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Radiolabel Study In Healthy Volunteers For Insomnia-Targeting Drug

Phase 1
Completed
Conditions
Sleep Initiation and Maintenance Disorders
Interventions
Drug: 14C-SB649868
Registration Number
NCT00520663
Lead Sponsor
GlaxoSmithKline
Brief Summary

The purpose of this study is to define the absorption, breakdown and excretion of a single dose of radiolabelled SB-649868 and its breakdown products by measuring their concentration in blood, urine and faeces over a 7-10 day period. "Radiolabelled" means that the test drug has a radioactive component to help us track the drug. The safety and tolerability of the test drug will also be assessed.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
8
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Healthy male subjects14C-SB649868Each subject will receive a single oral dose of 14C-SB649868 (containing approximately 70 microcuries of radiocarbon and 30 milligrams of SB649868).
Primary Outcome Measures
NameTimeMethod
Plasma levels of SB-649868 by measuring drug levels and radioactivity in plasma. Plasma, urine,faeces samples to study the metabolites of SB649868.over 4 days
Excretion of SB649868 by measuring radioactivity in urine and faecesover 7-10 days.
Secondary Outcome Measures
NameTimeMethod
Safety and tolerability of 14C-SB649868 by adverse event monitoring, lab samples and cardiovascular monitoring.over the course of the study

Trial Locations

Locations (1)

GSK Investigational Site

🇬🇧

Tranent, West Lothian, United Kingdom

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