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Efficacy, Tolerability and Safety of LAS41004 Formulations in a Psoriasis Plaque Test

Phase 1
Completed
Conditions
Psoriasis
Interventions
Drug: LAS41004-IMP1
Drug: LAS41004 IMP2
Drug: LAS41004 IMP3
Drug: LAS41004 IMP4
Drug: LAS41004 IMP6
Drug: LAS41004 IMP5
Registration Number
NCT02111499
Lead Sponsor
Almirall, S.A.
Brief Summary

Clinical investigation of anti-psoriatic efficacy and atrophy

Detailed Description

In this trial three concentrations of bexarotene in combination with a fixed concentration of betamethasone dipropionate, as well as monotherapy with bexarotene, will be investigated regarding their efficacy, tolerability and safety in patients with mild to moderate plaque psoriasis and will be compared with the vehicle and an active comparator.

Since a side effect of the application of corticosteroids is skin atrophy, additionally three non-lesional test areas (not affected by psoriasis) on the volar forearm will be treated with the active reference product, one of the fixed combinations and the vehicle. Skin atrophy will be investigated by visual assessment and ultrasound at these test areas

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
18
Inclusion Criteria
  • 18 to 75 years of age

  • Men and women with skin type I to IV (Fitzpatrick 1974).

  • Suffering from mild to moderate plaque psoriasis of at least 6 months duration that is amenable to local therapy.

  • With at least one stable psoriatic plaque in an area sufficient for product application meeting the following criteria:

    • Located at the trunk and/or the extremities (plaques located on the head, palms, or soles of the feet, intertriginous or genitoanal areas are not suitable).
    • Plaques with a clinical score of the parameter erythema and or induration of ≥ 2 for each sign at the screening visit. At Day 1 each parameter has to be scored ≥ 2.
    • Where more than one plaque is to be used, plaques should be comparable, with at least "2" in each score for erythema and induration.
    • • Body surface area (BSA) involvement < 10 %.
  • Prepared to give written informed consent specific to the trial, before any assessment is performed.

  • • In the case of women of childbearing potential using reliable methods of contraception which result in a low failure rate i.e. less than 1% per year (e.g. contraceptive implants or injectables, combined oral contraceptives, some intrauterine devices, sexual abstinence or vasectomized partner). During the study an additional barrier method (e.g. condoms) should be used. Non-childbearing potential is defined as surgical sterilization (hysterectomy, ovariectomy or tubal ligation), postmenopausal status (continuous amenorrhea of at least 2 years).

  • In the case of men with partners of childbearing potential willingness of using condoms during the study conduct and 1 month after end of treatment.

Main

Exclusion Criteria
  • • Patients who need systemic treatment for their psoriasis.

    • Severe forms of psoriasis or forms of psoriasis other than chronic plaque psoriasis,
    • Systemic treatment (see table below):

Corticosteroids, antibiotics 4 weeks prior to trial Day 1 and during conduct of trial Retinoids Ciclosporin Methotrexate Fumaric acid esters 3 months prior to trial Day 1 and during conduct of trial Anti-inflammatory substances, NSAIDs 2 weeks prior to trial Day 1 and during conduct of trial Biologics 6 months prior to trial Day 1 and during conduct of trial

  • Topical treatment of all other body regions with corticosteroids or immunosuppressants where more than 20 % of the body surface area is treated.
  • Diseases:

Significant skin infections caused by bacteria, viruses or fungi, including but not limited to tuberculosis, syphilis or varicella zoster infection Parasitic infections

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
formulation 2LAS41004 IMP3topical treatment, once daily for 4 weeks
formulation 2LAS41004 IMP4topical treatment, once daily for 4 weeks
formulation 1LAS41004-IMP1topical treatment, once daily for 4 weeks
formulation 1LAS41004 IMP2topical treatment, once daily for 4 weeks
formulation 1LAS41004 IMP3topical treatment, once daily for 4 weeks
formulation 1LAS41004 IMP4topical treatment, once daily for 4 weeks
formulation 1LAS41004 IMP6topical treatment, once daily for 4 weeks
formulation 1LAS41004 IMP5topical treatment, once daily for 4 weeks
formulation 2LAS41004-IMP1topical treatment, once daily for 4 weeks
formulation 2LAS41004 IMP2topical treatment, once daily for 4 weeks
formulation 2LAS41004 IMP6topical treatment, once daily for 4 weeks
formulation 3LAS41004 IMP3topical treatment, once daily for 4 weeks
formulation 3LAS41004 IMP4topical treatment, once daily for 4 weeks
formulation 2LAS41004 IMP5topical treatment, once daily for 4 weeks
formulation 3LAS41004-IMP1topical treatment, once daily for 4 weeks
formulation 3LAS41004 IMP2topical treatment, once daily for 4 weeks
formulation 3LAS41004 IMP6topical treatment, once daily for 4 weeks
formulation 3LAS41004 IMP5topical treatment, once daily for 4 weeks
formulation 4LAS41004-IMP1topical treatment,once daily for 4 weeks
formulation 4LAS41004 IMP2topical treatment,once daily for 4 weeks
formulation 4LAS41004 IMP3topical treatment,once daily for 4 weeks
formulation 4LAS41004 IMP4topical treatment,once daily for 4 weeks
formulation 4LAS41004 IMP6topical treatment,once daily for 4 weeks
formulation 4LAS41004 IMP5topical treatment,once daily for 4 weeks
formulation 5LAS41004 IMP5topical treatment, once daily for 4 weeks
formulation 5LAS41004-IMP1topical treatment, once daily for 4 weeks
formulation 5LAS41004 IMP2topical treatment, once daily for 4 weeks
formulation 5LAS41004 IMP3topical treatment, once daily for 4 weeks
formulation 5LAS41004 IMP4topical treatment, once daily for 4 weeks
formulation 5LAS41004 IMP6topical treatment, once daily for 4 weeks
formulation 6LAS41004-IMP1topical treatment, once daily for 4 weeks
formulation 6LAS41004 IMP2topical treatment, once daily for 4 weeks
formulation 6LAS41004 IMP3topical treatment, once daily for 4 weeks
formulation 6LAS41004 IMP4topical treatment, once daily for 4 weeks
formulation 6LAS41004 IMP6topical treatment, once daily for 4 weeks
formulation 6LAS41004 IMP5topical treatment, once daily for 4 weeks
Primary Outcome Measures
NameTimeMethod
Area under the curve, AUC, of the width of the echo-lucent band based on sonography measurementsday 1 vs day 29

The primary objective is to gain evidence suggesting efficacy of the investigational products in the treatment of plaque-type psoriasis as assessed by the AUC of the width of the echo-lucent band

Secondary Outcome Measures
NameTimeMethod
erythema and indurationday 1 vs day 29

investigation of the individual scores for erythema and induration

local skin tolerabilityevery day for 28 days

Safety investigation of tolerability parameters assessed by a dermatologist

atrophyday1 vs day 29

investigation of skin atrophy assessments on non-lesional test areas

assessment of (serious) Adverse Eventsfrom baseline to day 29

Daily record will be performed and - if needed - causality and severity assessed

Trial Locations

Locations (1)

proDERM GmbH

🇩🇪

Schenefeld, Schleswig-Holstein, Germany

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