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Efficacy and Safety of Silodosin in the Treatment of Natural Expulsion in Patients With Ureteral Stones

Phase 4
Completed
Conditions
Ureteral Stone
Interventions
Drug: Placebo
Registration Number
NCT01533389
Lead Sponsor
JW Pharmaceutical
Brief Summary

A lower ureteral calculus, which measures 5 millimeters and less, may be easily expelled by symptomatic therapy. Actually, it has about a 50% chance of successful expulsion.

However, a complication such as urinary tract infection or hydronephrosis or persistent pain may occur before it is expelled. Thus, it is imperative to minimize the occurrence of complications in the process of expectant treatment and also to reduce the time required to expel calculi.

Pharmacotherapy is to relieve ureteral obstruction and thus to expel urinary calculi easily.

This clinical trial is to evaluate the efficacy of silodosin, a selective α1A-blocker, on calculous expulsion in expectant treatment for patients with lower and mid ureteral calculi.

Detailed Description

Lower and mid ureteral calculi, accounting for approximately 70% of ureteral calculi, has a high chance of successful treatment thanks to ureteroscopic lithotripsy or extracorporeal shock wave lithotripsy (ESWL)1-3), but at the same time have problems of postprocedural complications and high expenses4). A lower ureteral calculus, which measures 5 millimeters and less, may be easily expelled by symptomatic therapy. Actually, it has about a 50% chance of successful expulsion5). However, a complication such as urinary tract infection or hydronephrosis or persistent pain may occur before it is expelled. Thus, it is imperative to minimize the occurrence of complications in the process of expectant treatment and also to reduce the time required to expel calculi.

It has been recently reported that pharmacotherapy is adhibited to the expulsion of urinary calculi and the relief of pain. The migration of ureteral calculi is influenced by both the calculus and the ureter. In the case of the calculus, size, shape, number and location influence it. In regard to the ureter, it is significantly influenced by the cramp of the ureteral smooth muscle, the edema of the ureteral submucosa, the pain caused by the calculus and the activities of adrenoreceptors6).

Pharmacotherapy is to relieve ureteral obstruction and thus to expel urinary calculi easily. Ureteral obstruction, caused by urinary calculi, obtunds ureteral peristalsis but strengthens ureteral contraction, which may cause urinary retention or regurgitation7-8). In this connection, studies have been conducted as to methods to reduce abnormal urinary reaction caused by urinary calculi and to smoothen uroflow. Currently, hormone drugs including hydroxyprogesterone, prostaglandin synthetase inhibitors, calcium-channel antagonists, α1-blockers and steroid drugs are used to expel urinary calculi and to suppress pain. The guidelines on urinary calculi, drawn up in 2007, recommend using α-blockers as they are superior to other drugs in efficacy9-12).

The drug to be used in this clinical trial, silodosin, was registered under the proprietary name of 'THRUPAS® Capsule 4mg' and is being marketed after being authorized by Korea Food and Drug Administration (FDA), which selectively acts on the α1A-adrenoreceptor.

This clinical trial is to evaluate the efficacy of silodosin, a selective α1A-blocker, on calculous expulsion in expectant treatment for patients with lower and mid ureteral calculi.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
114
Inclusion Criteria
  • Males or female patients aged 20 and over
  • Patients having ureteral calculi located mid or lower ureter on abdominal radiograms or excretory urograms or non-enhanced computed tomograms.
  • Patients whose calculi measure 10 millimeters and less.
  • Patients who voluntarily decided to take part in this clinical trial and gave written consent.
Exclusion Criteria
  • Patients who do not want to undergo expectant treatment
  • Female patients who are pregnant or nursing
  • Patients with febrile urinary tract infection or severe hydronephrosis or ulcerative diseases or hypotension.
  • Patients with severe hepatic dysfunction(e.g. hepatic failure, hepatic cirrhosis, icterus, hepatoma)
  • Patients who take α-blocker or α/β-blockers or calcium-channel blockers or steroid drugs
  • Patients with multiple ureteral calculi
  • Patients whose urinary tracts are anatomically deformed or stenosed
  • Patients who underwent invasive operations on their ureters before
  • Patients whose blood creatinine levels are 2mg/dL and over
  • Patients who are hypersensitive to silodosin
  • Patients who take part in clinical trials other than this one
  • Patients judged to be inappropriate for this clinical trial by investigators

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
PlaceboPlacebo8mg QD
SilodosinSilodosin8mg QD
Primary Outcome Measures
NameTimeMethod
Expulsion rate of stones4 weeks

1 week, 2 weeks, 4 weeks to visit and inspected. (Last visit four weeks) Results when the exhaust is used.

Secondary Outcome Measures
NameTimeMethod
Stone expulsion timeevery 1 week or 2 weeks
Migration distance of stoneevery 1 week or 2 weeks
Frequency of administration of oral or injectable analgesicsevery 1 week or 2 weeks
Number of cases where subjects visited ER due to uncontrolled painsevery 1 week or 2 weeks

Trial Locations

Locations (5)

Kangbuk Samsung Medical Center

🇰🇷

Seoul, Korea, Republic of

Eulji General Hospital

🇰🇷

Seoul, Korea, Republic of

NHIC Ilsan Hospital

🇰🇷

Goyang-Si, Gyonggi-Do, Korea, Republic of

Inje Univ. Sanggye Paik Hospital

🇰🇷

Seoul, Korea, Republic of

Myongji Hospital

🇰🇷

Goyang-Si, Gyonggi-Do, Korea, Republic of

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