MedPath

Ferumoxytol-enhanced Imaging and Mapping in neuroAIDS

Phase 2
Completed
Conditions
AIDS Dementia Complex
Interventions
Registration Number
NCT02678767
Lead Sponsor
Beau Nakamoto
Brief Summary

This project will investigate the ability of a novel MRI contrast agent to identify and quantitate ongoing monocyte/macrophage (M/MΦ)-mediated inflammation in the brains of HIV-infected individuals.

Detailed Description

HIV-associated neurocognitive disorders (HAND) continue to be prevalent despite effective combination antiretroviral therapy (cART) and have a significant impact on morbidity and quality of life. Monocytes/macrophages (M/MΦ) are believed to play a critical role in the pathogenesis of HAND. Neuroimaging HIV research has not focused on assessing M/MΦ-mediated inflammation in the brain. Currently, no neuroimaging modality exists that can define the extent of active inflammation due to M/MΦ in HAND either as a clinical diagnostic tool or to assist in defining objective improvement in clinical trials addressing HAND. Ferumoxytol is an ultra-small iron oxide MRI contrast agent avidly taken up by circulating M/MΦ. The investigators hypothesize that ferumoxytol-based imaging can identify ongoing inflammation due to perivascular M/MΦ which is believed to represent a key pathologic correlate of HAND.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
30
Inclusion Criteria
  • Age 40-65 years
  • Plasma HIV RNA < 48 copies/ml (HIV+ subjects only)
  • On stable cART >= 1 year (HIV+ subjects only)
  • Global neuropsychological (NP) score <-0.5 in at least one cognitive domain known to be affected by HIV (neurocognitively impaired subjects only)
  • Documentation of negative HIV infection by an FDA approved test (HIV- subjects only)
Exclusion Criteria
  • Active substance use
  • History of myocardial infarct or stroke
  • Diabetes
  • Chronic hepatitis C virus (HCV) infection
  • Uncontrolled major affective disorder, active psychosis, central nervous system disease that affects the brain structure, or other uncontrolled chronic medical condition that in the opinion of the investigator may impact NP testing or the study outcome
  • Psychoactive or other medications which may impact NP testing
  • Factors that preclude MRI
  • Known hypersensitivity to ferumoxytol
  • History of laboratory measurements consistent with an iron overload syndrome
  • Medical conditions that require frequent blood transfusions
  • Taking oral iron supplements
  • Elevated iron levels
  • Any condition, which in the opinion of the investigator, would compromise the subject's ability to participate
  • Multiple drug allergies that may pose a greater risk of anaphylaxis associated with ferumoxytol
  • Pregnant, unwillingness to practice birth control, or breastfeeding
  • Unable to give informed consent

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
HIV+ with neurocognitive disorderFerumoxytolAll subjects will receive neurocognitive testing. Subjects will have a brain MRI prior to drug infusion. A one-time ferumoxytol IV infusion will be given at a dose of 4mg Fe/kg up to a maximum of 510mg of elemental iron delivered at a rate of 1ml/sec. A second brain MRI will be completed post-infusion
HIV- without neurocognitive impairmentFerumoxytolAll subjects will receive neurocognitive testing. Subjects will have a brain MRI prior to drug infusion. A one-time ferumoxytol IV infusion will be given at a dose of 4mg Fe/kg up to a maximum of 510mg of elemental iron delivered at a rate of 1ml/sec. A second brain MRI will be completed post-infusion
HIV+ without neurocognitive impairmentFerumoxytolAll subjects will receive neurocognitive testing. Subjects will have a brain MRI prior to drug infusion. A one-time ferumoxytol IV infusion will be given at a dose of 4mg Fe/kg up to a maximum of 510mg of elemental iron delivered at a rate of 1ml/sec. A second brain MRI will be completed post-infusion
Primary Outcome Measures
NameTimeMethod
Change in the proportion of abnormal MRIsChange from Baseline MRI at 4-6 weeks post-infusion MRI

The proportion of abnormal MRIs will be compared for each group.

Secondary Outcome Measures
NameTimeMethod
Change in quantitative susceptibility mapping (QSM)Change from Baseline MRI at 4-6 weeks post-infusion MRI

Use of QSM to quantitate ferumoxytol accumulation in the brain

Trial Locations

Locations (1)

Hawaii Center for AIDS

🇺🇸

Honolulu, Hawaii, United States

© Copyright 2025. All Rights Reserved by MedPath