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Eltrombopag in Second Line Adult Primary Immune Thrombosytopenia

Phase 2
Completed
Conditions
Primacy Immune Thrombocytopenia
Interventions
Registration Number
NCT02402998
Lead Sponsor
Gruppo Italiano Malattie EMatologiche dell'Adulto
Brief Summary

A clinical study to evaluate the efficacy of a drug called eltrombopag in adult patients affected of primary immune thrombocytopenia as first treatment to address the disease.

Detailed Description

This is a prospective, multicenter phase II trial designed to evaluate the activity of Eltrombopag second line treatment in adult patients with primary Immune Thrombocytopenia (ITP) not responsive or in relapse after a full first line steroids treatment (prednisone or dexamethasone) ± Intravenous Immune Globulin (IVIG).

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
55
Inclusion Criteria
  1. Diagnosis of primary ITP;
  2. Age ≥ 18 years;
  3. Patients are in the new diagnosis or persistent phase of disease (i.e. within month 12 from diagnosis);
  4. Patients not responsive or in relapse after a full course of steroid therapy (prednisone 1 mg/kg/d for at least 28 days or 3 cycles of dexamethasone 40 mg/day for consecutive 4 days, according to the GIMEMA ITP0207 trial) ± IVIG;
  5. Patients have a platelet count < 10 x 109/L documented in a single blood cell count;
  6. Patients have bleeding symptoms and a platelet count > 10 < 30 x 109/L documented in a single blood cell count;
  7. Patients have no bleeding symptoms and a platelet count >10 < 30 x 109/L in at least 2 blood cell counts at 3 days interval in the week preceding the enrollment with the last count at the day of enrollment;
  8. Patients have corticosteroids or IVIG dependence (the need for ongoing or repeated doses administration of corticosteroids or IVIG to maintain a platelet count ≥ 30 x 109/L and/or to avoid bleeding;
  9. Written informed consent obtained from the subject;
  10. Men with a female partner of childbearing potential must have either had a prior vasectomy or agree to use effective contraception from time of enrollment until 6 months after the last dose of study treatment;
  11. Female subjects of non-childbearing potential may be enrolled in the study; for this study population, non-childbearing potential is defined as current tubal ligation, hysterectomy, ovariectomy or post-menopause; OR
  12. Female subjects of childbearing potential may be enrolled in the study, if the subject has practiced adequate contraception for 30 days prior to start of Eltrombopag, has a negative pregnancy test within 14 days of first dose of Eltrombopag, and has agreed to continue adequate contraception during the entire treatment period and for 6 months after completion of the treatment.
Exclusion Criteria
  1. Diagnosis of secondary ITP. As far as patients with immune thrombocytopenia and antiphospholipid antibodies positivity, individuals without a previous thromboembolic event are excluded only if lupus anticoagulant (LAC) is associated with the presence of anticardiolipin (aCL) and aβ2-Glycoprotein I (aβ2GPI) antibodies;

  2. Previous treatment with other anti-ITP second line therapies (i.e. Rituximab, Azathioprine, Cyclosporin-A or other); only patients with a previous full course of steroid (see inclusion criteria for definition) ± IVIG are admitted to the study;

  3. Previous treatment with any TPO-R agonists;

  4. Patients have life threatening bleeding complications;

  5. Patients had deep venous thrombosis (DVT) or arterial thrombosis in the 3 months preceding the enrollment;

  6. Patients are HIV, HCV, HBsAg positive;

  7. Patients with hepatic impairment (i.e. mild, moderate or severe hepatic impairment (Child-Pugh score > 6);

  8. Patients have a well established liver disease that represents a contraindication for the use of Eltrombopag;

  9. Patients are unable to respect the 4-hour interval between Eltrombopag and other medications (e.g. antacids), calcium-rich foods (e.g. dairy products and calcium fortified juices), or supplements containing polyvalent cations such as iron, calcium, aluminium, magnesium, selenium, and zinc;

  10. Patients are unable to stop medications that are known to cause a drug-drug interaction with Eltrombopag;

  11. Subjects meeting any of the following criteria must not be enrolled in an Eltrombopag study:

    • Lactating female.
    • History of another malignancy. Exception: subjects who have been disease-free for 5 years, or subjects with a history of completely resected non-melanoma skin cancer or successfully treated in situ carcinoma are eligible.
    • Any serious and/or unstable pre-existing medical, psychiatric disorder, or other conditions that could interfere with subject's safety, obtaining informed consent or compliance with the study procedures.
    • Hormone replacement therapy. Subjects must discontinue hormone replacement therapy prior to study enrollment due to the potential for inhibition of Cytochrome P450 (CYP) enzymes that metabolize estrogens and progestins.
    • Administration of an investigational drug within 30 days or 5 half-lives, whichever is longer, preceding the first dose of study treatment.
    • Have a known immediate or delayed hypersensitivity reaction or idiosyncrasy to drugs chemically related to Eltrombopag or excipients that contraindicate their participation.

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
EltrombopagEltrombopagEltrombopag 50 mg/daily.
Primary Outcome Measures
NameTimeMethod
Number of subjects who achieve long-term response (6 months sustained response) and able to taper down the dose.After one year from study treatment.

A patient will achieve this endpoint if at the end of the period of treatment he/she reaches to discontinue Eltrombopag and if, after discontinuation, has absence of bleeding and maintains a platelet count ≥ 30 x 109/L and at least a 2-fold increase from the baseline count in blood cell count performed in the 6 months of the period observation, during which no steroid, Eltrombopag, other anti TPO-R agonists and other anti-ITP medications are administered.

Secondary Outcome Measures
NameTimeMethod
Number of bleeding events.After one year from study treatment.
Number of months of response from eltrombopag discontinuation to the last follow-up.After one year from study treatment.
Number of months of complete response from eltrombopag discontinuation to the last follow-up.After one year from study treatment.

Trial Locations

Locations (14)

Fondazione IRCCS Ca' Granda Ospedale Maggiore Policlinico UOC Oncoematologia- Padiglione Marcora 2° piano

🇮🇹

Milano, Italy

Ospedale Niguarda " Ca Granda" - SC Ematologia Blocco SUD, Ponti Est, Scala E, 4° piano

🇮🇹

Milano, Italy

Università degli Studi "Sapienza" - Dip Biotecnologie Cellulari ed Ematologia - Divisione di Ematologia

🇮🇹

Roma, Italy

AO di Padova Università degli Studi Padova Dipartimento di Medicina Clinica Medica I - Medicina Interna CLOPD

🇮🇹

Padova, Italy

Università degli Studi di Verona - A. O. - Istituti Ospitalieri di Verona- Div. di Ematologia - Policlinico G.B. Rossi

🇮🇹

Verona, Italy

Azienda Ospedaliera Di Bologna Policlinico S. Orsola - Malpighi

🇮🇹

Bologna, Italy

Azienda Ospedaliera "S.Gerardo"

🇮🇹

Monza, Italy

S.C.D.U. Ematologia - DIMECS e Dipartimento Oncologico - Università del Piemonte Orientale Amedeo Avogadro

🇮🇹

Novara, Italy

Azienda Ospedale S. Luigi at University of Torino

🇮🇹

Orbassano, Italy

Ospedale "Infermi"

🇮🇹

Rimini, Italy

Policlinico A. Gemelli - Universita Cattolica del Sacro Cuore

🇮🇹

Rome, Italy

Azienda Ospedaliera di Rilievo Nazionale "A. Cardarelli"

🇮🇹

Napoli, Italy

Ospedale San Bortolo

🇮🇹

Vicenza, Italy

Clinica Ematologica-Centro Trapianti e Terapie cellulari Azienda Ospedaliero-Universitaria, Udine

🇮🇹

Udine, Italy

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