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A Study Evaluating the Safety and Efficacy of Inhaled AP01 in Participants With Progressive Pulmonary Fibrosis

Phase 2
Recruiting
Conditions
Progressive Pulmonary Fibrosis
Interventions
Other: Placebo
Registration Number
NCT06329401
Lead Sponsor
Avalyn Pharma Inc.
Brief Summary

A randomized, double-blind, placebo-controlled clinical study to evaluate the safety and efficacy of 2 doses of inhaled pirfenidone (AP01) versus placebo on top of standard of care in participants with PPF over 52 weeks.

Detailed Description

This is a randomized, double-blind, placebo-controlled clinical study to evaluate the safety and efficacy of 2 doses of AP01 (pirfenidone solution for inhalation) versus placebo on top of standard of care in participants with PPF over 52 weeks. Up to 300 eligible participants will be randomized to 1 of 3 treatment arms: AP01 high dose, AP01 low dose, or placebo.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
300
Inclusion Criteria
  • Participant meets criteria for PPF, as follows:
  • In participants with ILD of known or unknown etiology other than IPF who have radiological evidence of pulmonary fibrosis, PPF is defined as:

I. Physiological evidence of disease progression:

a. Absolute decline in FVC ≥5% predicted within the previous 6 to 12 months relative to Screening Visit 1

And at least 1 of the following 2 criteria occurring within the past year with no alternative explanation:

II. Worsening respiratory symptoms (Note: Changes attributable to comorbidities e.g., infection, heart failure must be excluded)

III. Radiological evidence of disease progression (one or more of the following):

a. Increased extent or severity of traction bronchiectasis and bronchiolectasis b. New ground-glass opacity with traction bronchiectasis c. New fine reticulation d. Increased extent or increased coarseness of reticular abnormality e. New or increased honeycombing f. Increased lobar volume loss

  • Meeting all of the following criteria during the Screening Period:

    1. FVC ≥45% of predicted normal at Screening Visit 1,
    2. Forced expiratory volume at 1 second (FEV1)/FVC ≥0.7 at Screening Visit 1,
    3. Diffusing capacity of lung for carbon monoxide (DLCO) ≥30% of predicted, corrected for hemoglobin at Screening Visit 1,
    4. Acceptability: Participants can perform acceptable spirometry (i.e., meet American Thoracic Society (ATS)/ European Respiratory Society (ERS) acceptability criteria at both Screening Visits).
  • For participants already on nintedanib (up to 30% of participants): Must have been on nintedanib for 6 to 12 months prior to Screening and have met criteria for PPF while on nintedanib for the same period in which the ≥5% decline in FVC was observed. Must have had no change in nintedanib dose for at least 12 weeks prior to Screening. For participants who have discontinued nintedanib prior to Screening: Must have been off of nintedanib for a minimum of 12 weeks.

Exclusion Criteria
  • Current treatment with oral pirfenidone or treatment with oral pirfenidone within 3 months prior to Screening.

  • Elevated liver enzymes and liver injury at Screening defined as:

    1. Alanine aminotransferase (ALT) or aspartate aminotransferase (AST) ˃ 3 times the upper limit of normal (ULN)
    2. Bilirubin > 1.5 x ULN
  • Renal disease with a creatinine clearance < 30 mL/min, calculated according to the Chronic Kidney Disease Epidemiology Collaboration formula. Retesting is allowed once.

  • Diagnosis of idiopathic pulmonary fibrosis (IPF) based on the ATS diagnostic algorithm for IPF. UIP that is not idiopathic, for example related to rheumatoid arthritis (RA), familial interstitial lung disease (ILD), or other is not exclusionary.

  • Greater extent of emphysema than of fibrotic ILD on HRCT. Note: CT results must be confirmed through the central over read process.

  • Significant clinical worsening of PPF between Screening

  • Participants who cannot meet protocol-specified Baseline stability criteria. FVC Baseline stability is defined as the FVC assessments at Visit 3 being within ±12% of the mean of the FVC assessments obtained at the 2 preceding visits. At Visit 3, if the pre-dose FVC is outside of ±12% range, the participant will not be randomized and will be considered a screen failure.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Placebo BIDPlaceboPlacebo solution for inhalation
AP01 High Dose BIDAP01Pirfenidone Solution for Inhalation
AP01 Low Dose BIDAP01Pirfenidone Solution for Inhalation
Primary Outcome Measures
NameTimeMethod
To evaluate the effect of AP01 high dose twice a day (BID) or AP01 low dose twice a day (BID) compared to placebo twice a day (BID)Week 52

Change from baseline in forced vital capacity (FVC) (mL)

Secondary Outcome Measures
NameTimeMethod
To evaluate the effect of AP01 high dose, AP01 low dose compared to placebo on quality of life (QoL)52 weeks

Absolute change from Baseline in QoL measurements as assessed by Living with Pulmonary Fibrosis Symptoms and Impact Questionnaire (L-PF) total score. The L-PF is a 44-item questionnaire to assess how impacted a participant is by disease symptoms on a scale from 0 (Not at all) to 4 (Extremely). The higher the summary score, the greater the impairment.

To evaluate the change from baseline in quantitative lung fibrosis score.52 weeks

Change in lung fibrosis score.

To evaluate the effect of AP01 high dose and AP01 low dose compared to placebo on disease progression (defined as absolute FVC percent predicted decline of ≥10% prior to Week 52)52 weeks

Time to disease progression

Trial Locations

Locations (118)

Instituto de Medicina Respiratoria

🇦🇷

Córdoba, Argentina

CIMER Centro Integral de Medicina Respiratoria

🇦🇷

Tucumán, Argentina

Investigaciones En Patologias Respiratorias

🇦🇷

Tucumán, Argentina

Nepean Lung & Sleep

🇦🇺

Kingswood, New South Wales, Australia

Dynamic Drug Advancement

🇨🇦

Ajax, Ontario, Canada

CIC Mauricie

🇨🇦

Trois-Rivières, Quebec, Canada

CHU de Rennes

🇫🇷

Rennes, Cedex NA, France

CHU Tours

🇫🇷

Tours, Indre et Loire, France

Robert Schuman Hospital UNEOS

🇫🇷

Metz, Lorraine, France

CHU Angers

🇫🇷

Angers, France

Louis Pradel Hospital

🇫🇷

Lyon, France

University of Montpellier

🇫🇷

Montpellier, France

Hôpital Haut-Lévêque

🇫🇷

Pessac, France

RoMed Klinikum Rosenheim

🇩🇪

Rosenheim, Bavaria, Germany

A.O.U. delle Marche - Ospedale di Torrette

🇮🇹

Torrette, Ancona, Italy

A.O.U. Policlinico G. Rodolico

🇮🇹

Catania, Sicilia, Italy

Ospedale San Giuseppe

🇮🇹

Milano, Italy

SEC Clinical Research

🇺🇸

Pensacola, Florida, United States

University of Alabama at Birmingham

🇺🇸

Birmingham, Alabama, United States

Pulmonary Associates, PA

🇺🇸

Phoenix, Arizona, United States

University of Southern California

🇺🇸

Los Angeles, California, United States

Cedars-Sinai

🇺🇸

Los Angeles, California, United States

UCLA

🇺🇸

Los Angeles, California, United States

Newport Native MD, Inc.

🇺🇸

Newport Beach, California, United States

Paradigm Clinical Research - Redding

🇺🇸

Redding, California, United States

University of Colorado, Anschutz Medical Campus

🇺🇸

Aurora, Colorado, United States

National Jewish Health

🇺🇸

Denver, Colorado, United States

UCONN Health

🇺🇸

Farmington, Connecticut, United States

Yale University

🇺🇸

New Haven, Connecticut, United States

Clinical Site Partners, LCC

🇺🇸

Leesburg, Florida, United States

Renstar Medical Research

🇺🇸

Ocala, Florida, United States

Central Florida Pulmonary Group

🇺🇸

Orlando, Florida, United States

Clinical Site Partners

🇺🇸

Winter Park, Florida, United States

Piedmont Healthcare, Inc.

🇺🇸

Atlanta, Georgia, United States

Northwestern University

🇺🇸

Chicago, Illinois, United States

Endeavor Health

🇺🇸

Evanston, Illinois, United States

Loyola University Medical Center

🇺🇸

Maywood, Illinois, United States

The University of Kansas Medical Center

🇺🇸

Kansas City, Kansas, United States

University of Maryland

🇺🇸

Baltimore, Maryland, United States

Johns Hopkins University

🇺🇸

Baltimore, Maryland, United States

Beth Israel Deaconess Medical Center

🇺🇸

Boston, Massachusetts, United States

University of Michigan

🇺🇸

Ann Arbor, Michigan, United States

University of Minnesota

🇺🇸

Minneapolis, Minnesota, United States

Mayo Clinic Rochester

🇺🇸

Rochester, Minnesota, United States

Hannibal Regional Healthcare System

🇺🇸

Hannibal, Missouri, United States

Montefiore Medical Center

🇺🇸

Bronx, New York, United States

Northwell Health - Mount Kisco

🇺🇸

Mount Kisco, New York, United States

NYU Langone Health

🇺🇸

New York, New York, United States

Weill Cornell

🇺🇸

New York, New York, United States

Icahn School of Medicine at Mount Sinai

🇺🇸

New York, New York, United States

Columbia University

🇺🇸

New York, New York, United States

Duke University

🇺🇸

Durham, North Carolina, United States

Pulmonix

🇺🇸

Greensboro, North Carolina, United States

Piedmont HealthCare, PA

🇺🇸

Statesville, North Carolina, United States

Accellacare

🇺🇸

Wilmington, North Carolina, United States

Southeastern Research Center

🇺🇸

Winston-Salem, North Carolina, United States

University of Cincinnati

🇺🇸

Cincinnati, Ohio, United States

Summit Health

🇺🇸

Bend, Oregon, United States

The Oregon Clinic Pulmonary East

🇺🇸

Portland, Oregon, United States

The Oregon Clinic Pulmonary West

🇺🇸

Portland, Oregon, United States

The Pennsylvania State University

🇺🇸

Hershey, Pennsylvania, United States

Thomas Jefferson University

🇺🇸

Philadelphia, Pennsylvania, United States

Temple University

🇺🇸

Philadelphia, Pennsylvania, United States

Lowcountry Lung and Critical Care

🇺🇸

Charleston, South Carolina, United States

Medical University of South Carolina

🇺🇸

Charleston, South Carolina, United States

Clinical Trials Center of Middle Tennessee

🇺🇸

Franklin, Tennessee, United States

Vanderbilt Lung Institute

🇺🇸

Nashville, Tennessee, United States

Baylor Scott & White Research Institute, Baylor University Medical Center

🇺🇸

Dallas, Texas, United States

El Paso Pulmonary Association

🇺🇸

El Paso, Texas, United States

Baylor College of Medicine

🇺🇸

Houston, Texas, United States

The University of Texas Health Science Center

🇺🇸

Houston, Texas, United States

Metroplex Pulmonary and Sleep Center, PA

🇺🇸

McKinney, Texas, United States

Intermountain Medical Center

🇺🇸

Murray, Utah, United States

University of Utah Health

🇺🇸

Salt Lake City, Utah, United States

Inova Healthcare

🇺🇸

Falls Church, Virginia, United States

University of Washington

🇺🇸

Seattle, Washington, United States

Fundacion Respirar

🇦🇷

Buenos Aires, Argentina

CINME

🇦🇷

Buenos Aires, Argentina

Royal Prince Alfred Hospital

🇦🇺

Camperdown, New South Wales, Australia

John Hunter Hospital

🇦🇺

New Lambton, New South Wales, Australia

Macquarie University Clinical Trials Unit

🇦🇺

Sydney, New South Wales, Australia

Westmead Hospital

🇦🇺

Westmead, New South Wales, Australia

Institute for Respiratory Health

🇦🇺

Nedlands, Perth West Australia, Australia

Lung Research Victoria

🇦🇺

Footscray, Victoria, Australia

Alfred Health

🇦🇺

Melbourne, Victoria, Australia

Vancouver General Hospital

🇨🇦

Vancouver, British Columbia, Canada

St. Joseph's Healthcare Hamilton

🇨🇦

Hamilton, Ontario, Canada

Research Institute McGill University Health Center

🇨🇦

Montreal, Quebec, Canada

Institut universitaire de cardiologie et de pneumologie de Québec-Université Laval

🇨🇦

Québec, Quebec, Canada

Pneumologisches Studienzentrum München-West

🇩🇪

Muenchen, Bavaria, Germany

Medizinische Hochschule Hannover

🇩🇪

Hannover, Lower Saxony, Germany

Studienzentrum Dr. Claus Keller

🇩🇪

Frankfurt, Main Hessia, Germany

Ruhrlandklinik Essen, Klinik fuer Pneumologie

🇩🇪

Essen, Northrhine westphalia, Germany

Universitätsmedizin Mainz - Zentrum für Thoraxerkrankungen

🇩🇪

Mainz, Rhineland-Palatinate, Germany

Uniklinikum Leipzig Medizinische Klinik II - Bereich

🇩🇪

Leipzig, Saxony, Germany

Azienda Sanitaria Universitaria Giuliano Isontina

🇮🇹

Venezia, Giulia, Italy

Fondazione IRCCS Policlinico San Matteo - UOC Pneumologia

🇮🇹

Pavia, Lombardia, Italy

HUMANITAS Research Hospital

🇮🇹

Rozzano, Milano, Italy

IRCCS AOU di Bologna - Policlinico Sant' Orsola

🇮🇹

Bologna, Romagna, Italy

Health New Zealand

🇳🇿

Christchurch, Canterbury, New Zealand

Dunedin Hospital

🇳🇿

Dunedin, Dunedine, New Zealand

Bay of Plenty Clinical School

🇳🇿

Tauranga, South Tauranga, New Zealand

Greenlane Clinical Centre

🇳🇿

Auckland, New Zealand

Vitamed Galaj I Cichomski sp.j.

🇵🇱

Bydgoszcz, Bydgoszc, Poland

AppleTreeClinics Network

🇵🇱

Lodz, Poland

Hospital Universitario Virgen de las Nieves

🇪🇸

Granada, Andalucía, Spain

Hospital Universitario Central de Asturias

🇪🇸

Oviedo, Asturias, Spain

Hospital de Sant Pau y la Santa Creu

🇪🇸

Barcelona, Spain

Hospital Universitario Puerta del Mar - Leon-Jimenez

🇪🇸

Cadiz, Spain

Hospital Gregorio Marañon

🇪🇸

Madrid, Spain

Hospital Universitario Virgen de la Victoria

🇪🇸

Málaga, Spain

Ege University Medical Faculty Hospital

🇹🇷

Bornova, Izmir, Turkey

Hull University Teaching Hospital NHS Trust

🇬🇧

Cottingham, East Yorkshire, United Kingdom

Leicester Biomedical Research Centre - Respiratory Theme

🇬🇧

Glenfield, Leicester, United Kingdom

Royal Devon

🇬🇧

Exeter, South West, United Kingdom

The Royal Wolverhampton NHS Trust, New Cross Hospital, Research and Development

🇬🇧

Wolverhampton, West Midlands, United Kingdom

St James University Hospital - LTHT

🇬🇧

Leeds, West Yorkshire, United Kingdom

St George's University Hospitals NHS Foundation Trust

🇬🇧

London, United Kingdom

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