose regimen diluted in sodium chloride solution
Primary Outcome Measures
NameTimeMethod
Number and Percentage of Participants With at Least One TEAE Per Treatment Group.Week 24

Number and percentage of participants who experience at least one treatment-emergent adverse event (TEAE) per treatment group.

Secondary Outcome Measures
NameTimeMethod
Percentage of Participants Achieving Clinical ResponseWeek 16

Efficacy Endpoint based on clinical response evaluated through BVAS. Clinical response is defined as a reduction in BVAS of ≥50% and no worsening in any body system and no administration of rescue medication prior to the response assessment.

Percentage of Participants With Clinical Remission (BVAS = 0)Week 16

Efficacy Endpoint that evaluates participants with complete remission

IFX-1 Concentration Pre-doseWeek 16

Assess the pharmacokinetic of the investigational medicinal product.

IFX 1 Concentration at Predose (0 Hours), After the End of the Infusion (+10minutes), and at 2, 6, 24, and 48 Hours After the Start of the Infusion for Participants in the PK SubstudyWeeks 1, 4 and 16

Analyze the IMP plasma concentration using a PK model: IFX 1 concentration at predose (0 hours), after the end of the infusion (+10minutes), and at 2, 6, 24, and 48 hours after the start of the infusion for participants in the PK substudy

C5a Plasma ConcentrationWeek 16

Pharmacodynamic parameter concentration

IFX-1 Blocking Activity 2.5 nMWeek 16

Pharmacodynamic Parameter of IFX-1 blocking activity 2.5 nM

IFX-1 Blocking Activity 10 nMWeek 16

Pharmacodynamic Parameter of IFX-1 blocking activity 10 nM

Trial Locations

Locations (38)

Texas Health Resources

🇺🇸

Dallas, Texas, United States

Rush University Medical Center

🇺🇸

Chicago, Illinois, United States

Massachusetts General Hospital

🇺🇸

Boston, Massachusetts, United States

University of New Mexico

🇺🇸

Albuquerque, New Mexico, United States

University of Miami

🇺🇸

Miami, Florida, United States

Johns Hopkins Bayview Medical Center

🇺🇸

Baltimore, Maryland, United States

LSU Health Sciences Center Shreveport

🇺🇸

Shreveport, Louisiana, United States

Ohio State University Clinical Trials Management Office

🇺🇸

Columbus, Ohio, United States

Washington University

🇺🇸

Saint Louis, Missouri, United States

Altoona Center for Clinical Research, P.C.

🇺🇸

Duncansville, Pennsylvania, United States

BRCR Medical Center, Inc.

🇺🇸

Camp Hill, Pennsylvania, United States

CHUM Centre de Recherche

🇨🇦

Québec, Quebec, Canada

University of Alberta Hospital

🇨🇦

Edmonton, Alberta, Canada

Centre de Recherche Musculo-Squelettique

🇨🇦

Trois-Rivières, Quebec, Canada

Low Country Rheumatology, PA

🇺🇸

North Charleston, South Carolina, United States

Mount Sinai Hospital

🇨🇦

Toronto, Ontario, Canada

Texas Research Institute

🇺🇸

Fort Worth, Texas, United States

UVA University Physicians Charlottesville

🇺🇸

Charlottesville, Virginia, United States

St. Josephs Healthcare

🇨🇦

Hamilton, Ontaria, Canada

University of Minnesota

🇺🇸

Minneapolis, Minnesota, United States

University of Kansas Medical Center Research Institute, Inc.

🇺🇸

Kansas City, Kansas, United States

Science Connections, LLC

🇺🇸

Doral, Florida, United States

Mayo Clinic Scottsdale

🇺🇸

Scottsdale, Arizona, United States

Northwell Health, LLC PRIME

🇺🇸

New Hyde Park, New York, United States

Hospital for Special Surgery

🇺🇸

New York, New York, United States

Trinity Medical Group

🇺🇸

Minot, North Dakota, United States

University of Pennsylvania

🇺🇸

Philadelphia, Pennsylvania, United States

Pioneer Research Solutions, Inc.

🇺🇸

Houston, Texas, United States

West Virginia University

🇺🇸

Morgantown, West Virginia, United States

Loma Linda University Clinical Trial Center

🇺🇸

Loma Linda, California, United States

University of Rochester Medical Center - Strong Memorial Hospital

🇺🇸

Rochester, New York, United States

Adriana Pop Moody Clinic PA

🇺🇸

Corpus Christi, Texas, United States

University Of MI Medcl Ctr-RHU

🇺🇸

Ann Arbor, Michigan, United States

Henry Ford Hospital

🇺🇸

Detroit, Michigan, United States

Mayo Clinic

🇺🇸

Rochester, Minnesota, United States

Oregon Health & Science University

🇺🇸

Portland, Oregon, United States

UNC Kidney Center, UNC-CH Division of Nephrology and Hypertension

🇺🇸

Chapel Hill, North Carolina, United States

Rhode Island Hospital

🇺🇸

Providence, Rhode Island, United States

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