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Relatlimab With Nivolumab and 5-Azacytidine for the Treatment of AML

Phase 2
Recruiting
Conditions
Acute Myeloid Leukemia
Interventions
Registration Number
NCT04913922
Lead Sponsor
Ludwig-Maximilians - University of Munich
Brief Summary

The clinical trial will test the safety and tolerability of a combination therapy (azacitidine in combination with two checkpoint inhibitors, nivolumab \[Anti-PD1\] and relatlimab \[Anti-LAG3\]) in patients with relapsed/refractory Acute Myeloid Leukemia (AML) and patients ≥ 65 years with initial diagnosis of AML.

Primary objectives are:

* maximum tolerated dose (MTD) and dose-limiting toxicities (DLT) of the combination therapy during the lead-in phase of the clinical trial (6-12 patients) and

* objective response rate (ORR) of the combination therapy in the phase II part of the study (up to 24 patients).

Detailed Description

Not available

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
30
Inclusion Criteria

Cohort 1 (R/R AML):

  • Patients with AML who have failed first line induction chemotherapy (consisting of a minimum of two intensive chemotherapy cycles, e.g. 7+3 or HAM) or patients with AML who have relapsed after achieving complete remission (CR), CRi, or CRp, or patients who have failed up to one prior salvage therapy

Cohort 2 (frontline older AML):

  • Patients aged ≥65 years with previously untreated AML who are unfit for or decline standard induction therapy.

General inclusion criteria:

  • Patients not eligible for intensive induction chemotherapy and/or allogeneic stem cell transplant.
  • Age ≥18 years
  • ECOG Performance Status ≤2
  • Adequate organ function:

Total bilirubin ≤2 x ULN (≤3 × ULN if due to leukemic involvement or Gilbert's syndrome) AST and ALT ≤2.5 × ULN (≤5.0 × ULN if due to leukemic involvement) Serum creatinine ≤2 × ULN or glomerular filtration rate (GFR) ≥50 mL/h

  • Adequate cardiac function: TTE with documented LVEF ≥50%
  • At least 2 weeks OR at least 5 half-lives interval from prior treatment to time of initiation of study medication
  • GvHD of grade ≤A on ≤10 mg prednisone without any additional immunosuppressive therapies (tacrolimus, ciclosporin, etc.)
  • Written informed consent
  • Negative pregnancy test and adequate methods of contraception for females of childbearing potential, adequate methods of contraception for males
Exclusion Criteria
  • Acute promyelocytic leukemia (APL)
  • Biphenotypic or bilineage leukemia
  • Known allergy or hypersensitivity to 5-azacytidine, nivolumab, relatlimab, or any of their components
  • History of life-threatening toxicity related to prior immune therapy
  • Previous treatment with immunotherapeutic drugs targeting PD-1/PD-L1 in combination with 5-azacytidine
  • Previous treatment with LAG-3 targeted agents
  • Known history of severe interstitial lung disease or severe pneumonitis
  • Known history (active, known, or suspected) of any of the following autoimmune diseases:

inflammatory bowel disease rheumatoid arthritis systemic progressive sclerosis systemic lupus erythematosus autoimmune vasculitis

  • Active uncontrolled pneumonitis
  • Active uncontrolled infection
  • Symptomatic or poorly controlled CNS leukemia
  • Confirmed history of encephalitis, meningitis, or uncontrolled seizures in the year prior to informed consent
  • Uncontrolled or significant cardiovascular disease
  • Troponin T (TnT) or I (TnI) > 2 × institutional ULN
  • Organ allografts
  • Allogeneic hematopoietic stem cell transplantation within the last 100 days before first study drug administration
  • Active GvHD > grade A
  • Known human immunodeficiency virus seropositivity
  • Known positivity for hepatitis B by surface antigen expression or active hepatitis C infection
  • Other medical, psychological, or social condition that may interfere with study participation or compliance, or compromise patient safety
  • Patients unwilling or unable to comply with the protocol
  • Patients who are pregnant or breastfeeding
  • Prisoners and subjects who are compulsory detained

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Combination therapyAzacitidine Injection5-azacitidine 75 mg/m2 body surface area s.c. for 7 days nivolumab 480mg i.v. day 1 relatlimab 80-160mg i.v. day 1 repeat day 28
Combination therapyNivolumab5-azacitidine 75 mg/m2 body surface area s.c. for 7 days nivolumab 480mg i.v. day 1 relatlimab 80-160mg i.v. day 1 repeat day 28
Combination therapyRelatlimab5-azacitidine 75 mg/m2 body surface area s.c. for 7 days nivolumab 480mg i.v. day 1 relatlimab 80-160mg i.v. day 1 repeat day 28
Primary Outcome Measures
NameTimeMethod
Objective response rate (ORR)During Phase II expansion phase, after completion of lead-in phase, approximately during months 7-48 of study conduct

To estimate the ORR to treatment with relatlimab + nivolumab + 5-azacytidine in patients with R/R AML and Patients ≥65 years with initial diagnosis of AML

Maximum tolerated dose (MTD)after completion of the first cycle in the fist 6-12 patients, approximately during the first 6-12 months of study conduct

To determine the MTD of relatlimab in combination with nivolumab and 5-azacytidine in patients with R/R AML.

Dose-limiting toxicities (DLTs)after completion of the first cycle in the fist 6-12 patients, approximately during the first 6-12 months of study conduct

To determine the DLT of relatlimab in combination with nivolumab and 5-azacytidine in patients with R/R AML.

Secondary Outcome Measures
NameTimeMethod
Blast reductionDuring Phase II expansion phase, after completion of lead-in phase, approximately during months 7-48 of study conduct

To determine the number of patients with R/R AML or Patients ≥65 years with initial diagnosis of AML treated with relatlimab + nivolumab + 5-azacytidine who have a blast reduction (defined as ≥50% reduction in blast percentage compared to baseline blast percentage in bone marrow)

Duration of response (DOR)During Phase II expansion phase, after completion of lead-in phase, approximately during months 7-48 of study conduct

To assess the duration of response (DOR) of patients with R/R AML or Patients ≥65 years with initial diagnosis of AML treated with relatlimab + nivolumab + 5-azacytidine.

Overall survival (OS)During Phase II expansion phase, after completion of lead-in phase, approximately during months 7-48 of study conduct

To assess the overall survival (OS) of patients with R/R AML or Patients ≥65 years with initial diagnosis of AML treated with relatlimab + nivolumab + 5-azacytidine.

Hematologic improvementDuring Phase II expansion phase, after completion of lead-in phase, approximately during months 7-48 of study conduct

To determine the number of patients with R/R AML or Patients ≥65 years with initial diagnosis of AML treated with relatlimab + nivolumab + 5-azacytidine who have a hematologic improvement (HI) in platelets, hemoglobin, or absolute neutrophil count (ANC)

Disease-free survival (DFS)During Phase II expansion phase, after completion of lead-in phase, approximately during months 7-48 of study conduct

To assess the disease-free survival (DFS) of patients with R/R AML or Patients ≥65 years with initial diagnosis of AML treated with relatlimab + nivolumab + 5-azacytidine.

Trial Locations

Locations (1)

University Hospital, LMU Munich

🇩🇪

Munich, Germany

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