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A Study to Evaluate the Mass Balance of 14C-Napabucasin in Healthy Adult Male Subjects

Phase 1
Completed
Conditions
ADME
Healthy
Interventions
Registration Number
NCT03525405
Lead Sponsor
Sumitomo Pharma America, Inc.
Brief Summary

This is a Phase I, single-center, open-label, single-sequence, study evaluating the absorption, metabolism, and excretion of napabucasin in healthy adult male volunteers using a mixture 14C-radiolabeled and unlabeled material.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
8
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Single Dosenapabucasin-
Primary Outcome Measures
NameTimeMethod
Pharmacokinetics for napabucasin and metabolites by assessing urinary concentrationUp to 12 days
Pharmacokinetics for napabucasin and metabolites by assessing plasma concentration1 week
Pharmacokinetics for napabucasin and metabolites by assessing fecal concentrationUp to 12 days
Secondary Outcome Measures
NameTimeMethod
Number of Patients with Adverse Events4 weeks

Trial Locations

Locations (1)

Covance Clinical Research Unit

🇺🇸

Madison, Wisconsin, United States

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