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A Phase III Superiority Study of Vernakalant vs Amiodarone in Subjects With Recent Onset Atrial Fibrillation

Phase 3
Completed
Conditions
Atrial Fibrillation
Interventions
Registration Number
NCT00668759
Lead Sponsor
Advanz Pharma
Brief Summary

The primary objective of the study is to demonstrate the superiority of vernakalant injection over amiodarone injection in the conversion of atrial fibrillation (AF) to sinus rhythm (SR) within 90 minutes of the start of drug administration. The secondary objective is to compare the safety of vernakalant to amiodarone.

Detailed Description

This is a double-blind, active-controlled, double-dummy, multi-center, randomized trial in subjects with symptomatic AF of 3 to 48 hours duration.

Subjects will be randomized to receive vernakalant injection or amiodarone injection in a 1:1 ratio.

Safety will be assessed through the monitoring of adverse events, vital signs, continuous telemetry monitoring, 12-lead Holter monitoring, 12-lead ECGs, and laboratory tests.

At 2 hours after the start of infusion, electrical cardioversion may be performed or rate control medication may be administered. Class I and Class III antiarrhythmics are not to be administered for 24 hours after the start of infusion.

Subjects are to remain in the clinic for at least 6 hours after the start of infusion. Subjects will attend a follow-up visit at 7 (±2) days after treatment and will receive a follow-up telephone call at 30 (±3) days for assessment of serious adverse events, concomitant medications related to serious adverse events, and recurrence of AF.

All roles were blinded with the exception of each site's designated unblinded personnel who were responsible for randomization and preparation, dispensation and accountability of the study medication.

Expanded Access was not available through this protocol.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
254
Inclusion Criteria
  • Have symptomatic AF of 3 to 48 hours duration at baseline.
  • Be eligible for cardioversion.
  • Have adequate anticoagulation therapy for cardioversion in accordance with standard of practice as recommended by ACC/AHA/ESC guidelines [1].
  • Be hemodynamically stable and have systolic blood pressure (BP) above 100 mmHg and less than 160 mmHg and diastolic BP less than 95 mmHg at screening and baseline.

Key

Exclusion Criteria
  • Known or suspected prolonged QT or uncorrected QT interval of >440 msec as measured at screening on a 12 lead ECG, familial long QT syndrome, or previous torsades de pointes, ventricular fibrillation; or sustained ventricular tachycardia (VT).
  • Symptomatic bradycardia, sick sinus syndrome, or ventricular rate less than 50 beats per minute (bpm) as documented by 12-lead ECG at screening.
  • A QRS interval >140 msec.
  • Atrial flutter.
  • Significant valvular stenosis, hypertrophic obstructive cardiomyopathy, restrictive cardiomyopathy or constrictive pericarditis.
  • Documented previous episodes of second or third degree atrioventricular (AV) block.
  • Had a myocardial infarction (MI), acute coronary syndrome or cardiac surgery within 30 days prior to entry into the study.
  • Uncorrected electrolyte imbalance of serum potassium or magnesium. Both K+ and Mg2+ must be corrected prior to dosing.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
1Vernakalant InjectionVernakalant Injection: In one infusion line, subjects will receive a 10-minute infusion of vernakalant followed by a 15-minute observation period, followed by an additional 10-minute infusion of vernakalant if required (if the subject is still in AF). To maintain blinding, a 60-minute infusion of placebo (D5W) will be administered in a second infusion line, followed by a maintenance infusion of placebo for a minimum of an additional 60 minutes.
Primary Outcome Measures
NameTimeMethod
Proportion of subjects with conversion of atrial fibrillation to sinus rhythm within 90 minutes after the start of infusion.Conversion of AF to SR for a minimum duration of one minute within 90 minutes after start of infusion.
Secondary Outcome Measures
NameTimeMethod
Time to conversion within 90 minutes after the start of infusion.Time to conversion of AF to SR within 90 minutes after start of infusion.
Proportion of subjects with symptom relief at 90 minutes after the start of infusion.Relief of AF symptoms 90 minutes after start of infusion.
EQ-5D quality of life assessment.Assessment of quality of life 2 hours after start of infusion.
Monitoring of adverse events, vital signs, continuous telemetry monitoring, 12-lead Holter monitoring, 12-lead ECGs, and laboratory tests.Specified safety assessments completed at specified time points throughout the study from Screening to Discharge, at the Day 7 visit, and at the Day 30 follow-up call.

Trial Locations

Locations (100)

Royal Perth Hospital Emergency Research

🇦🇺

Perth, Western Australia, Australia

Gentofte Amtssygehus Kardiologisk afdeling

🇩🇰

Hellerup, Denmark

Herlev Amtssygehus, Kardiologisk

🇩🇰

Herlev, Denmark

Sygehus Vendsyssel Hjorring

🇩🇰

Hjorring, Denmark

Roskilde Amts Sygehus Køge

🇩🇰

Koge, Denmark

Regionshospitalet Silkeborg

🇩🇰

Silkeborg, Denmark

Nemocnice v Semilech Interní oddělení

🇨🇿

Semily, Czech Republic

Uherskohradistska nemocnice

🇨🇿

Uherské Hradiste, Czech Republic

VFN - III. Interni Klinika

🇨🇿

Praha, Czech Republic

Viimsi Hospital, Heart Clinic

🇪🇪

Haabneeme, Estonia

Ustredni vojenska nemocnice Koronarni jednotka

🇨🇿

Praha, Czech Republic

Oblastni nemocnice Pribram Interni Oddeleni

🇨🇿

Pribram, Czech Republic

Oulu University Hospital - Dept of Internal Medicine

🇫🇮

Oulu, Finland

Hôpital Lariboisiere

🇫🇷

Paris, France

Universitätsklinikum Bonn, Med. Klinik und Poliklinik II

🇩🇪

Bonn, Germany

Medizinische Klinik, Klinikum Hannover Nordstadt

🇩🇪

Hannover, Germany

Charite Campus Mitte, Med. Klinik und Poliklinik mit Schwerpunkt Kardiologie und Angiologie

🇩🇪

Berlin, Germany

CHU de Strasbourg - Hopital Hautepierre - Service de Cardiologie

🇫🇷

Strasbourg, France

Universitatsklinikum Gottingen, Herzzentrum

🇩🇪

Gottingen, Germany

Universitetssjukhuset MAS

🇸🇪

Malmo, Sweden

Kingston General Hospital

🇨🇦

Kingston, Ontario, Canada

Herzzentrum Brandenburg in Bernau Innere Medizin

🇩🇪

Bernau, Germany

Klinik Hamburg Bambek Kardiologie

🇩🇪

Hamburg, Germany

Ambulantes Herzzentrum Kassel Innere Medizin

🇩🇪

Kassel, Germany

Klaipeda Seamen's Hospital

🇱🇹

Klaipeda, Lithuania

WCN - Bethesda ziekenhuis

🇳🇱

Hoogeveen, Netherlands

Specjalistyczny Szpital Miejski im. Mikołaja Kopernika

🇵🇱

Toruń, Poland

Launceston General Hospital Cardiac Research Unit

🇦🇺

Launceston, Tasmania, Australia

Royal Hobart Hospital Cardiology Research

🇦🇺

Hobart, Tasmania, Australia

The Ottawa Hospital

🇨🇦

Ottawa, Ontario, Canada

Hopital de la Cite-de-la-Sante

🇨🇦

Laval, Quebec, Canada

Institut de Cardiologie de Montreal

🇨🇦

Montreal, Quebec, Canada

Centre Hopitalier de L'Universite de Montreal - Hotel Dieu

🇨🇦

Montreal, Quebec, Canada

McGill University Health Center The Montreal General Hospital

🇨🇦

Montreal, Quebec, Canada

Centre de santé et de services sociaux du Sud de Lanaudière - Hôpital Pierre-Le Gardeur

🇨🇦

Terrebonne, Quebec, Canada

Mestrska nemocnice Caslav

🇨🇿

Caslav, Czech Republic

Nemocnice Kroměříž

🇨🇿

Kroměříž, Czech Republic

CHU de Nancy - Hopital Brabois - Service de Cardiologie

🇫🇷

Nancy, France

Nemocnice Kutna Hora s.r.o. Interni Oddeleni

🇨🇿

Kutna Hora, Czech Republic

Nemocnice Decin Internal Medicine

🇨🇿

Nove Město, Czech Republic

Fakultní nemocnice v Motole, KAR

🇨🇿

Praha, Czech Republic

Nemocnice Tabor

🇨🇿

Tabor, Czech Republic

Tartu University Hospital Heart Clinic

🇪🇪

Tartu, Estonia

Nemocnice Slaný Interní oddělení

🇨🇿

Slaný, Czech Republic

Hopital Trousseau - Service de Cardiologie

🇫🇷

Chambray-les-Tours, France

Latvian Center of Cardiology, P. Stradins Clinical University Hospital

🇱🇻

Riga, Latvia

Academisch Ziekenhuis Maastricht

🇳🇱

Maastricht, Netherlands

Catharina Ziekenhuis Eindhoven

🇳🇱

Eindhoven, Netherlands

WCN - St. Franciscus Gasthuis

🇳🇱

Rotterdam, Netherlands

WCN - Canisius-Wilhelmina Ziekenhuis

🇳🇱

Nijmegen, Netherlands

Oddzial Kardiologiczny Wielospecjalityczny Szpital Miejski im.

🇵🇱

Bydgoszcz, Poland

Universityetssjukhuset, Orebro

🇸🇪

Orebro, Sweden

Szpital Miejski im. J. Brudzinskiego Oddzial Kardiologii

🇵🇱

Gdynia, Poland

Oddział Internistyczno-Kardiologiczny Samodzielny Publiczny Szpital Wojewódzki im. Jana Bożego w Lublinie

🇵🇱

Lublin, Poland

Oddzial Kardiologii Inwazyjnej Szpital Specjalistyczny im. E.Szczeklika w Tarnowie

🇵🇱

Tarnow, Poland

Oddział Kardiologiczno-Internistyczny Specjalistyczny Szpital Miejski im. Mikołaja Kopernika

🇵🇱

Toruń, Poland

III Klinika Chorob Wewnetrznych i Kardiologii

🇵🇱

Warszawa, Poland

Wojskowy Instytut Medyczny, CSK MON

🇵🇱

Warszawa, Poland

Osrodek Chorob Serca, Klinika Kardiologii, 4 Wojskowy Szpital Kliniczny z Poliklinika Samodzielny

🇵🇱

Wroclaw, Poland

Klinika Kardiologii Zachowawczej Centralny Szpital Kliniczny Ministerstwa Spraw Wewnętrznych i Administracji w Warszawie

🇵🇱

Warszawa, Poland

Institute of Treatment and Reahabilitation 'Niska Banja'

🇷🇸

Niska Banja, Serbia

Clinical Center Zemun, Dept. of Cardiology

🇷🇸

Zemun, Serbia

Interna klinika FN Trnava, Fakultna nemocnica Trnava

🇸🇰

Trnava, Slovakia

Middle Slovak Institute of Cardiovascular Diseases (SUSCCH)

🇸🇰

Banska Bysterica, Slovakia

Slovensky ustav srdcovych a cevnych chorob

🇸🇰

Bratislava, Slovakia

ICU, Hospital Lipt. Mikulas

🇸🇰

Liptovsky Mikulas, Slovakia

NsP Prievidza so sidlom v Bojniciah

🇸🇰

Bojnice, Slovakia

City Clinical Hospital #1 Intensive Care Unit

🇺🇦

Kiev, Ukraine

Akademiska Sjukhuset, Uppsala

🇸🇪

Uppsala, Sweden

Kiev City Clinical Hospital No 5, Coronary Care Unit

🇺🇦

Kiev, Ukraine

City Clinical Hospital #8

🇺🇦

Kharkiv, Ukraine

Lugansk First Clinical Multiprofile Hospital #1, Cardiology

🇺🇦

Lugansk, Ukraine

N.D. Strazhesko Institute of Cardiology Intensive Care Unit

🇺🇦

Kiev, Ukraine

Lviv Reg St Clinical Treat-and-Diagn Cardio. Centre Dept of Myocardial Infarction

🇺🇦

Lviv, Ukraine

City Clinical Hospital #9 Dept of Arrhythmia

🇺🇦

Odessa, Ukraine

Royal Adelaide Hospital

🇦🇺

Adelaide, South Australia, Australia

Pärnu Hospital Department of Cardiology

🇪🇪

Parnu, Estonia

Carl-von Basedow-Klinikum Merseburg

🇩🇪

Merseburg, Germany

Kaunas Medical University Hospital - Department of Cardiology

🇱🇹

Kaunas, Lithuania

Medizinisches Versorgungszentrum Prof. Mathey, Prof. Schofer GmbH

🇩🇪

Hamburg, Germany

East Tallinn Central Hospital-Clinic of Cardiology

🇪🇪

Tallinn, Estonia

WCN - Department of Cardiology Rijnstate Ziekenhuls

🇳🇱

Arnhem, Netherlands

Campus Virchow-Klinikum, Charite - Universitaetsmedizin Berlin

🇩🇪

Berlin, Germany

Johann Wolfgang Goethe Universitaet Med Klinik III - Kardiologie

🇩🇪

Frankfurt, Germany

Klinikum der Stadt Ludwigshafen am Rhein gGmbH

🇩🇪

Ludwigshafen, Germany

Krankenhaus Reinbek, St. Adolf-Stift

🇩🇪

Reinbek, Germany

Groene Hart Zeikenhhaus

🇳🇱

Gouda, Netherlands

FN - I. interna klinika

🇸🇰

Nitra, Slovakia

Liva - Central Military Hospital

🇸🇰

Ruzomberok, Slovakia

Donetsk Regional Clinical Hospital

🇺🇦

Donetsk, Ukraine

Martin-Luther Universitat Halle, Med. Klinik und Poliklinik III- Fachrichtung Kardiologie

🇩🇪

Halle, Germany

Vilnius University Hospital Santariskiu Clinic - Center of Cardiology and Angiology

🇱🇹

Vilnius, Lithuania

Klinika Chorob Wewnetrznych z Oddzialem Farmakologii Klinicznej i Terapii Monitorowanej

🇵🇱

Lodz, Poland

Okregowy Szpital Kolejowy w Lublinie Samodzielny

🇵🇱

Lublin, Poland

Clinical Center of Serbia, Institute of CV Diseases

🇷🇸

Belgrade, Serbia

"Dedinje" Cardiovascular Institute

🇷🇸

Belgrade, Serbia

Klinikum der Universität Köln, Medizinische Klinik III

🇩🇪

Köln, Germany

Klinikum Pirna GmbH, Innere Medizin II, Kardiologie

🇩🇪

Pirna, Germany

Robert-Bosch-Krankenhaus, Abt. Kardiologie / Pulmologie

🇩🇪

Stuttgart, Germany

Internal Dep. Hospital Žilina

🇸🇰

Žilina, Slovakia

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